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Found 56 Enz. Inhib. hit(s) with Target = 'Sensory histidine kinase DcuS'
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151871(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]...)
Affinity DataIC50:  0.300nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151874(CHEMBL362838 | Tyr-Ser-Thr-cyclo(Cys-Ala-Phe-Ile-M...)
Affinity DataIC50:  0.300nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151880(CHEMBL426697 | YSTCYFIM)
Affinity DataIC50:  1nMAssay Description:Concentration required to antagonise accessory gene regulator C3 of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50526860(CHEMBL4554516)
Affinity DataIC50: <1nMAssay Description:Inhibition of AgrC in mid-exponential phase Staphylococcus aureus RN6390B assessed as beta-lactamase activity incubated for 80 mins by spectrophotome...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151876(CHEMBL182783 | GVNACSSLF)
Affinity DataIC50:  1nMAssay Description:Concentration required to antagonise accessory gene regulator C3 of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151873(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]...)
Affinity DataIC50:  2.80nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151876(CHEMBL182783 | GVNACSSLF)
Affinity DataIC50:  2.90nMAssay Description:Antagonistic concentration for accessory gene regulator C1 of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50020375(CHEMBL3289785)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of AgrC in mid-exponential phase Staphylococcus aureus RN6390B assessed as beta-lactamase activity incubated for 80 mins by spectrophotome...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50526861(CHEMBL2337554)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of AgrC in mid-exponential phase Staphylococcus aureus RN8463 assessed as beta-lactamase activity incubated for 80 mins by spectrophotomet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50020375(CHEMBL3289785)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of AgrC in mid-exponential phase Staphylococcus aureus RN8463 assessed as beta-lactamase activity incubated for 80 mins by spectrophotomet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50526861(CHEMBL2337554)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of AgrC in mid-exponential phase Staphylococcus aureus SA502A assessed as beta-lactamase activity incubated for 80 mins by spectrophotomet...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151880(CHEMBL426697 | YSTCYFIM)
Affinity DataIC50:  4nMAssay Description:Concentration required to antagonise accessory gene regulator C2 of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151877(CHEMBL182114 | N-[9-Benzyl-6-sec-butyl-12-methyl-3...)
Affinity DataIC50:  5nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151877(CHEMBL182114 | N-[9-Benzyl-6-sec-butyl-12-methyl-3...)
Affinity DataIC50:  5nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151879(2-{2-[2-(2-{2-[2-(2-Amino-3-methyl-pentanoylamino)...)
Affinity DataIC50:  6nMAssay Description:Concentration required to antagonise accessory gene regulator C2 of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50526859(CHEMBL4518791)
Affinity DataIC50:  7.90nMAssay Description:Inhibition of AgrC in mid-exponential phase Staphylococcus aureus RN6390B assessed as beta-lactamase activity incubated for 80 mins by spectrophotome...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151874(CHEMBL362838 | Tyr-Ser-Thr-cyclo(Cys-Ala-Phe-Ile-M...)
Affinity DataIC50:  8nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151871(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]...)
Affinity DataIC50:  10nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151871(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]...)
Affinity DataIC50:  10nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151883(CHEMBL276191 | N-[9-Benzyl-6-sec-butyl-12-methyl-3...)
Affinity DataIC50:  19nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151874(CHEMBL362838 | Tyr-Ser-Thr-cyclo(Cys-Ala-Phe-Ile-M...)
Affinity DataIC50:  21nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151874(CHEMBL362838 | Tyr-Ser-Thr-cyclo(Cys-Ala-Phe-Ile-M...)
Affinity DataIC50:  21nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151879(2-{2-[2-(2-{2-[2-(2-Amino-3-methyl-pentanoylamino)...)
Affinity DataIC50:  70nMAssay Description:Antagonistic concentration for accessory gene regulator C1 of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151876(CHEMBL182783 | GVNACSSLF)
Affinity DataIC50:  86nMAssay Description:Concentration required to antagonise accessory gene regulator C4 of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151873(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]...)
Affinity DataIC50:  137nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151879(2-{2-[2-(2-{2-[2-(2-Amino-3-methyl-pentanoylamino)...)
Affinity DataIC50:  150nMAssay Description:Concentration required to antagonise accessory gene regulator C4 of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151871(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]...)
Affinity DataIC50:  230nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151878(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]...)
Affinity DataIC50:  256nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151878(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]...)
Affinity DataIC50:  256nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151883(CHEMBL276191 | N-[9-Benzyl-6-sec-butyl-12-methyl-3...)
Affinity DataIC50:  295nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151872(2-{2-[4-(4-Benzoyl-phenoxy)-butyrylamino]-3-hydrox...)
Affinity DataIC50:  303nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151872(2-{2-[4-(4-Benzoyl-phenoxy)-butyrylamino]-3-hydrox...)
Affinity DataIC50:  303nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50406396(CHEMBL4159129)
Affinity DataIC50:  456nMAssay Description:Inhibition of AIP-stimulated quorum sensing system AgrC activation in Staphylococcus aureus RN10829 harboring P3:blaZ fusion assessed as reduction in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50406468(CHEMBL4169564)
Affinity DataIC50:  608nMAssay Description:Inhibition of AIP-stimulated quorum sensing system AgrC activation in Staphylococcus aureus RN10829 harboring P3:blaZ fusion assessed as reduction in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50406354(CHEMBL4169312)
Affinity DataIC50:  622nMAssay Description:Inhibition of AIP-stimulated quorum sensing system AgrC activation in Staphylococcus aureus RN10829 harboring P3:blaZ fusion assessed as reduction in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50406399(CHEMBL4161642)
Affinity DataIC50:  738nMAssay Description:Inhibition of AIP-stimulated quorum sensing system AgrC activation in Staphylococcus aureus RN10829 harboring P3:blaZ fusion assessed as reduction in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50406469(CHEMBL4174843)
Affinity DataIC50:  913nMAssay Description:Inhibition of AIP-stimulated quorum sensing system AgrC activation in Staphylococcus aureus RN10829 harboring P3:blaZ fusion assessed as reduction in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50406360(CHEMBL4167382)
Affinity DataIC50:  1.43E+3nMAssay Description:Inhibition of AIP-stimulated quorum sensing system AgrC activation in Staphylococcus aureus RN10829 harboring P3:blaZ fusion assessed as reduction in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151875(CHEMBL369309 | N-(3-Benzyl-9,12-bis-hydroxymethyl-...)
Affinity DataIC50:  4.00E+3nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151875(CHEMBL369309 | N-(3-Benzyl-9,12-bis-hydroxymethyl-...)
Affinity DataIC50:  4.00E+3nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151880(CHEMBL426697 | YSTCYFIM)
Affinity DataIC50:  7.00E+3nMAssay Description:Antagonistic concentration for accessory gene regulator C1 of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50151881(CHEMBL362839 | Cyclo(Ac-Cys-Asp-Phe-Ile-Met))
Affinity DataIC50:  8.00E+3nMAssay Description:Concentration required to inhibit quorum sensor of Staphylococcus aureusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50406270(CHEMBL4163103)
Affinity DataIC50:  1.91E+4nMAssay Description:Inhibition of AIP-stimulated quorum sensing system AgrC activation in Staphylococcus aureus RN10829 harboring P3:blaZ fusion assessed as reduction in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50406397(CHEMBL4162686)
Affinity DataIC50:  6.90E+4nMAssay Description:Inhibition of AIP-stimulated quorum sensing system AgrC activation in Staphylococcus aureus RN10829 harboring P3:blaZ fusion assessed as reduction in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50468034(CHEMBL4286992)
Affinity DataIC50:  1.40E+5nMAssay Description:Inhibition of recombinant Staphylococcus aureus AgrC autophosphorylation expressed in Escherichia coli BL21(DE3) preincubated for 15 mins followed by...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM76798((E)-1-[2,4-dihydroxy-3-[(2E)-6-hydroxy-3,7-dimethy...)
Affinity DataIC50:  3.39E+5nMAssay Description:Inhibition of recombinant Staphylococcus aureus AgrC autophosphorylation expressed in Escherichia coli BL21(DE3) preincubated for 15 mins followed by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50497019(CHEMBL3235588)
Affinity DataKd:  2.58E+5nMAssay Description:Binding affinity to AgrC in Staphylococcus aureus assessed as disruption of membrane dipole potential by di-8-ANEPPS fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50497020(CHEMBL3235590)
Affinity DataKd:  4.00E+3nMAssay Description:Binding affinity to AgrC in Staphylococcus aureus assessed as disruption of membrane dipole potential by di-8-ANEPPS fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50497021(CHEMBL3235597)
Affinity DataKd:  2.00E+3nMAssay Description:Binding affinity to AgrC in Staphylococcus aureus assessed as disruption of membrane dipole potential by di-8-ANEPPS fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSensory histidine kinase DcuS(Staphylococcus aureus)
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50497022(CHEMBL1213657)
Affinity DataKd:  2.22E+5nMAssay Description:Binding affinity to AgrC in Staphylococcus aureus assessed as disruption of membrane dipole potential by di-8-ANEPPS fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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