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Found 742 Enz. Inhib. hit(s) with Target = 'M1 family aminopeptidase'
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497543(CHEMBL3359693)
Affinity DataKi:  0.700nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497544(CHEMBL3359688)
Affinity DataKi:  0.800nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497553(CHEMBL3359696)
Affinity DataKi:  1.90nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497545(CHEMBL3359697)
Affinity DataKi:  4nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497556(CHEMBL3359699)
Affinity DataKi:  5.5nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497551(CHEMBL3359700)
Affinity DataKi:  7.40nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497552(CHEMBL3359698)
Affinity DataKi:  11nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497557(CHEMBL3359692)
Affinity DataKi:  12nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497547(CHEMBL3359694)
Affinity DataKi:  15nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497546(CHEMBL3359695)
Affinity DataKi:  23nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497548(CHEMBL3359691)
Affinity DataKi:  41nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50339789((S)-2-((2S,3R)-3-amino-2-hydroxy-4-(4-methoxypheny...)
Affinity DataKi:  43nMAssay Description:Inhibition of Plasmodium falciparum recombinant M1-aminopeptidase expressed in Escherichia coli after 40 mins uisng fluorigenic substrate L-Leucyl-7-...More data for this Ligand-Target Pair
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497554(CHEMBL3359689)
Affinity DataKi:  75nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497549(CHEMBL3359690)
Affinity DataKi:  113nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM23971((2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanami...)
Affinity DataKi:  190nMAssay Description:Inhibition of Plasmodium falciparum recombinant M1-aminopeptidase expressed in Escherichia coli after 40 mins uisng fluorigenic substrate L-Leucyl-7-...More data for this Ligand-Target Pair
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50339790((S)-2-((2S,3R)-3-amino-4-(4-(benzyloxy)phenyl)-2-h...)
Affinity DataKi:  490nMAssay Description:Inhibition of Plasmodium falciparum recombinant M1-aminopeptidase expressed in Escherichia coli after 40 mins uisng fluorigenic substrate L-Leucyl-7-...More data for this Ligand-Target Pair
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497555(CHEMBL3359686)
Affinity DataKi: >500nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50497550(CHEMBL3359687)
Affinity DataKi: >500nMAssay Description:Inhibition of Plasmodium falciparum M1 incubated for 10 mins before H-Leu-NHMec substrate addition by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50339784((S)-2-((2S,3R)-3-amino-2-hydroxy-4-phenylbutanamid...)
Affinity DataKi:  900nMAssay Description:Inhibition of Plasmodium falciparum recombinant M1-aminopeptidase expressed in Escherichia coli after 40 mins uisng fluorigenic substrate L-Leucyl-7-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50339785((S)-2-((2S,3R)-3-amino-2-hydroxy-4-phenylbutanamid...)
Affinity DataKi:  1.45E+3nMAssay Description:Inhibition of Plasmodium falciparum recombinant M1-aminopeptidase expressed in Escherichia coli after 40 mins uisng fluorigenic substrate L-Leucyl-7-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50339791((S)-2-((2S,3R)-3-amino-2-hydroxy-4-(naphthalen-2-y...)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of Plasmodium falciparum recombinant M1-aminopeptidase expressed in Escherichia coli after 40 mins uisng fluorigenic substrate L-Leucyl-7-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50339792((S)-2-((2S,3R)-3-amino-2-hydroxyheptanamido)-4-met...)
Affinity DataKi:  5.30E+3nMAssay Description:Inhibition of Plasmodium falciparum recombinant M1-aminopeptidase expressed in Escherichia coli after 40 mins uisng fluorigenic substrate L-Leucyl-7-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50339786((S)-2-((2S,3R)-3-amino-2-hydroxy-4-phenylbutanamid...)
Affinity DataKi: >1.50E+4nMAssay Description:Inhibition of Plasmodium falciparum recombinant M1-aminopeptidase expressed in Escherichia coli after 40 mins uisng fluorigenic substrate L-Leucyl-7-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50339787((S)-2-((2S,3R)-3-amino-2-hydroxy-4-phenylbutanamid...)
Affinity DataKi: >1.50E+4nMAssay Description:Inhibition of Plasmodium falciparum recombinant M1-aminopeptidase expressed in Escherichia coli after 40 mins uisng fluorigenic substrate L-Leucyl-7-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50339788((S)-2-((2S,3R)-3-amino-2-hydroxy-4-phenylbutanamid...)
Affinity DataKi: >1.50E+4nMAssay Description:Inhibition of Plasmodium falciparum recombinant M1-aminopeptidase expressed in Escherichia coli after 40 mins uisng fluorigenic substrate L-Leucyl-7-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50206554(CHEMBL219777 | N-(4-fluoro-benzyl)-N'-hydroxy-2-[1...)
Affinity DataIC50:  6nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50206558(CHEMBL375521 | N-hydroxy-N'-(4-phenyl-butyl)-2-[1-...)
Affinity DataIC50:  13nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50206550(2-benzyl-N-hydroxy-N'-(2-methyl-benzyl)-malonamide...)
Affinity DataIC50:  41nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50197503(CHEMBL425291 | N-hydroxy-2-isobutyl-N'-(3-phenoxy-...)
Affinity DataIC50:  45nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50197497(2-benzyl-N-hydroxy-N'-(4-phenyl-butyl)-malonamide ...)
Affinity DataIC50:  46nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50206556(2-Benzyl-N-(4-fluoro-benzyl)-N'-hydroxy-malonamide...)
Affinity DataIC50:  57nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50206547(CHEMBL374479 | N-hydroxy-2-isobutyl-N'-naphthalen-...)
Affinity DataIC50:  91nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50206543(2-benzyl-N-hydroxy-N'-naphthalen-1-ylmethyl-malona...)
Affinity DataIC50:  107nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50206551(CHEMBL376198 | N-hydroxy-2-isobutyl-N'-(1,2,3,4-te...)
Affinity DataIC50:  109nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50062474(2,N-Dibenzyl-N'-hydroxy-malonamide | 2N-dibenzyl-N...)
Affinity DataIC50:  125nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50062453(2-Benzyl-N-hydroxy-N'-(3-phenyl-propyl)-malonamide...)
Affinity DataIC50:  125nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50206552(2-(3-phenoxybenzyl)-N1-(4-chlorobenzyl)-N3-hydroxy...)
Affinity DataIC50:  130nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50197501(2-(3-phenoxybenzyl)-N1-benzyl-N3-hydroxymalonamide...)
Affinity DataIC50:  164nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50206546(2-benzyl-N-(4-chloro-benzyl)-N'-hydroxy-malonamide...)
Affinity DataIC50:  170nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50206557(2-benzyl-3-(4-benzyl-piperidin-1-yl)-N-hydroxy-3-o...)
Affinity DataIC50:  206nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50197505(2-(3-phenoxybenzyl)-N1-hydroxy-N3-(4-phenylbutyl)m...)
Affinity DataIC50:  225nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50206566(2-(3-phenoxybenzyl)-N1-(4-(trifluoromethyl)benzyl)...)
Affinity DataIC50:  231nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50206564(2-(3-phenoxybenzyl)-3-(4-benzylpiperidin-1-yl)-N-h...)
Affinity DataIC50:  248nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50206545(2-benzyl-3-(3,4-dihydro-1H-isoquinolin-2-yl)-N-hyd...)
Affinity DataIC50:  253nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM23971((2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-phenylbutanami...)
Affinity DataIC50:  284nMAssay Description:Inhibitory activity for Plasmodium falciparum Zinc aminopeptidaseMore data for this Ligand-Target Pair
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50206555(2-[1-Phenyl-meth-(Z)-ylidene]-malonic Acid Monoeth...)
Affinity DataIC50:  330nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50197495(2-(4-benzyl-piperidine-1-carbonyl)-4-methyl-pentan...)
Affinity DataIC50:  406nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50197494(CHEMBL220253 | N-benzyl-N'-hydroxy-2-isobutyl-malo...)
Affinity DataIC50:  495nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50206565(2-(3-phenoxybenzyl)-N1-hydroxy-N3-(3-phenylpropyl)...)
Affinity DataIC50:  527nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetM1 family aminopeptidase(Plasmodium falciparum (isolate FcB1 / Columbia))
Monash University

Curated by ChEMBL
LigandPNGBDBM50062478(CHEMBL116641 | N-Hydroxy-2-isobutyl-N'-(3-phenyl-p...)
Affinity DataIC50:  790nMAssay Description:Inhibition of Plasmodium falciparum FcB1 M1 aminopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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