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Found 5 Enz. Inhib. hit(s) with Target = 'Solute carrier family 22 member 4'
TargetSolute carrier family 22 member 4(Rattus norvegicus)
Medical College Of Georgia

Curated by ChEMBL
LigandPNGBDBM35229(3-(10,11-dihydro-5H-dibenzo[b,f]azepin-5-yl)-N-met...)
Affinity DataIC50:  8.00E+4nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake in Octn1-HRPE cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 4(Rattus norvegicus)
Medical College Of Georgia

Curated by ChEMBL
LigandPNGBDBM50485565(CHEMBL465179)
Affinity DataIC50:  2.00E+5nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake in Octn1-HRPE cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 4(Rattus norvegicus)
Medical College Of Georgia

Curated by ChEMBL
LigandPNGBDBM39344(4-amino-N-[2-(diethylamino)ethyl]benzamide;hydroch...)
Affinity DataIC50:  1.00E+6nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake in Octn1-HRPE cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 4(Rattus norvegicus)
Medical College Of Georgia

Curated by ChEMBL
LigandPNGBDBM50149890(CHEMBL9324 | tetraethylammonium)
Affinity DataIC50:  1.00E+6nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake in Octn1-HRPE cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 22 member 4(Rattus norvegicus)
Medical College Of Georgia

Curated by ChEMBL
LigandPNGBDBM50103595(Brumetadina | CHEBI:3699 | Cimetidine | Tagamet | ...)
Affinity DataIC50:  1.50E+6nMAssay Description:TP_TRANSPORTER: inhibition of TEA uptake in Octn1-HRPE cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed