TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 0.140nMAssay Description:Displacement of [3H]-PDBU from protein kinase C-alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Bos taurus (bovine))
National Cancer Institute-Frederick
Curated by ChEMBL
National Cancer Institute-Frederick
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Ability to displace bound [20-3H]-PDBU from a recombinant single isozyme (PKCalpha) in the presence of phosphatidylserineMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 0.200nMAssay Description:Binding Affinity against protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 0.260nMAssay Description:Inhibition of [3H]PDBu binding to PKCalpha C1A domainMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 0.400nMAssay Description:Inhibition of [3H]PDBu binding to PKC alpha C1A peptideMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 0.480nMAssay Description:Inhibition of [20-3H]phorbol 12,13-dibutyrate binding to human PKCalpha by scintillation counting based poly(ethylene) glycol precipitation assayMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 0.5nMAssay Description:Displacement of [3H]- PDBu from recombinant PKC alpha expressed in baculovirusMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 0.540nMAssay Description:Displacement of [3H]-PDBU from protein kinase C-alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 0.780nMAssay Description:Binding affinity (Ki) towards Protein kinase CMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 0.930nMAssay Description:Inhibition of human Protein kinase C alpha with [Ca2+]More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 1nMAssay Description:Displacement of [3H]PDBu from PKCalpha C1A domain (unknown origin)More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 1nMAssay Description:Reversible competitive inhibition of PKCalpha (unknown origin)More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 1.20nMAssay Description:Affinity for protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 1.5nMAssay Description:Displacement of [20-3H]PDBu from recombinant PKC alpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]PDBu form PKCalphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 1.60nMAssay Description:Displacement of 3[H]PDBu from Protein kinase C alpha C1a domainMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Bos taurus (bovine))
National Cancer Institute-Frederick
Curated by ChEMBL
National Cancer Institute-Frederick
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant bovine Protein kinase C alpha in presence of [Ca2+]More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 1.80nMAssay Description:Affinity for protein kinase C alphaMore data for this Ligand-Target Pair
Affinity DataKi: 2.07nMAssay Description:Displacement of [3H]PDBu form mouse PKCalpha by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.07nMAssay Description:Displacement of [3H]PDBu form mouse PKCalpha by scintillation countingMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 2.30nMAssay Description:Binding Affinity against protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 2.30nMAssay Description:Affinity for protein kinase-C alpha (PK-C alpha)More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 2.30nMAssay Description:Displacement of [20-3H]-phorbol 12,13-dibutyrate (PDBU) from protein kinase C alpha with phosphatidylserineMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 2.30nMAssay Description:Affinity for protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Bos taurus (bovine))
National Cancer Institute-Frederick
Curated by ChEMBL
National Cancer Institute-Frederick
Curated by ChEMBL
Affinity DataKi: 2.40nMAssay Description:Tested for ability to displace [20e3] phorbol 12,13- dibutyrate binding from recombinant bovine Protein kinase C alpha in presence of [Ca2+]More data for this Ligand-Target Pair
Affinity DataKi: 2.45nMAssay Description:Displacement of [3H]PDBu form mouse PKCalpha by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.45nMAssay Description:Displacement of [3H]PDBu form mouse PKCalpha by scintillation countingMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 2.5nMAssay Description:Inhibition of [3H]-phorbol 12,13-dibutyrate (PDBu) binding to human recombinant protein kinase C alphaMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Displacement of [3H]PDBu form mouse PKCalpha by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Displacement of [3H]PDBu form mouse PKCalpha by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.66nMAssay Description:Displacement of [3H]PDBu form mouse PKCalpha by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.66nMAssay Description:Displacement of [3H]PDBu form mouse PKCalpha by scintillation countingMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 2.70nMAssay Description:Binding Affinity against protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 2.70nMAssay Description:Displacement of [20-3H]-PDBU ligand from recombinant protein kinase C (baculovirus)More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 2.80nMAssay Description:Displacement of [20-3H] phorbol 12, 13-dibutylate from recombinant PKCalpha (unknown origin) in presence of 100 ug/ml 100% phosphatidylserineMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Displacement of [3H]PDBu form mouse PKCalpha by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Displacement of [3H]PDBu form mouse PKCalpha by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Displacement of [3H]PDBu from mouse recombinant PKCalpha expressed in Escherichia coliMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 2.90nMAssay Description:Displacement of [20-3H]phorbol 12,13-dibutyrate from recombinant PKCalphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 2.90nMAssay Description:Binding affinity for Protein kinase C alpha C1a or C1b domainMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 2.90nMpH: 7.4Assay Description:Inhibition of [3H]PDBu binding to recombinant protein kinase C alpha was determined at pH 7.4, 37 degree C for 5 minMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 2.90nMAssay Description:Displacement of [20-3H]PDBu from recombinant PKC alpha in presence of phosphatidylserineMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 2.90nMAssay Description:Displacement of [20-3H]phorbol-12,13-dibutyrate (PDBu) from recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 2.90nMAssay Description:Binding Affinity against protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Homo sapiens (Human))
University Of Pittsburgh
Curated by PDSP Ki Database
University Of Pittsburgh
Curated by PDSP Ki Database
Affinity DataKi: 2.90nMAssay Description:Affinity for protein kinase-C alpha (PK-C alpha)More data for this Ligand-Target Pair