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Found 40 Enz. Inhib. hit(s) with Target = 'Opioid receptor delta 1'
TargetOpioid receptor delta 1(Cavia porcellus)
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50083926((6S,11R)-3-Cyclopropylmethyl-6,11-dimethyl-1,2,3,4...)
Affinity DataKi:  0.580nMAssay Description:Displacement of [3H]Naltrindole from DOR in guinea pig brain membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOpioid receptor delta 1(Bos taurus)
University Of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM85393(14β-(p-chlorocinnamoylamino)-7,8-dihydrocodei...)
Affinity DataKi:  0.75nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOpioid receptor delta 1(Cavia porcellus)
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50018731((Cyclazocine) 3-Cyclopropylmethyl-6,11-dimethyl-1,...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]Naltrindole from DOR in guinea pig brain membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOpioid receptor delta 1(Bos taurus)
University Of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM82090(DALLE)
Affinity DataKi:  1.80nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOpioid receptor delta 1(Bos taurus)
University Of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM21025((2R)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydro...)
Affinity DataKi:  1.80nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOpioid receptor delta 1(Cavia porcellus)
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50007102(6,11-Dimethyl-3-(tetrahydro-furan-2-ylmethyl)-1,2,...)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]Naltrindole from DOR in guinea pig brain membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOpioid receptor delta 1(Cavia porcellus)
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50045114(3-Cyclopropylmethyl-6-ethyl-8-hydroxy-11-methyl-3,...)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]Naltrindole from DOR in guinea pig brain membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOpioid receptor delta 1(Macaca mulatta)
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50458147(CHEMBL4204891)
Affinity DataKi:  4.20nMAssay Description:Displacement of [3H]naltrindole from DOR in monkey brain cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOpioid receptor delta 1(Cavia porcellus)
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50085020(((6S,11R)-3-Cyclopropylmethyl-6,11-dimethyl-1,2,3,...)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]Naltrindole from DOR in guinea pig brain membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOpioid receptor delta 1(Macaca mulatta)
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50001031(3-Allyl-6,11-dimethyl-1,2,3,4,5,6-hexahydro-2,6-me...)
Affinity DataKi:  5.5nMAssay Description:Displacement of [3H]naltrindole from DOR in monkey brain cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOpioid receptor delta 1(Macaca mulatta)
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50458145(CHEMBL4207341)
Affinity DataKi:  5.80nMAssay Description:Displacement of [3H]naltrindole from DOR in monkey brain cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOpioid receptor delta 1(Bos taurus)
University Of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM82090(DALLE)
Affinity DataKi:  7.40nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOpioid receptor delta 1(Cavia porcellus)
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50458137(CHEMBL4210742)
Affinity DataKi:  8.30nMAssay Description:Displacement of [3H]Naltrindole from DOR in guinea pig brain membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOpioid receptor delta 1(Cavia porcellus)
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50101160(3-Cyclopropylmethyl-6,11-dimethyl-1,2,3,4,5,6-hexa...)
Affinity DataKi:  8.30nMAssay Description:Displacement of [3H]Naltrindole from DOR in guinea pig brain membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOpioid receptor delta 1(Bos taurus)
University Of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM21025((2R)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydro...)
Affinity DataKi:  9.70nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOpioid receptor delta 1(Cavia porcellus)
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50254563(3-Cyclopropylmethyl-6-ethyl-11-methyl-1-oxo-1,2,3,...)
Affinity DataKi:  9.80nMAssay Description:Displacement of [3H]Naltrindole from DOR in guinea pig brain membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOpioid receptor delta 1(Cavia porcellus)
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50458143(CHEMBL4215981)
Affinity DataKi:  9.80nMAssay Description:Displacement of [3H]Naltrindole from DOR in guinea pig brain membranesMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetOpioid receptor delta 1(Macaca mulatta)
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50458146(CHEMBL4209962)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]naltrindole from DOR in monkey brain cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOpioid receptor delta 1(Cavia porcellus)
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50092176(3-Cyclopropylmethyl-6,11-dimethyl-1,2,3,4,5,6-hexa...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]Naltrindole from DOR in guinea pig brain membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOpioid receptor delta 1(Bos taurus)
University Of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM85395(MC-CAM)
Affinity DataKi:  12nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOpioid receptor delta 1(Bos taurus)
University Of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM81934(Beta-Endorphin)
Affinity DataKi:  14nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOpioid receptor delta 1(Bos taurus)
University Of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM85394(N-CPM-CACO)
Affinity DataKi:  16nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOpioid receptor delta 1(Bos taurus)
University Of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM50000788((morphine)4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...)
Affinity DataKi:  18.5nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOpioid receptor delta 1(Cavia porcellus)
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50458152(CHEMBL4207167)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]Naltrindole from DOR in guinea pig brain membranes after 3 hrs by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOpioid receptor delta 1(Macaca mulatta)
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50458148(CHEMBL4214248)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]naltrindole from DOR in monkey brain cortex membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOpioid receptor delta 1(Bos taurus)
University Of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM50000788((morphine)4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...)
Affinity DataKi:  29.7nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOpioid receptor delta 1(Bos taurus)
University Of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM50021325(4-methyl-(1S,5R,13R,14S)-12-oxa-4-azapentacyclo[9....)
Affinity DataKi:  35.6nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOpioid receptor delta 1(Cavia porcellus)
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50458141(CHEMBL4204304)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]Naltrindole from DOR in guinea pig brain membranesMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetOpioid receptor delta 1(Bos taurus)
University Of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM50021325(4-methyl-(1S,5R,13R,14S)-12-oxa-4-azapentacyclo[9....)
Affinity DataKi:  38.1nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOpioid receptor delta 1(Cavia porcellus)
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50458142(CHEMBL4208635)
Affinity DataKi:  52nMAssay Description:Displacement of [3H]Naltrindole from DOR in guinea pig brain membranesMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetOpioid receptor delta 1(Bos taurus)
University Of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM81934(Beta-Endorphin)
Affinity DataKi:  58.1nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOpioid receptor delta 1(Bos taurus)
University Of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  63nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOpioid receptor delta 1(Bos taurus)
University Of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  73nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOpioid receptor delta 1(Bos taurus)
University Of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM86258(CAS_23552-18-3 | Morphine | NSC_5980)
Affinity DataKi:  278nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOpioid receptor delta 1(Bos taurus)
University Of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM50139013((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in calf frontal cortex after 1 hr by gamma counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOpioid receptor delta 1(Bos taurus)
University Of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM50106276(1-[2-Amino-3-(4-hydroxy-phenyl)-propionyl]-pyrroli...)
Affinity DataKi:  500nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetOpioid receptor delta 1(Bos taurus)
University Of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM86518(CAS_509-60-4 | DIHYDROMORPHINE | NSC_273032)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOpioid receptor delta 1(Bos taurus)
University Of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM86519(CAS_11221 | Dihydroheroin | NSC_11221)
Affinity DataKi:  2.47E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOpioid receptor delta 1(Bos taurus)
University Of Rochester

Curated by PDSP Ki Database
LigandPNGBDBM86757(CAS_0 | NSC_11603174 | [11C]MMP)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOpioid receptor delta 1(Cavia porcellus)
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50268462(CHEMBL506616 | c[L-Phe-D-pro-L-Phe-L-trp])
Affinity DataIC50:  2.60E+3nMAssay Description:Displacement of [3H]DPDPE from delta-opioid receptor in guinea pig brain membranes after 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed