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Found 354 Enz. Inhib. hit(s) with Target = 'Probable nicotinate-nucleotide adenylyltransferase'
TargetProbable nicotinate-nucleotide adenylyltransferase(Bacillus anthracis)
Burnham Institute For Medical Research

LigandPNGBDBM50318652((E)-4-(2-(anthracen-9-ylmethylene)hydrazinyl)-N-(3...)
Affinity DataKi:  9.00E+3nM IC50:  2.50E+4nMAssay Description:The enzymatic assay was masured at fixed NaMN and ATP concentration (equal to two-fold km values)with various concentration of inhibitory compounds.More data for this Ligand-Target Pair
TargetProbable nicotinate-nucleotide adenylyltransferase(Bacillus anthracis)
Burnham Institute For Medical Research

LigandPNGBDBM50318652((E)-4-(2-(anthracen-9-ylmethylene)hydrazinyl)-N-(3...)
Affinity DataKi:  9.00E+3nMAssay Description:Inhibition of Bacillus anthracis nicotinate-nucleotide adenylyltransferase preincubated for 5 mins before addition of NaMN substrate by malachite gre...More data for this Ligand-Target Pair
TargetProbable nicotinate-nucleotide adenylyltransferase(Bacillus anthracis)
Burnham Institute For Medical Research

LigandPNGBDBM50318652((E)-4-(2-(anthracen-9-ylmethylene)hydrazinyl)-N-(3...)
Affinity DataKi:  1.00E+4nMAssay Description:The enzymatic assay was masured at fixed NaMN and ATP concentration (equal to two-fold km values)with various concentration of inhibitory compounds.More data for this Ligand-Target Pair
TargetProbable nicotinate-nucleotide adenylyltransferase(Bacillus anthracis)
Burnham Institute For Medical Research

LigandPNGBDBM50318652((E)-4-(2-(anthracen-9-ylmethylene)hydrazinyl)-N-(3...)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of Bacillus anthracis nicotinate-nucleotide adenylyltransferase preincubated for 5 mins before addition of ATP substrate by malachite gree...More data for this Ligand-Target Pair
TargetProbable nicotinate-nucleotide adenylyltransferase(Bacillus anthracis)
Burnham Institute For Medical Research

LigandPNGBDBM50318653(3-amino-N-(3-fluorophenyl)-6-(thiophen-2-yl)thieno...)
Affinity DataKi:  1.80E+4nM IC50:  3.60E+4nMAssay Description:The enzymatic assay was masured at fixed NaMN and ATP concentration (equal to two-fold km values)with various concentration of inhibitory compounds.More data for this Ligand-Target Pair
TargetProbable nicotinate-nucleotide adenylyltransferase(Bacillus anthracis)
Burnham Institute For Medical Research

LigandPNGBDBM50318653(3-amino-N-(3-fluorophenyl)-6-(thiophen-2-yl)thieno...)
Affinity DataKi:  1.80E+4nMAssay Description:Inhibition of Bacillus anthracis nicotinate-nucleotide adenylyltransferase preincubated for 5 mins before addition of NaMN substrate by malachite gre...More data for this Ligand-Target Pair
TargetProbable nicotinate-nucleotide adenylyltransferase(Bacillus anthracis)
Burnham Institute For Medical Research

LigandPNGBDBM50318653(3-amino-N-(3-fluorophenyl)-6-(thiophen-2-yl)thieno...)
Affinity DataKi:  3.20E+4nMAssay Description:Inhibition of Bacillus anthracis nicotinate-nucleotide adenylyltransferase preincubated for 5 mins before addition of ATP substrate by malachite gree...More data for this Ligand-Target Pair
TargetProbable nicotinate-nucleotide adenylyltransferase(Bacillus anthracis)
Burnham Institute For Medical Research

LigandPNGBDBM50318653(3-amino-N-(3-fluorophenyl)-6-(thiophen-2-yl)thieno...)
Affinity DataKi:  3.20E+4nMAssay Description:The enzymatic assay was masured at fixed NaMN and ATP concentration (equal to two-fold km values)with various concentration of inhibitory compounds.More data for this Ligand-Target Pair
TargetProbable nicotinate-nucleotide adenylyltransferase(Staphylococcus aureus subsp. aureus N315)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM33039(2-amino-4-(4-chlorophenyl)-6-(5-methyl-2-furanyl)-...)
Affinity DataIC50:  808nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProbable nicotinate-nucleotide adenylyltransferase(Bacillus anthracis)
Burnham Institute For Medical Research

LigandPNGBDBM50266764(CHEMBL475957 | Compound ID 5824 | N-(3,4-dichlorop...)
Affinity DataIC50:  2.00E+3nMpH: 7.5 T: 2°CAssay Description:Inhibitory concentration of the compound measured against B. anthracis Nicotinic acid mononucleotide adenylyltransferase (NaMNAT)using HPLC Enzyme As...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable nicotinate-nucleotide adenylyltransferase(Staphylococcus aureus subsp. aureus N315)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM33041(2-amino-6-(5-methyl-2-furanyl)-4-(4-methylphenyl)-...)
Affinity DataIC50:  2.43E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProbable nicotinate-nucleotide adenylyltransferase(Staphylococcus aureus subsp. aureus N315)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM81213(1-nitro-3-[(3-nitrophenyl)disulfanyl]benzene | MLS...)
Affinity DataIC50:  3.73E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProbable nicotinate-nucleotide adenylyltransferase(Bacillus anthracis)
Burnham Institute For Medical Research

LigandPNGBDBM50318660((E)-4-(2-(anthracen-9-ylmethylene)hydrazinyl)-N-(3...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of Bacillus anthracis nicotinate-nucleotide adenylyltransferase preincubated for 5 mins before addition of substrate by malachite green re...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable nicotinate-nucleotide adenylyltransferase(Staphylococcus aureus subsp. aureus N315)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM88962((6R,7R)-7-[[(2E)-2-(2-amino-1,3-thiazol-4-yl)-2-(c...)
Affinity DataIC50:  4.25E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProbable nicotinate-nucleotide adenylyltransferase(Staphylococcus aureus subsp. aureus N315)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM61897(7-methyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carbox...)
Affinity DataIC50:  4.50E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProbable nicotinate-nucleotide adenylyltransferase(Staphylococcus aureus subsp. aureus N315)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM80066(1-(4-methyl-3,5-dinitro-phenyl)-3-pyrroline-2,5-qu...)
Affinity DataIC50:  6.33E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProbable nicotinate-nucleotide adenylyltransferase(Staphylococcus aureus subsp. aureus N315)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM283(6-[(8-chloro-4-hydroxy-3-{[4-hydroxy-3-(3-methylbu...)
Affinity DataIC50:  7.01E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProbable nicotinate-nucleotide adenylyltransferase(Bacillus anthracis)
Burnham Institute For Medical Research

LigandPNGBDBM98089(1-[4-[(3,4-dichlorophenyl)sulfonylamino]phenyl]-3-...)
Affinity DataIC50:  7.30E+3nMpH: 7.5 T: 2°CAssay Description:Inhibitory concentration of the compound measured against B. anthracis Nicotinic acid mononucleotide adenylyltransferase (NaMNAT)using HPLC Enzyme As...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable nicotinate-nucleotide adenylyltransferase(Staphylococcus aureus subsp. aureus N315)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM95184(2-amino-4-(2-chlorophenyl)-6-(5-methyl-2-furanyl)-...)
Affinity DataIC50:  7.76E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProbable nicotinate-nucleotide adenylyltransferase(Staphylococcus aureus subsp. aureus N315)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM95178(5-bromanyl-N-[2-(2,4-dimethylphenyl)-4,6-dihydroth...)
Affinity DataIC50:  8.03E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProbable nicotinate-nucleotide adenylyltransferase(Bacillus anthracis)
Burnham Institute For Medical Research

LigandPNGBDBM81357(NadD inhibitor 3_05 | US8785499, 3_05)
Affinity DataIC50:  9.00E+3nMAssay Description:The enzymatic assay was masured at fixed NaMN and ATP concentration (equal to two-fold km values)with various concentration of inhibitory compounds.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable nicotinate-nucleotide adenylyltransferase(Staphylococcus aureus subsp. aureus N315)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM81225(2-(2-hydroxyphenyl)sulfinylsulfinylphenol | MLS002...)
Affinity DataIC50:  9.15E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetProbable nicotinate-nucleotide adenylyltransferase(Bacillus anthracis)
Burnham Institute For Medical Research

LigandPNGBDBM98138(1-[4-[(4-methoxyphenyl)sulfonylamino]phenyl]-3-(4-...)
Affinity DataIC50:  1.01E+4nMpH: 7.5 T: 2°CAssay Description:Inhibitory concentration of the compound measured against B. anthracis Nicotinic acid mononucleotide adenylyltransferase (NaMNAT)using HPLC Enzyme As...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable nicotinate-nucleotide adenylyltransferase(Staphylococcus aureus subsp. aureus N315)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM95186(2-Chloro-5-{5-[(naphtho[2,1-b]furan-2-carbonyl)-hy...)
Affinity DataIC50:  1.07E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProbable nicotinate-nucleotide adenylyltransferase(Staphylococcus aureus subsp. aureus N315)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM47367((4Z)-2-(3,4-dimethylphenyl)-4-[[2-(5-keto-3-thioxo...)
Affinity DataIC50:  1.12E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProbable nicotinate-nucleotide adenylyltransferase(Staphylococcus aureus subsp. aureus N315)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM88679((7E)-7-[(2E)-2-(6-ethoxy-1-methyl-2-quinolinyliden...)
Affinity DataIC50:  1.17E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetProbable nicotinate-nucleotide adenylyltransferase(Staphylococcus aureus subsp. aureus N315)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM95187(2-Amino-benzoic acid N'-((Z)-2-hydroxy-4-oxo-4...)
Affinity DataIC50:  1.20E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProbable nicotinate-nucleotide adenylyltransferase(Bacillus anthracis)
Burnham Institute For Medical Research

LigandPNGBDBM81358(NadD inhibitor 3_15 | US8785499, 3_15)
Affinity DataIC50:  1.20E+4nMAssay Description:The enzymatic assay was masured at fixed NaMN and ATP concentration (equal to two-fold km values)with various concentration of inhibitory compounds.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable nicotinate-nucleotide adenylyltransferase(Bacillus anthracis)
Burnham Institute For Medical Research

LigandPNGBDBM98099(1-[4-[(4-ethylphenyl)sulfonylamino]phenyl]-3-(3-ni...)
Affinity DataIC50:  1.20E+4nMpH: 7.5 T: 2°CAssay Description:Inhibitory concentration of the compound measured against B. anthracis Nicotinic acid mononucleotide adenylyltransferase (NaMNAT)using HPLC Enzyme As...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable nicotinate-nucleotide adenylyltransferase(Bacillus anthracis)
Burnham Institute For Medical Research

LigandPNGBDBM98161(1-[4-[[4-(aminomethyl)phenyl]sulfonylamino]phenyl]...)
Affinity DataIC50:  1.21E+4nMpH: 7.5 T: 2°CAssay Description:Inhibitory concentration of the compound measured against B. anthracis Nicotinic acid mononucleotide adenylyltransferase (NaMNAT)using HPLC Enzyme As...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable nicotinate-nucleotide adenylyltransferase(Staphylococcus aureus subsp. aureus N315)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM61528(MLS000862515 | N-(4-{[(3,4-dimethyl-5-isoxazolyl)a...)
Affinity DataIC50:  1.25E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProbable nicotinate-nucleotide adenylyltransferase(Bacillus anthracis)
Burnham Institute For Medical Research

LigandPNGBDBM50318661(CHEMBL1084867 | N-(2-Chloro-phenyl)-3-(4-{[3-(2-ch...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of Bacillus anthracis nicotinate-nucleotide adenylyltransferase preincubated for 5 mins before addition of substrate by malachite green re...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable nicotinate-nucleotide adenylyltransferase(Bacillus anthracis)
Burnham Institute For Medical Research

LigandPNGBDBM50318661(CHEMBL1084867 | N-(2-Chloro-phenyl)-3-(4-{[3-(2-ch...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of Bacillus anthracis nicotinate-nucleotide adenylyltransferase preincubated for 5 mins before addition of substrate by malachite green re...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable nicotinate-nucleotide adenylyltransferase(Bacillus anthracis)
Burnham Institute For Medical Research

LigandPNGBDBM98122(1-(4-nitrophenyl)-3-[4-[[2-(trifluoromethyl)phenyl...)
Affinity DataIC50:  1.33E+4nMpH: 7.5 T: 2°CAssay Description:Inhibitory concentration of the compound measured against B. anthracis Nicotinic acid mononucleotide adenylyltransferase (NaMNAT)using HPLC Enzyme As...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable nicotinate-nucleotide adenylyltransferase(Staphylococcus aureus subsp. aureus N315)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM95154(3-[(3-fluorophenyl)methylsulfanylmethyl]-7-[3-meth...)
Affinity DataIC50:  1.38E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProbable nicotinate-nucleotide adenylyltransferase(Staphylococcus aureus subsp. aureus N315)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM52889(4-(7-hydrocinnamoyloxy-6,8-diketo-7-methyl-isochro...)
Affinity DataIC50:  1.42E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProbable nicotinate-nucleotide adenylyltransferase(Staphylococcus aureus subsp. aureus N315)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM83188((3Z)-3-(2-furanylmethylidene)-1,2-dihydrocyclopent...)
Affinity DataIC50:  1.46E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProbable nicotinate-nucleotide adenylyltransferase(Staphylococcus aureus subsp. aureus N315)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM83905(4-[(3-keto-5-methyl-3-pyrazolin-4-yl)-[1-(1-naphth...)
Affinity DataIC50:  1.47E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProbable nicotinate-nucleotide adenylyltransferase(Staphylococcus aureus subsp. aureus N315)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM50548(MLS001017412 | N-[(E)-1-(2-furyl)ethylideneamino]-...)
Affinity DataIC50:  1.48E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProbable nicotinate-nucleotide adenylyltransferase(Staphylococcus aureus subsp. aureus N315)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM29685((3E)-3-(2-furanylmethylidene)-1,2-dihydrocyclopent...)
Affinity DataIC50:  1.50E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProbable nicotinate-nucleotide adenylyltransferase(Staphylococcus aureus subsp. aureus N315)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM70614(2-(3,4-dimethylphenyl)-4-[[1-(3,4-dimethylphenyl)-...)
Affinity DataIC50:  1.51E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProbable nicotinate-nucleotide adenylyltransferase(Staphylococcus aureus subsp. aureus N315)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM33116((E)-3-(5-methyl-2-furanyl)-N-[3-[[(E)-3-(5-methyl-...)
Affinity DataIC50:  1.53E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProbable nicotinate-nucleotide adenylyltransferase(Staphylococcus aureus subsp. aureus N315)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM37848(2-[[3-carbethoxy-4-(4-phenylphenyl)-2-thienyl]carb...)
Affinity DataIC50:  1.53E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProbable nicotinate-nucleotide adenylyltransferase(Staphylococcus aureus subsp. aureus N315)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM51992(3-[[(E)-[2-(4-bromobenzyl)oxybenzylidene]amino]thi...)
Affinity DataIC50:  1.54E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProbable nicotinate-nucleotide adenylyltransferase(Staphylococcus aureus subsp. aureus N315)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM45519(2-(2,4-dimethylphenyl)-N-(4-{[(5-methyl-3-isoxazol...)
Affinity DataIC50:  1.54E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProbable nicotinate-nucleotide adenylyltransferase(Staphylococcus aureus subsp. aureus N315)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM82868(4-[(2-ketoindol-3-yl)amino]-N-thiazol-2-yl-benzene...)
Affinity DataIC50:  1.55E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetProbable nicotinate-nucleotide adenylyltransferase(Staphylococcus aureus subsp. aureus N315)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM80054(2-[[4-[2-[(4-ethoxyphenyl)methylidene]hydrazinyl]-...)
Affinity DataIC50:  1.56E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProbable nicotinate-nucleotide adenylyltransferase(Staphylococcus aureus subsp. aureus N315)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM95127(5-(2,5-dichlorobenzyl)-4-methyl-4-thiazoline-2-thi...)
Affinity DataIC50:  1.57E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProbable nicotinate-nucleotide adenylyltransferase(Staphylococcus aureus subsp. aureus N315)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM95173(MLS000438847 | SMR000452599 | [3-(4-cyanophenyl)-7...)
Affinity DataIC50:  1.57E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetProbable nicotinate-nucleotide adenylyltransferase(Staphylococcus aureus subsp. aureus N315)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM51991(3-[[(E)-[2-(3-bromobenzyl)oxybenzylidene]amino]thi...)
Affinity DataIC50:  1.58E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
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