TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataKi: 2.80E+3nMAssay Description:Compound was evaluated for its ability to inhibit carnitine palmitoyltransferase I activity in intact mitochondria from rat heartMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataKi: 1.00E+5nMAssay Description:Tested against neonatal rat cardiac myocyte carnitine palmitoyltransferase 1More data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataKi: 1.40E+6nMAssay Description:Tested against neonatal rat cardiac myocyte carnitine palmitoyltransferase 1More data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataKi: 3.60E+6nMAssay Description:Tested against neonatal rat cardiac myocyte carnitine palmitoyltransferase 1More data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of rat CPT1B expressed in intact Saccharomyces cerevisiae using [methyl-3H]carnitine by radiometric assayMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche
Curated by ChEMBL
F. Hoffmann-La Roche
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche
Curated by ChEMBL
F. Hoffmann-La Roche
Curated by ChEMBL
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of Wistar rat heart mitochondrial CPT-1 assessed as reduction in conversion of palmitoyl CoA and L-carnitine into palmitoylcarnitine prein...More data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of CPT1A in rat myocardiumMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataIC50: 1.45E+3nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]-palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataIC50: 3.40E+3nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]-palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche
Curated by ChEMBL
F. Hoffmann-La Roche
Curated by ChEMBL
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche
Curated by ChEMBL
F. Hoffmann-La Roche
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]-palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche
Curated by ChEMBL
F. Hoffmann-La Roche
Curated by ChEMBL
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]-palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataIC50: 5.80E+3nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche
Curated by ChEMBL
F. Hoffmann-La Roche
Curated by ChEMBL
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]-palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]-palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche
Curated by ChEMBL
F. Hoffmann-La Roche
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of CPT1B in heart mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of Wistar rat heart mitochondrial CPT-1 assessed as reduction in conversion of palmitoyl CoA and L-carnitine into palmitoylcarnitine prein...More data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of Wistar rat heart mitochondrial CPT-1 assessed as reduction in conversion of palmitoyl CoA and L-carnitine into palmitoylcarnitine prein...More data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of Wistar rat heart mitochondrial CPT-1 assessed as reduction in conversion of palmitoyl CoA and L-carnitine into palmitoylcarnitine prein...More data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of Wistar rat heart mitochondrial CPT-1 assessed as reduction in conversion of palmitoyl CoA and L-carnitine into palmitoylcarnitine prein...More data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche
Curated by ChEMBL
F. Hoffmann-La Roche
Curated by ChEMBL
Affinity DataIC50: 2.17E+4nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataIC50: 2.73E+4nMAssay Description:Maximal inhibition of rat CPT1AMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of Wistar rat heart mitochondrial CPT-1 assessed as reduction in conversion of palmitoyl CoA and L-carnitine into palmitoylcarnitine prein...More data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataIC50: 4.34E+4nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibition of Wistar rat heart mitochondrial CPT-1 assessed as reduction in conversion of palmitoyl CoA and L-carnitine into palmitoylcarnitine prein...More data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataIC50: 4.62E+4nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche
Curated by ChEMBL
F. Hoffmann-La Roche
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of CPT1BMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche
Curated by ChEMBL
F. Hoffmann-La Roche
Curated by ChEMBL
Affinity DataIC50: 6.03E+4nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataIC50: 7.70E+4nMAssay Description:Inhibition of rat heart mitochondrial CPT-1More data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataIC50: 8.01E+4nMAssay Description:In vitro inhibition of [14C]-palmitoyl-CoA and carnitine binding to carnitine palmitoyltransferase I of rat heart mitochondriaMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataIC50: 8.32E+4nMAssay Description:Inhibitory activity against rat heart mitochondrial carnitine palmitoyltransferase 1b using [14C]-palmitoyl-CoA as radioligandMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche
Curated by ChEMBL
F. Hoffmann-La Roche
Curated by ChEMBL
Affinity DataIC50: 8.53E+4nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Rattus norvegicus)
Louisiana State University
Curated by ChEMBL
Louisiana State University
Curated by ChEMBL
Affinity DataIC50: 8.80E+4nMAssay Description:Inhibition of Wistar rat heart mitochondrial CPT-1 assessed as reduction in conversion of palmitoyl CoA and L-carnitine into palmitoylcarnitine prein...More data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche
Curated by ChEMBL
F. Hoffmann-La Roche
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche
Curated by ChEMBL
F. Hoffmann-La Roche
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair
TargetCarnitine O-palmitoyltransferase 1, muscle isoform(Homo sapiens (Human))
F. Hoffmann-La Roche
Curated by ChEMBL
F. Hoffmann-La Roche
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human CPT1BMore data for this Ligand-Target Pair