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Found 179 Enz. Inhib. hit(s) with Target = 'Fibroblast growth factor receptor 3 [397-806]'
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350059(US10208024, Example 58 | US10766881, Example 58)
Affinity DataIC50:  0.700nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350052(US10208024, Example 51 | US10766881, Example 51)
Affinity DataIC50:  1nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350049(6-(3-amino-6-(1-methyl- 1H-pyrazol-4-yl)pyrazin- 2...)
Affinity DataIC50:  1.40nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350048(US10208024, Example 47 | US10766881, Example 47)
Affinity DataIC50:  1.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350015(6-(3-amino-6-(1- methyl-1H-pyrazol-4- yl)pyrazin-2...)
Affinity DataIC50:  1.70nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350044(US10208024, Example 43 | US10766881, Example 43)
Affinity DataIC50:  1.70nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350033(US10208024, Example 32 | US10766881, Example 32)
Affinity DataIC50:  1.80nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350051(US10208024, Example 50 | US10766881, Example 50)
Affinity DataIC50:  1.80nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350050(6-(3-amino-6-(1-methyl- 1H-pyrazol-4-yl)pyrazin- 2...)
Affinity DataIC50:  2.10nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350083(US10208024, Example 82 | US10766881, Example 82)
Affinity DataIC50:  2.20nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350020(US10208024, Example 19 | US10766881, Example 19)
Affinity DataIC50:  2.20nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350005(1-((4-(5-amino-6-(1- (3,5- dimethoxyphenyl)-6- oxo...)
Affinity DataIC50:  2.40nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350024(US10208024, Example 23 | US10766881, Example 23)
Affinity DataIC50:  2.80nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350006(6-(3-amino-6-(1- (4,4,4-trifluoro-2- hydroxybutyl)...)
Affinity DataIC50:  2.90nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350042(US10208024, Example 41 | US10766881, Example 41)
Affinity DataIC50:  3.20nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350018(6-(3-amino-6-(1- (cyclopropylmethyl)- 1H-pyrazol-4...)
Affinity DataIC50:  3.80nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350067(US10208024, Example 66 | US10766881, Example 66)
Affinity DataIC50:  3.90nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350032(US10208024, Example 31 | US10766881, Example 31)
Affinity DataIC50:  3.90nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350025(US10208024, Example 24 | US10766881, Example 24)
Affinity DataIC50:  4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350002(US10208024, Example 1 | US10766881, Example 1)
Affinity DataIC50:  4.30nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350027(US10208024, Example 26 | US10766881, Example 26)
Affinity DataIC50:  4.30nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350034(US10208024, Example 33 | US10766881, Example 33)
Affinity DataIC50:  4.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350029(US10208024, Example 28 | US10766881, Example 28)
Affinity DataIC50:  4.70nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350036(US10208024, Example 35 | US10766881, Example 35)
Affinity DataIC50:  4.80nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350022(6-(3-amino-6-(1- isobutyl-1H-pyrazol- 4-yl)pyrazin...)
Affinity DataIC50:  4.90nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350073(6-(3-amino-6-(1-(1- hydroxy-2- methylpropan-2-yl)-...)
Affinity DataIC50:  5.20nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350057(US10208024, Example 56 | US10766881, Example 56)
Affinity DataIC50:  5.70nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350074(6-(3-amino-6-(1- isopropyl-1H-pyrazol-4- yl)pyrazi...)
Affinity DataIC50:  6nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350075(6-(3-amino-6-(1- cyclopropyl-1H-pyrazol- 4-yl)pyra...)
Affinity DataIC50:  6.10nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350058(US10208024, Example 57 | US10766881, Example 57)
Affinity DataIC50:  6.20nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350045(US10208024, Example 44 | US10766881, Example 44)
Affinity DataIC50:  6.20nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350069(US10208024, Example 68 | US10766881, Example 68)
Affinity DataIC50:  6.40nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350031(US10208024, Example 30 | US10766881, Example 30)
Affinity DataIC50:  6.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350023(6-(3-amino-6-(1- cyclobutyl-1H- pyrazol-4-yl)pyraz...)
Affinity DataIC50:  6.70nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350079(US10208024, Example 78 | US10766881, Example 78)
Affinity DataIC50:  6.90nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350016(6-(3-amino-6-(1- isopropyl-1H-pyrazol- 4-yl)pyrazi...)
Affinity DataIC50:  7nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350077(US10208024, Example 76 | US10766881, Example 76)
Affinity DataIC50:  7.10nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350030(US10208024, Example 29 | US10766881, Example 29)
Affinity DataIC50:  7.10nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806]/Glutathione S-transferase P(Homo sapiens (Human))
Bayer Intelletual Property

US Patent
LigandPNGBDBM255620(US9475815, 5)
Affinity DataIC50:  7.40nMpH: 7.0 T: 2°CAssay Description:A recombinant tagged FGFR-3 fusion protein [fusion of glutathione-S-transferase (GST) (N-terminally), His6-tag, thrombin cleavage site, and the intra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806]/Glutathione S-transferase P(Homo sapiens (Human))
Bayer Intelletual Property

US Patent
LigandPNGBDBM255624(US9475815, 9)
Affinity DataIC50:  7.40nMpH: 7.0 T: 2°CAssay Description:A recombinant tagged FGFR-3 fusion protein [fusion of glutathione-S-transferase (GST) (N-terminally), His6-tag, thrombin cleavage site, and the intra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806]/Glutathione S-transferase P(Homo sapiens (Human))
Bayer Intelletual Property

US Patent
LigandPNGBDBM255633(US9475815, 18)
Affinity DataIC50:  7.80nMpH: 7.0 T: 2°CAssay Description:A recombinant tagged FGFR-3 fusion protein [fusion of glutathione-S-transferase (GST) (N-terminally), His6-tag, thrombin cleavage site, and the intra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806]/Glutathione S-transferase P(Homo sapiens (Human))
Bayer Intelletual Property

US Patent
LigandPNGBDBM255636(US9475815, 21)
Affinity DataIC50:  8nMpH: 7.0 T: 2°CAssay Description:A recombinant tagged FGFR-3 fusion protein [fusion of glutathione-S-transferase (GST) (N-terminally), His6-tag, thrombin cleavage site, and the intra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350028(US10208024, Example 27 | US10766881, Example 27)
Affinity DataIC50:  8.20nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350043(US10208024, Example 42 | US10766881, Example 42)
Affinity DataIC50:  8.60nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350019(6-(3-amino-6-(1-(2- hydroxy-2- methylpropyl)-1H- p...)
Affinity DataIC50:  8.70nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350070(US10208024, Example 69 | US10766881, Example 69)
Affinity DataIC50:  9.60nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806]/Glutathione S-transferase P(Homo sapiens (Human))
Bayer Intelletual Property

US Patent
LigandPNGBDBM255701(US9475815, 86)
Affinity DataIC50:  9.60nMpH: 7.0 T: 2°CAssay Description:A recombinant tagged FGFR-3 fusion protein [fusion of glutathione-S-transferase (GST) (N-terminally), His6-tag, thrombin cleavage site, and the intra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806]/Glutathione S-transferase P(Homo sapiens (Human))
Bayer Intelletual Property

US Patent
LigandPNGBDBM255712(US9475815, 97)
Affinity DataIC50:  9.90nMpH: 7.0 T: 2°CAssay Description:A recombinant tagged FGFR-3 fusion protein [fusion of glutathione-S-transferase (GST) (N-terminally), His6-tag, thrombin cleavage site, and the intra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350055(US10208024, Example 54 | US10766881, Example 54)
Affinity DataIC50:  10.1nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFibroblast growth factor receptor 3 [397-806](Homo sapiens (Human))
Array Biopharma

US Patent
LigandPNGBDBM350076(6-(3-amino-6-(1- (azetidin-3-yl)-1H- pyrazol-4-yl)...)
Affinity DataIC50:  10.2nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Displayed 1 to 50 (of 179 total ) | Next | Last >>
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