Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily V member 5'
TargetTransient receptor potential cation channel subfamily V member 5(Homo sapiens)
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50550078(CHEMBL4777551)
Affinity DataIC50:  560nMAssay Description:Inhibition of human TRPV5 expressed in HEK293 cells assessed as reduction in Cd2+ influx by calcium-5 fluorescence dye-based FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 5(Homo sapiens)
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50511105(GWP-42004 | Gwp42004 | O-4394 | THCV | Tetrahydroc...)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of TRPV5 channel (unknown origin) by Patch-clamp assayMore data for this Ligand-Target Pair
In DepthDetails PubMed