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Found 971 Enz. Inhib. hit(s) with Target = 'Cysteine protease'
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50509389(CHEMBL4566436)
Affinity DataKi:  0.000600nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris assessed as inhibition constant measured for 30 mins using Cbz-Ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50509387(CHEMBL4475066)
Affinity DataKi:  0.00110nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris assessed as inhibition constant measured for 30 mins using Cbz-Ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50509386(CHEMBL4515298)
Affinity DataKi:  0.00300nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris assessed as inhibition constant measured for 30 mins using Cbz-Ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50509388(CHEMBL4587965)
Affinity DataKi:  0.00440nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris assessed as inhibition constant measured for 30 mins using Cbz-Ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50509383(CHEMBL4441635)
Affinity DataKi:  0.00760nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris assessed as inhibition constant measured for 30 mins using Cbz-Ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50509390(CHEMBL4436812)
Affinity DataKi:  0.0150nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris assessed as inhibition constant measured for 30 mins using Cbz-Ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50509381(CHEMBL4453415)
Affinity DataKi:  0.0230nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris assessed as inhibition constant measured for 30 mins using Cbz-Ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50509394(CHEMBL4584291)
Affinity DataKi:  0.0290nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris assessed as inhibition constant measured for 30 mins using Cbz-Ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50509395(CHEMBL4437914)
Affinity DataKi:  0.0340nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris assessed as inhibition constant measured for 30 mins using Cbz-Ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50258507(CHEMBL4078345)
Affinity DataKi:  0.0380nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris using Cbz-Phe-Arg-AMC as substrate after 30 min by fl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50258514(CHEMBL4062015)
Affinity DataKi:  0.0740nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris using Cbz-Phe-Arg-AMC as substrate after 30 min by fl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50594411(CHEMBL5173102)
Affinity DataKi:  0.150nMAssay Description:Binding affinity to recombinant Trypanosoma brucei rhodesiense rhodesain assessed as inhibition constant using Cbz-Phe-Arg-AMC as fluorogenic substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50594420(CHEMBL5200091)
Affinity DataKi:  0.420nMAssay Description:Binding affinity to recombinant Trypanosoma brucei rhodesiense rhodesain assessed as inhibition constant using Cbz-Phe-Arg-AMC as fluorogenic substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50574836(CHEMBL4871105)
Affinity DataKi:  0.450nMAssay Description:Inhibition of Trypanosoma brucei rhodesain assessed as fluorescence using Cbz-Phe-Arg-AMC as substrate measured at second inhibition step by fluorome...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50201259(CHEMBL3907022)
Affinity DataKi:  0.490nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris using Cbz-Phe-Arg-AMC as substrate after 15 to 30 mins by fluores...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50568077(CHEMBL4865195)
Affinity DataKi:  0.5nMAssay Description:Binding affinity to Trypanosoma brucei rhodesainMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50258506(CHEMBL4072275)
Affinity DataKi:  0.5nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris using Cbz-Phe-Arg-AMC as substrate after 30 min by fl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50509391(CHEMBL4459413)
Affinity DataKi:  0.5nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris assessed as inhibition constant measured for 30 mins using Cbz-Ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50594417(CHEMBL5170687)
Affinity DataKi:  0.510nMAssay Description:Binding affinity to recombinant Trypanosoma brucei rhodesiense rhodesain assessed as inhibition constant using Cbz-Phe-Arg-AMC as fluorogenic substra...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50594413(CHEMBL5209133)
Affinity DataKi:  0.510nMAssay Description:Binding affinity to recombinant Trypanosoma brucei rhodesiense rhodesain assessed as inhibition constant using Cbz-Phe-Arg-AMC as fluorogenic substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50509392(CHEMBL4456010)
Affinity DataKi:  0.740nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris assessed as inhibition constant measured for 30 mins using Cbz-Ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50594416(CHEMBL5207517)
Affinity DataKi:  0.780nMAssay Description:Binding affinity to recombinant Trypanosoma brucei rhodesiense rhodesain assessed as inhibition constant using Cbz-Phe-Arg-AMC as fluorogenic substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50594414(CHEMBL5186393)
Affinity DataKi:  0.850nMAssay Description:Binding affinity to recombinant Trypanosoma brucei rhodesiense rhodesain assessed as inhibition constant using Cbz-Phe-Arg-AMC as fluorogenic substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50258544(CHEMBL4096388)
Affinity DataKi:  0.900nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris using Cbz-Phe-Arg-AMC as substrate after 30 min by fl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50594421(CHEMBL5190766)
Affinity DataKi:  0.930nMAssay Description:Binding affinity to recombinant Trypanosoma brucei rhodesiense rhodesain assessed as inhibition constant using Cbz-Phe-Arg-AMC as fluorogenic substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50594418(CHEMBL5205818)
Affinity DataKi:  1nMAssay Description:Binding affinity to recombinant Trypanosoma brucei rhodesiense rhodesain assessed as inhibition constant using Cbz-Phe-Arg-AMC as fluorogenic substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50263570(CHEMBL4066422)
Affinity DataKi:  1nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain using Cbz-Phe-Arg-AMC as substrate by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50594415(CHEMBL5176432)
Affinity DataKi:  1.10nMAssay Description:Binding affinity to recombinant Trypanosoma brucei rhodesiense rhodesain assessed as inhibition constant using Cbz-Phe-Arg-AMC as fluorogenic substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50594412(CHEMBL5175052)
Affinity DataKi:  1.10nMAssay Description:Binding affinity to recombinant Trypanosoma brucei rhodesiense rhodesain assessed as inhibition constant using Cbz-Phe-Arg-AMC as fluorogenic substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50574837(CHEMBL4855902)
Affinity DataKi:  1.5nMAssay Description:Inhibition of Trypanosoma brucei rhodesain assessed as fluorescence using Cbz-Phe-Arg-AMC as substrate measured at second inhibition step by fluorome...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50509384(CHEMBL4456727)
Affinity DataKi:  1.80nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris assessed as inhibition constant measured for 30 mins using Cbz-Ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50258542(CHEMBL4082758)
Affinity DataKi:  2nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris using Cbz-Phe-Arg-AMC as substrate after 30 min by fl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50263634(CHEMBL4073014)
Affinity DataKi:  2nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain using Cbz-Phe-Arg-AMC as substrate by fluorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50263572(CHEMBL4092050)
Affinity DataKi:  2nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain using Cbz-Phe-Arg-AMC as substrate by fluorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50505323(CHEMBL4556848)
Affinity DataKi:  2nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesainMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50509385(CHEMBL4454883)
Affinity DataKi:  2.10nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris assessed as inhibition constant measured for 30 mins using Cbz-Ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM210854(US9290467, 24 | US9290467, 25 | US9290467, 26)
Affinity DataKi:  2.5nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain using Cbz-Phe-Arg-AMC as substrate by fluorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50594419(CHEMBL5198708)
Affinity DataKi:  2.5nMAssay Description:Binding affinity to recombinant Trypanosoma brucei rhodesiense rhodesain assessed as inhibition constant using Cbz-Phe-Arg-AMC as fluorogenic substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50322349((R)-Methyl4-(2-(3-((adamantan-1-ylcarbamoyloxy)met...)
Affinity DataKi:  2.60nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50322349((R)-Methyl4-(2-(3-((adamantan-1-ylcarbamoyloxy)met...)
Affinity DataKi:  2.60nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50263632(CHEMBL4080286)
Affinity DataKi:  2.90nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain using Cbz-Phe-Arg-AMC as substrate by fluorimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50574818(CHEMBL4861941)
Affinity DataKi:  3nMAssay Description:Inhibition of Trypanosoma brucei rhodesain assessed as fluorescence using Cbz-Phe-Arg-AMC as substrate measured using Dixon equation by fluorometric ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50263647(CHEMBL4099905)
Affinity DataKi:  3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain using Cbz-Phe-Arg-AMC as substrate by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50263571(CHEMBL4062591)
Affinity DataKi:  3nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain using Cbz-Phe-Arg-AMC as substrate by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50509382(CHEMBL4464737)
Affinity DataKi:  3.10nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris assessed as inhibition constant measured for 30 mins using Cbz-Ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50258500(CHEMBL4093034)
Affinity DataKi:  3.60nMAssay Description:Inhibition of recombinant Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris using Cbz-Phe-Arg-AMC as substrate after 30 min by fl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50263689(CHEMBL4064430)
Affinity DataKi:  4nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain using Cbz-Phe-Arg-AMC as substrate by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50201212(CHEMBL3974129)
Affinity DataKi:  4.20nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain expressed in Pichia pastoris using Cbz-Phe-Arg-AMC as substrate after 15 to 30 mins by fluores...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50263573(CHEMBL4080708)
Affinity DataKi:  4.80nMAssay Description:Agonist activity at human SP/Myc epitope-tagged muscarinic M1 receptor expressed in HEK293T cells assessed as RLuc8-fused Galphaq activation after 2 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteine protease(Trypanosoma brucei rhodesiense)
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50263573(CHEMBL4080708)
Affinity DataKi:  4.80nMAssay Description:Inhibition of Trypanosoma brucei rhodesiense rhodesain using Cbz-Phe-Arg-AMC as substrate by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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