TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataKi: 1.30E+4nMAssay Description:Binding affinity to human EAAT1 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataKi: 1.30E+4nMAssay Description:Binding affinity to human EAAT1 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataKi: 2.30E+4nMAssay Description:Binding affinity to human EAAT1 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataKi: 2.90E+4nMAssay Description:Binding affinity to human EAAT1 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataKi: 3.50E+4nMAssay Description:Binding affinity to human EAAT1 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataKi: 3.50E+4nMAssay Description:Inhibition of [3H]D-Asp uptake at EAAT1 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataKi: 5.00E+4nMAssay Description:Binding affinity to human EAAT1 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataKi: 5.50E+4nMAssay Description:Binding affinity to human EAAT1 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataKi: 1.20E+5nMAssay Description:Binding affinity to human EAAT1 expressed in HEK293 cells in FMP (FLPR) assayMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataKi: 1.27E+5nMAssay Description:Activity against human EAAT1 transfected in HEK293 cellsMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataKi: 2.00E+5nMAssay Description:Inhibition of human EAAT1 expressed in HEK293 cells by FLIPR membrane potential assayMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataKi: 2.00E+5nMAssay Description:Inhibition of human EAAT1 expressed in HEK293 cells by FLIPR membrane potential assayMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataKi: >4.00E+5nMAssay Description:Activity against human EAAT1 transfected in HEK293 cellsMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataKi: 4.50E+5nMAssay Description:Inhibition of [3H]D-Asp uptake at EAAT1 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataKi: 1.00E+6nMAssay Description:Inhibition of [3H]D-Asp uptake at EAAT1 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataKi: 1.00E+6nMAssay Description:Inhibition of [3H]D-Asp uptake at EAAT1 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataKi: 1.00E+6nMAssay Description:Inhibition of [3H]D-Asp uptake at EAAT1 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataKi: >3.00E+6nMAssay Description:Inhibition of [3H]D-Asp uptake at EAAT1 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataKi: >3.00E+6nMAssay Description:Inhibition of [3H]D-Asp uptake at EAAT1 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataKi: 3.00E+6nMAssay Description:Inhibition of [3H]D-Asp uptake at EAAT1 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataKi: >3.00E+6nMAssay Description:Inhibition of [3H]D-Asp uptake at EAAT1 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataKi: >3.00E+6nMAssay Description:Inhibition of [3H]D-Asp uptake at EAAT1 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataKi: >3.00E+6nMAssay Description:Inhibition of [3H]D-Asp uptake at EAAT1 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataIC50: 3.5nMAssay Description:Inhibition of human EAAT1 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataIC50: 3.60nMAssay Description:Inhibition of human EAAT1 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataIC50: 5.10nMAssay Description:Inhibition of human EAAT1 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataIC50: 5.10nMAssay Description:Inhibition of human EAAT1 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataIC50: 6.10nMAssay Description:Inhibition of human EAAT1 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataIC50: 6.20nMAssay Description:Inhibition of human EAAT1 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataIC50: 11nMAssay Description:Inhibition of human EAAT1 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataIC50: 11nMAssay Description:Inhibition of human EAAT1 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataIC50: 12nMAssay Description:Inhibition of human EAAT1 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataIC50: 12nMAssay Description:Inhibition of human EAAT1 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataIC50: 21nMAssay Description:Inhibition of human EAAT1 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataIC50: 21nMAssay Description:Inhibition of human EAAT1 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataIC50: 22nMAssay Description:Inhibition of EAAT1 (unknown origin) transiently expressed in COS1 cells by [14C]glutamate based uptake assayMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataIC50: 31nMAssay Description:Inhibition of human EAAT1 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataIC50: 31nMAssay Description:Inhibition of human EAAT1 expressed in HEK293 cells assessed as reduction in [3H]-D-Asp uptake incubated for 4 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataIC50: 100nMAssay Description:Inhibitory concentration against glutamate uptake in HEK cells expressing human Excitatory amino acid transporter 1More data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataIC50: 100nMAssay Description:Inhibitory concentration against glutamate uptake in HEK cells expressing human Excitatory amino acid transporter 1More data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataIC50: 120nMAssay Description:Activity at human EAAT1 expressed in HEK293 cells assessed as inhibition of Glu-induced fluorescent response by FLIPR membrane potential blue assayMore data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataIC50: 130nMAssay Description:Inhibitory concentration against glutamate uptake in HEK cells expressing human Excitatory amino acid transporter 1More data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataIC50: 150nMAssay Description:Inhibitory concentration against glutamate uptake in HEK cells expressing human Excitatory amino acid transporter 1More data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataIC50: 200nMAssay Description:Inhibitory concentration against glutamate uptake in HEK cells expressing human Excitatory amino acid transporter 1More data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataIC50: 200nMAssay Description:Inhibitory concentration against glutamate uptake in HEK cells expressing human Excitatory amino acid transporter 1More data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataIC50: 300nMAssay Description:Inhibitory concentration against glutamate uptake in HEK cells expressing human Excitatory amino acid transporter 1More data for this Ligand-Target Pair
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
Wyeth Research
Curated by PDSP Ki Database
Wyeth Research
Curated by PDSP Ki Database
Affinity DataIC50: 300nMAssay Description:Inhibitory concentration against glutamate uptake in HEK cells expressing human Excitatory amino acid transporter 1More data for this Ligand-Target Pair