TargetSerine/threonine-protein kinase VRK1(Homo sapiens (Human))
Universidade Estadual De Campinas (Unicamp)
Curated by ChEMBL
Universidade Estadual De Campinas (Unicamp)
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of full length wild-type VRK1 (unknown origin) expressed in insect cells using ULight-Histone 3-Thr3 peptide as substrate incubated for 30...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase VRK1(Homo sapiens (Human))
Universidade Estadual De Campinas (Unicamp)
Curated by ChEMBL
Universidade Estadual De Campinas (Unicamp)
Curated by ChEMBL
Affinity DataIC50: 150nMAssay Description:Inhibition of full length wild-type VRK1 (unknown origin) expressed in insect cells using ULight-Histone 3-Thr3 peptide as substrate incubated for 30...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase VRK1(Homo sapiens (Human))
Universidade Estadual De Campinas (Unicamp)
Curated by ChEMBL
Universidade Estadual De Campinas (Unicamp)
Curated by ChEMBL
Affinity DataIC50: 260nMAssay Description:Inhibition of full length wild-type VRK1 (unknown origin) expressed in insect cells using ULight-Histone 3-Thr3 peptide as substrate incubated for 30...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase VRK1(Homo sapiens (Human))
Universidade Estadual De Campinas (Unicamp)
Curated by ChEMBL
Universidade Estadual De Campinas (Unicamp)
Curated by ChEMBL
Affinity DataIC50: 674nMAssay Description:Inhibition of full length wild-type VRK1 (unknown origin) expressed in insect cells using ULight-Histone 3-Thr3 peptide as substrate incubated for 30...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase VRK1(Homo sapiens (Human))
Universidade Estadual De Campinas (Unicamp)
Curated by ChEMBL
Universidade Estadual De Campinas (Unicamp)
Curated by ChEMBL
Affinity DataIC50: 743nMAssay Description:Inhibition of human VRK1 using KEAKEKRQEQIAKRRRLSSLRASTSKSGGSQK as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase VRK1(Homo sapiens (Human))
Universidade Estadual De Campinas (Unicamp)
Curated by ChEMBL
Universidade Estadual De Campinas (Unicamp)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human VRK1 using [KEAKEKRQEQIAKRRRLSSLRASTSKSGGSQK] as substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase VRK1(Homo sapiens (Human))
Universidade Estadual De Campinas (Unicamp)
Curated by ChEMBL
Universidade Estadual De Campinas (Unicamp)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human VRK1 in presence of 10 uM ATP by radiometric analysisMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase VRK1(Homo sapiens (Human))
Universidade Estadual De Campinas (Unicamp)
Curated by ChEMBL
Universidade Estadual De Campinas (Unicamp)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human VRK1More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase VRK1(Homo sapiens (Human))
Universidade Estadual De Campinas (Unicamp)
Curated by ChEMBL
Universidade Estadual De Campinas (Unicamp)
Curated by ChEMBL
Affinity DataIC50: 1.29E+5nMAssay Description:Inhibition of human VRK1More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase VRK1(Homo sapiens (Human))
Universidade Estadual De Campinas (Unicamp)
Curated by ChEMBL
Universidade Estadual De Campinas (Unicamp)
Curated by ChEMBL
Affinity DataKd: 190nMAssay Description:Binding affinity to recombinant full length N-terminal His-tagged VRK1 (unknown origin) (1 to 396 residues) expressed in Escherichia coli BL 21 DE3-R...More data for this Ligand-Target Pair