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Found 52 Enz. Inhib. hit(s) with Target = 'Transcriptional regulator ERG'
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417421(CHEMBL1290597)
Affinity DataKi:  794nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417418(CHEMBL1289617)
Affinity DataKi:  1.26E+3nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417417(CHEMBL1289509)
Affinity DataKi:  1.58E+3nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417426(CHEMBL1289721)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413549(CHEMBL513715)
Affinity DataKi:  2.51E+3nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417414(CHEMBL1289276)
Affinity DataKi:  2.51E+3nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417419(CHEMBL1289618)
Affinity DataKi:  2.51E+3nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417420(CHEMBL1290486)
Affinity DataKi:  3.16E+3nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417409(CHEMBL1290487)
Affinity DataKi:  3.98E+3nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50413550(CHEMBL469345)
Affinity DataKi:  3.98E+3nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417410(CHEMBL1290596)
Affinity DataKi:  3.98E+3nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417422(CHEMBL1289048)
Affinity DataKi:  3.98E+3nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417416(CHEMBL1287827)
Affinity DataKi:  5.01E+3nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417423(CHEMBL1289164)
Affinity DataKi:  5.01E+3nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417425(CHEMBL1289510)
Affinity DataKi:  6.31E+3nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417415(CHEMBL1289277)
Affinity DataKi:  7.94E+3nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417424(CHEMBL1289394)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417427(CHEMBL1290716)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417412(CHEMBL1289047)
Affinity DataKi:  2.51E+4nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417413(CHEMBL1289163)
Affinity DataKi:  3.16E+4nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417411(CHEMBL1290715)
Affinity DataKi: >3.16E+4nMAssay Description:Displacement of [3H]-dofetilide in human ERG expressed in CHO cells by proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50003336(CHEMBL3234565)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50003076(CHEMBL3234574)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50003334(CHEMBL3234564)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50003407(CHEMBL3234568)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50003477(CHEMBL3234569)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50003286(CHEMBL3234576)
Affinity DataIC50:  5.50E+3nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50003289(CHEMBL3234578)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50003287(CHEMBL3234577)
Affinity DataIC50:  9.80E+3nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50352421(CHEMBL1823591)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM251922(US10065961, Compound 22 | US10683295, Compound 22 ...)
Affinity DataIC50:  1.20E+4nMAssay Description:The human Ether-a-go-go Related Gene (hERG) encodes the inward rectifying voltage gated potassium channel in the heart (IKr) which is involved in car...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50003283(CHEMBL3234575)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50420920(CHEMBL2087549 | CHEMBL2087567)
Affinity DataIC50:  1.63E+4nMAssay Description:Inhibition of human ERG channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50081399(CHEMBL3422016 | US10065961, Compound 19 | US106832...)
Affinity DataIC50:  1.70E+4nMAssay Description:The human Ether-a-go-go Related Gene (hERG) encodes the inward rectifying voltage gated potassium channel in the heart (IKr) which is involved in car...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50003563(CHEMBL3234573)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50003562(CHEMBL3234572)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM251928(US10065961, Compound 31 | US10683295, Compound 31 ...)
Affinity DataIC50:  2.00E+4nMAssay Description:The human Ether-a-go-go Related Gene (hERG) encodes the inward rectifying voltage gated potassium channel in the heart (IKr) which is involved in car...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50003561(CHEMBL3234571)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM251927(US10065961, Compound 29 | US10683295, Compound 29 ...)
Affinity DataIC50:  2.50E+4nMAssay Description:The human Ether-a-go-go Related Gene (hERG) encodes the inward rectifying voltage gated potassium channel in the heart (IKr) which is involved in car...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50081363(CHEMBL3422012 | US10065961, Compound 3 | US1068329...)
Affinity DataIC50:  2.60E+4nMAssay Description:The human Ether-a-go-go Related Gene (hERG) encodes the inward rectifying voltage gated potassium channel in the heart (IKr) which is involved in car...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50352420(CHEMBL1823865)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM251905(US10065961, Compound 2 | US10683295, Compound 2 | ...)
Affinity DataIC50: >3.00E+4nMAssay Description:The human Ether-a-go-go Related Gene (hERG) encodes the inward rectifying voltage gated potassium channel in the heart (IKr) which is involved in car...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50003559(CHEMBL3234570)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50081195(CHEMBL3422010 | US10065961, Compound 1 | US1068329...)
Affinity DataIC50: >3.00E+4nMAssay Description:The human Ether-a-go-go Related Gene (hERG) encodes the inward rectifying voltage gated potassium channel in the heart (IKr) which is involved in car...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50003291(CHEMBL3234579)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50352296(CHEMBL1822468)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM251906(US10065961, Compound 4 | US10683295, Compound 4 | ...)
Affinity DataIC50: >3.00E+4nMAssay Description:The human Ether-a-go-go Related Gene (hERG) encodes the inward rectifying voltage gated potassium channel in the heart (IKr) which is involved in car...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM251913(US10065961, Compound 11 | US10683295, Compound 11 ...)
Affinity DataIC50: >3.00E+4nMAssay Description:The human Ether-a-go-go Related Gene (hERG) encodes the inward rectifying voltage gated potassium channel in the heart (IKr) which is involved in car...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50003573(CHEMBL3234871)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human ERG by patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscriptional regulator ERG(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50352422(CHEMBL1823616)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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