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Found 91 Enz. Inhib. hit(s) with Target = 'ADP-ribosylation factor GTPase-activating protein 1'
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM94663((6Z)-6-[[5-(3-chlorophenyl)-2-furanyl]methylidene]...)
Affinity DataIC50: >2.03E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM94657(5-amino-N-(5-chloro-2-methoxy-phenyl)-1-[2-keto-2-...)
Affinity DataIC50:  5.04E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM43208(4-benzyl-N-[5-(2,3-dihydro-1,4-benzodioxin-6-yl)-1...)
Affinity DataIC50:  7.92E+3nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM94686(MLS000687260 | N'-[(E)-(4-benzoxybenzylidene)amino...)
Affinity DataIC50:  1.03E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM94655(2-[2-(2,6-dimethylmorpholin-4-yl)-2-oxidanylidene-...)
Affinity DataIC50:  1.07E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM94665(MLS001230224 | N-[(Z)-[4-methoxy-3-[(2,3,5,6-tetra...)
Affinity DataIC50:  1.24E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM40968(7-methyl-N-piperonyl-furo[2,3-b]quinoline-2-carbox...)
Affinity DataIC50:  1.67E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM94683(MLS000698868 | N-(4-aminocarbonylphenyl)-5-[(4-met...)
Affinity DataIC50:  1.67E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM94681(1-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-2-[1-(2,4-di...)
Affinity DataIC50:  1.77E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95208(2-(5-amino-1-tetrazolyl)-N-[(E)-[5-(2,5-dimethyl-4...)
Affinity DataIC50:  1.78E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM41086(MLS000582064 | N-[3-chloranyl-4-(2-oxidanylidenech...)
Affinity DataIC50:  1.79E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95229(MLS001234985 | N-(3-chlorophenyl)-2-(7-methyl-4-ox...)
Affinity DataIC50: >1.83E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95242(MLS003123272 | N-[2-(dimethylamino)ethyl]-4-[3-(4-...)
Affinity DataIC50: >1.83E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM67822(1-[2-(2,4-dichlorophenoxy)ethyl]-3-methyl-1,3-dihy...)
Affinity DataIC50:  1.84E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95203((E)-3-[1-phenyl-3-(p-tolyl)pyrazol-4-yl]-N-thiazol...)
Affinity DataIC50:  2.03E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM94694(1,3-benzodioxole-5-carboxylic acid [2-methoxy-4-[(...)
Affinity DataIC50:  2.10E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM41188(MLS000111800 | SMR000107719 | cid_2909321)
Affinity DataIC50:  2.31E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM94689(2-[2-(azepan-1-yl)-2-oxidanylidene-ethyl]sulfanyl-...)
Affinity DataIC50:  2.31E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM88864(2-(2,4-Dichloro-benzylsulfanyl)-6,7,8,9-tetrahydro...)
Affinity DataIC50:  2.38E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM94700(1,3-bis(o-anisylideneamino)urea | 1,3-bis[(2-metho...)
Affinity DataIC50:  2.56E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM94705(2-[[2-keto-2-(4-methylpiperidino)ethyl]thio]-7-met...)
Affinity DataIC50:  2.62E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM94693(2-[2-(4-benzylpiperidin-1-yl)-2-oxoethyl]sulfanyl-...)
Affinity DataIC50:  2.69E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95200(2-[4-[(Z)-(2-amino-4-keto-2-thiazolin-5-ylidene)me...)
Affinity DataIC50:  2.83E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95236(1-methyl-3-indolecarboxylic acid [2-(3,5-dimethyl-...)
Affinity DataIC50:  2.84E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM94697(2-(2-furanyl)-6-[2-oxo-2-(1-piperidinyl)ethoxy]-1-...)
Affinity DataIC50:  2.85E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95211(MLS000621169 | N-(2,3-dimethylphenyl)-2-(4-ketoben...)
Affinity DataIC50:  2.87E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM55790((E)-3-phenyl-N-(4-pyridin-4-yl-1,3-thiazol-2-yl)pr...)
Affinity DataIC50:  2.88E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM54212(MLS000326804 | N'-[(2,6-dichlorobenzyl)oxy]-N-...)
Affinity DataIC50:  3.03E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95204(4-[(2-keto-4-methyl-chromen-7-yl)oxymethyl]benzoic...)
Affinity DataIC50:  3.13E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM94669(2-[(2-keto-2-piperidino-ethyl)thio]-7-methyl-pyrid...)
Affinity DataIC50:  3.20E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM67993((Z)-3-(1,3-diphenyl-4-pyrazolyl)-N-(2-thiazolyl)-2...)
Affinity DataIC50:  3.21E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM48131(1H-indazole-3-carboxylic acid [2-keto-2-(1,2,5-tri...)
Affinity DataIC50:  3.24E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95241(MLS001125783 | N-[2-methoxy-4-[2-(4-nitrophenoxy)e...)
Affinity DataIC50:  3.36E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95224(MLS001146387 | N-[(E)-[3-(4-bromobenzyl)-4-chloro-...)
Affinity DataIC50:  3.43E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95225(1-(3,4-dimethylphenyl)-3-[2-(4-nitrophenoxy)ethano...)
Affinity DataIC50:  3.45E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM94673(5-bromanyl-N-(2-methoxy-5-nitro-phenyl)thiophene-2...)
Affinity DataIC50:  3.56E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM94668(4-acetamido-N-(4-pyridin-3-yl-1,3-thiazol-2-yl)ben...)
Affinity DataIC50:  3.66E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM28655(2-(5-butoxy-1-oxo-1,2-dihydroisoquinolin-2-yl)-N-(...)
Affinity DataIC50:  3.68E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM34388(MLS000085595 | N-[5-(4-chlorophenyl)-1,2,4-thiadia...)
Affinity DataIC50:  3.76E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM94706(MLS000830253 | SMR000034292 | cid_658947)
Affinity DataIC50:  3.81E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95214(3-(2-Pyridin-3-yl-quinazolin-4-ylamino)-benzoic ac...)
Affinity DataIC50:  3.83E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95217(1-[2-(4-methoxyphenyl)-3,4-dimethyl-7-pyrazolo[3,4...)
Affinity DataIC50:  4.06E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95209(MLS000687875 | N-[4-[2-[[1-(2,3-dihydro-1,4-benzod...)
Affinity DataIC50:  4.07E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95198(Benzo[1,3]dioxole-5-carboxylic acid [4-(1H-benzoim...)
Affinity DataIC50:  4.20E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95215(4-[[(2,5,6-trimethyl-4-thieno[2,3-d]pyrimidinyl)am...)
Affinity DataIC50:  4.25E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM43011(2-(6-Amino-3,5-dicyano-4-thiophen-2-yl-pyridin-2-y...)
Affinity DataIC50:  4.32E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95201(3-(2-Chloro-6-fluoro-phenyl)-4,5-dihydro-isoxazole...)
Affinity DataIC50:  4.36E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM40512(2-({3-[2-(3,4-dimethoxyphenyl)ethyl]-4-oxo-3,4-dih...)
Affinity DataIC50:  4.40E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95230(MLS001234953 | N-(3-fluorophenyl)-2-(7-methyl-4-ox...)
Affinity DataIC50:  4.49E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetADP-ribosylation factor GTPase-activating protein 1(Rattus norvegicus)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM95233(5-methoxy-3-methyl-2-benzofurancarboxylic acid [2-...)
Affinity DataIC50:  4.49E+4nMMore data for this Ligand-Target Pair
In DepthDetails PCBioAssay
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