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Found 316 Enz. Inhib. hit(s) with Target = 'Galanin receptor type 3'
TargetGalanin receptor type 3(RAT)
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50307256(CHEMBL604373 | GWTLNSAGYLLGPrPKPQQwFwLL-CONH2 | Ga...)
Affinity DataKi:  0.75nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(RAT)
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM85168(M32)
Affinity DataKi:  1.23nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(RAT)
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM85164(Galanin (1-29), rat)
Affinity DataKi:  1.47nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(RAT)
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50273370(CHEMBL503473 | GWTLNSAGYLLGPPPGFSPFR-CONH2 | Galan...)
Affinity DataKi:  2.09nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(RAT)
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM85200(Galanin (1-19), rat | Galanin rat)
Affinity DataKi:  3.31nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(RAT)
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM85068(Gal(1-13)-Std I)
Affinity DataKi:  4.47nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187911(1,3-dihydro-1-[3-(2-pyrrolidinylethoxy)phenyl]-3-[...)
Affinity DataKi:  5nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM85168(M32)
Affinity DataKi:  6.03nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM85168(M32)
Affinity DataKi:  6.03nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(RAT)
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM85200(Galanin (1-19), rat | Galanin rat)
Affinity DataKi:  6.25nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(RAT)
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM85070(Galanin, Porcine)
Affinity DataKi:  7.24nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(RAT)
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50273370(CHEMBL503473 | GWTLNSAGYLLGPPPGFSPFR-CONH2 | Galan...)
Affinity DataKi:  7.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187925(1-(3-(2-(piperidin-1-yl)ethoxy)phenyl)-3-(3-(trifl...)
Affinity DataKi:  8nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM85068(Gal(1-13)-Std I)
Affinity DataKi:  8.13nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM85068(Gal(1-13)-Std I)
Affinity DataKi:  8.13nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM85070(Galanin, Porcine)
Affinity DataKi:  9.77nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM85070(Galanin, Porcine)
Affinity DataKi:  9.77nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(RAT)
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM85073(CAS_3043476 | Galantide (M15) | NSC_3043476)
Affinity DataKi:  10.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM85200(Galanin (1-19), rat | Galanin rat)
Affinity DataKi:  12.3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM85200(Galanin (1-19), rat | Galanin rat)
Affinity DataKi:  12.3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(RAT)
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM85069(Galanin (2-29), rat | Galanin Porcine 2-29)
Affinity DataKi:  12.6nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50273370(CHEMBL503473 | GWTLNSAGYLLGPPPGFSPFR-CONH2 | Galan...)
Affinity DataKi:  14.4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50273370(CHEMBL503473 | GWTLNSAGYLLGPPPGFSPFR-CONH2 | Galan...)
Affinity DataKi:  14.4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187919(1-(3-(3-(diethylamino)-2-hydroxypropoxy)phenyl)-3-...)
Affinity DataKi:  15nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187923(1,3-dihydro-1-phenyl-3-[[3-(trilfluoromethyl)pheny...)
Affinity DataKi:  17nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187923(1,3-dihydro-1-phenyl-3-[[3-(trilfluoromethyl)pheny...)
Affinity DataKi:  17nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(RAT)
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM85201(Galanin (1-15)-ol,[Ala6,D-trp8])
Affinity DataKi:  17.9nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187922(1-(3-(3-(diethylamino)propoxy)phenyl)-3-(3-(triflu...)
Affinity DataKi:  21nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187912(1-(3-(2-(dimethylamino)ethoxy)phenyl)-3-(3-(triflu...)
Affinity DataKi:  26nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187908((S)-1-(3-(3-(diethylamino)-2-hydroxypropoxy)phenyl...)
Affinity DataKi:  27nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187916(1-(3-(3-(dimethylamino)propoxy)phenyl)-3-(3-(trifl...)
Affinity DataKi:  29nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187918(1-(4-(3-(diethylamino)propoxy)phenyl)-3-(3-(triflu...)
Affinity DataKi:  34nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187914(1-(3-((diethylamino)methoxy)phenyl)-3-(3-(trifluor...)
Affinity DataKi:  38nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM85073(CAS_3043476 | Galantide (M15) | NSC_3043476)
Affinity DataKi:  39.8nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM85073(CAS_3043476 | Galantide (M15) | NSC_3043476)
Affinity DataKi:  39.8nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187913(1-(3-(4-(diethylamino)butoxy)phenyl)-3-(3-(trifluo...)
Affinity DataKi:  45nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187926(1-(3-(3-(pyrrolidin-1-yl)propoxy)phenyl)-3-(3-(tri...)
Affinity DataKi:  49nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(RAT)
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM85205(Galanin (1-16) | Galanin (1-16), rat)
Affinity DataKi:  49.6nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50189598(1-(ethylpropyl)-3-{[3-(trifluoromethyl)phenyl]azam...)
Affinity DataKi:  52nMAssay Description:Displacement of [125I]galanin from human GAL3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(RAT)
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM85072(Galanin, Human)
Affinity DataKi:  52.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(RAT)
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50307254(CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2 | M40)
Affinity DataKi:  54nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM85069(Galanin (2-29), rat | Galanin Porcine 2-29)
Affinity DataKi:  60.3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM85072(Galanin, Human)
Affinity DataKi:  69.2nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM85072(Galanin, Human)
Affinity DataKi:  69.2nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187915(1-(4-(4-(diethylamino)butoxy)phenyl)-3-(3-(trifluo...)
Affinity DataKi:  70nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187910(1-(4-(2-(diethylamino)ethoxy)phenyl)-3-(3-(trifluo...)
Affinity DataKi:  78nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(RAT)
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50307254(CHEMBL604990 | GWTLNSAGYLLGPPPALALA-CONH2 | M40)
Affinity DataKi:  79.4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(RAT)
Schering-Plough Research Institute

Curated by PDSP Ki Database
LigandPNGBDBM50273369(CHEMBL526003 | GWTLNSAGYLLGPQQFFGLM-CONH2 | Galani...)
Affinity DataKi:  85nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187909(1-(3-(2-(diethylamino)ethoxy)phenyl)-3-(3-(trifluo...)
Affinity DataKi:  87nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGalanin receptor type 3(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50187917(1-(4-(2-(dimethylamino)ethoxy)phenyl)-3-(3-(triflu...)
Affinity DataKi:  89nMAssay Description:Displacement of [125I]galanin from human galanin Gal3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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