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Found 2366 Enz. Inhib. hit(s) with Target = 'Endothelin receptor type B'
TargetEndothelin receptor type B(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50000558(CHEMBL437472 | ET-1 | Endothelin -1 | Endothelin 1...)
Affinity DataKi:  0.00800nMAssay Description:Ability to inhibit [125I]ET-3 binding to the Endothelin B receptor from porcine lung membranes was evaluatedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000558(CHEMBL437472 | ET-1 | Endothelin -1 | Endothelin 1...)
Affinity DataKi:  0.0100nMAssay Description:Compound was evaluated for the binding affinity to Endothelin B receptor in the rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368606(Sarafotoxin S6B)
Affinity DataKi:  0.0120nMAssay Description:Compound was evaluated for the binding affinity to Endothelin B receptor in the rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368606(Sarafotoxin S6B)
Affinity DataKi:  0.0130nMAssay Description:Compound was evaluated for the binding affinity to Endothelin B receptor in the rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50000558(CHEMBL437472 | ET-1 | Endothelin -1 | Endothelin 1...)
Affinity DataKi:  0.0150nMAssay Description:Compound was evaluated for the binding affinity to Endothelin B receptor in the rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368605(CHEMBL1790178)
Affinity DataKi:  0.0160nMAssay Description:Compound was evaluated for the binding affinity to Endothelin B receptor in the rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368607(CHEMBL1790180)
Affinity DataKi:  0.0210nMAssay Description:Compound was evaluated for the binding affinity to Endothelin B receptor in the rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368605(CHEMBL1790178)
Affinity DataKi:  0.0230nMAssay Description:Compound was evaluated for the binding affinity to Endothelin B receptor in the rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50368607(CHEMBL1790180)
Affinity DataKi:  0.0360nMAssay Description:Compound was evaluated for the binding affinity to Endothelin B receptor in the rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50287890(CHEMBL427778 | Suc-Glu-Ala-Val-Tyr-Phe-Ala-His-Leu...)
Affinity DataKi:  0.0770nMAssay Description:Ability to inhibit [125I]ET-3 binding to the Endothelin B receptor from porcine lung membranes was evaluatedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Homo sapiens (Human))
Banyu Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50143784((5S,6R,7R)-5-Benzo[1,3]dioxol-5-yl-2-butyl-7-[2-((...)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Banyu Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50071445(CHEMBL310039 | N-[(R)-1-[(S)-2-Ethenesulfonylamino...)
Affinity DataKi:  0.140nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Banyu Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50071438((S)-2-[(R)-2-[(3,5-Dimethyl-benzoyl)-methyl-amino]...)
Affinity DataKi:  0.210nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Banyu Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50071435((S)-2-[(R)-2-[(3,5-Dimethyl-benzoyl)-methyl-amino]...)
Affinity DataKi:  0.230nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Banyu Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50071437(CHEMBL308102 | N-[(R)-1-[(S)-1-(1H-Indol-3-ylmethy...)
Affinity DataKi:  0.230nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Banyu Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50071423(CHEMBL72924 | N-[(R)-1-[(S)-2-(2-Ethoxy-ethanesulf...)
Affinity DataKi:  0.230nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Banyu Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50071420(CHEMBL72348 | N-[(R)-1-[(S)-1-(1H-Indol-3-ylmethyl...)
Affinity DataKi:  0.240nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Banyu Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50071436(CHEMBL306950 | N-[(R)-1-[(S)-2-(Butane-1-sulfonyla...)
Affinity DataKi:  0.240nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50287885(CHEMBL405377 | Suc-Glu-Ala-Val-Tyr-Phe-Ala-His-Leu...)
Affinity DataKi:  0.25nMAssay Description:Ability to inhibit [125I]ET-3 binding to the Endothelin B receptor from porcine lung membranes was evaluatedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Homo sapiens (Human))
Banyu Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50071421(CHEMBL310920 | N-[(R)-1-[(S)-2-Benzenesulfonylamin...)
Affinity DataKi:  0.340nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Banyu Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50071439(CHEMBL73000 | N-[(R)-1-[(S)-1-(1H-Indol-3-ylmethyl...)
Affinity DataKi:  0.380nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Banyu Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50071430(CHEMBL73373 | N-[(R)-1-[(S)-2-Ethanesulfonylamino-...)
Affinity DataKi:  0.380nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Banyu Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50071428(CHEMBL307471 | N-[(R)-1-{(S)-1-(1H-Indol-3-ylmethy...)
Affinity DataKi:  0.390nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Banyu Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50071444(CHEMBL307045 | N-[(R)-1-[1-(Butane-1-sulfonylamino...)
Affinity DataKi:  0.490nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Banyu Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50071443(CHEMBL308269 | N-[(R)-1-[(S)-1-(1H-Indol-3-ylmethy...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Banyu Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50071440(CHEMBL307384 | N-[(R)-1-[2-(Butane-1-sulfonylamino...)
Affinity DataKi:  0.590nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Banyu Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50071432((S)-2-[(R)-2-[(3,5-Dimethyl-benzoyl)-methyl-amino]...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Banyu Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50071426(CHEMBL73835 | N-[(R)-1-[1-(Butane-1-sulfonylaminoc...)
Affinity DataKi:  0.700nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Banyu Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50071441((S)-2-[(R)-2-[(3,5-Dimethyl-benzoyl)-methyl-amino]...)
Affinity DataKi:  0.760nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Banyu Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50071427((S)-2-[(R)-2-[(3,5-Dimethyl-benzoyl)-methyl-amino]...)
Affinity DataKi:  0.790nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50287883(CHEMBL412003 | Suc-Glu-Ala-Gly-Tyr-Phe-Ala-His-Leu...)
Affinity DataKi:  0.910nMAssay Description:Ability to inhibit [125I]ET-3 binding to the Endothelin B receptor from porcine lung membranes was evaluatedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50071433((S)-2-{(R)-3-Biphenyl-4-yl-2-[(3,5-dimethyl-benzoy...)
Affinity DataKi:  1nMAssay Description:Ability to inhibit [125I]ET-3 binding to the Endothelin B receptor from porcine lung membranes was evaluatedMore data for this Ligand-Target Pair
TargetEndothelin receptor type B(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50287882(CHEMBL412065 | Suc-Glu-Ala-Val-Tyr-Phe-Ala-Gly-Leu...)
Affinity DataKi:  1nMAssay Description:Ability to inhibit [125I]ET-3 binding to the Endothelin B receptor from porcine lung membranes was evaluatedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Homo sapiens (Human))
Banyu Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50071433((S)-2-{(R)-3-Biphenyl-4-yl-2-[(3,5-dimethyl-benzoy...)
Affinity DataKi:  1nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
TargetEndothelin receptor type B(Homo sapiens (Human))
Banyu Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50071425(CHEMBL311854 | N-[(R)-1-[(S)-1-(Butane-1-sulfonyla...)
Affinity DataKi:  1.20nMAssay Description:Compound was tested for the binding affinity against Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Banyu Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50071425(CHEMBL311854 | N-[(R)-1-[(S)-1-(Butane-1-sulfonyla...)
Affinity DataKi:  1.20nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Mus musculus)
University Hospital M£Nster

Curated by ChEMBL
LigandPNGBDBM50304497(2-(5-{[4-(Benzo[1,3]dioxol-5-yl)-2-hydroxy-2-(4-me...)
Affinity DataKi:  1.26nMAssay Description:Displacement of [125I]ET1 from endothelin B receptor in DBA mouse microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Banyu Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50071434(CHEMBL72217 | N-[(R)-1-[1-(Butane-1-sulfonylaminoc...)
Affinity DataKi:  1.30nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Banyu Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50071442(CHEMBL72358 | N-[(R)-1-[2-(Butane-1-sulfonylamino)...)
Affinity DataKi:  3.10nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Banyu Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50071424(CHEMBL263301 | N-[(R)-1-[1-(Butane-1-sulfonylamino...)
Affinity DataKi:  3.20nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Banyu Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50079426(2-(4,6-Dimethyl-pyrimidin-2-yloxy)-3,3-diphenyl-3-...)
Affinity DataKi:  3.21nMAssay Description:Inhibition of [125I]-ET-3 (ETB assay) binding to human cloned Endothelin B receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Banyu Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50071422(CHEMBL73042 | N-[(R)-1-[1-(Butane-1-sulfonylaminoc...)
Affinity DataKi:  3.5nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Banyu Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50071429((S)-2-[(R)-2-[(3,5-Dimethyl-benzoyl)-methyl-amino]...)
Affinity DataKi:  4.40nMAssay Description:Binding affinity to Endothelin B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Banyu Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50079424((S)-3-[2-(3,4-Dimethoxy-phenyl)-ethoxy]-2-(4,6-dim...)
Affinity DataKi:  4.75nMAssay Description:Inhibition of [125I]-ET-3 (ETB assay) binding to human cloned Endothelin B receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Banyu Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50079424((S)-3-[2-(3,4-Dimethoxy-phenyl)-ethoxy]-2-(4,6-dim...)
Affinity DataKi:  4.80nMAssay Description:Displacement of [125I]ET-3 from human ET-B receptor expressed in CHO cell membrane incubated for 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50287878(CGP-49941 | CHEMBL305615 | N-{(R)-1-[2-(1H-Indol-3...)
Affinity DataKi:  5nMAssay Description:Ability to inhibit [125I]ET-3 binding to the Endothelin B receptor from porcine lung membranes was evaluatedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50287888(CHEMBL407559 | Suc-Glu-Ala-Val-Tyr-Phe-Gly-His-Leu...)
Affinity DataKi:  5.30nMAssay Description:Ability to inhibit [125I]ET-3 binding to the Endothelin B receptor from porcine lung membranes was evaluatedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Homo sapiens (Human))
Banyu Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50050964(4-[1-Benzo[1,3]dioxol-5-yl-2-(4-isopropyl-benzenes...)
Affinity DataKi:  5.40nMAssay Description:Inhibitory activity of the compound against human Endothelin B receptor in chinese hamster ovary cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Sus scrofa)
TBA

Curated by ChEMBL
LigandPNGBDBM50287886(CHEMBL405796 | Suc-Glu-Ala-Val-Tyr-Phe-Ala-His-Gly...)
Affinity DataKi:  5.90nMAssay Description:Ability to inhibit [125I]ET-3 binding to the Endothelin B receptor from porcine lung membranes was evaluatedMore data for this Ligand-Target Pair
In DepthDetails Article
TargetEndothelin receptor type B(Homo sapiens (Human))
Banyu Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50079417(3-[2-(3,4-Dimethoxy-phenyl)-ethoxy]-2-(4,6-dimethy...)
Affinity DataKi:  7.15nMAssay Description:Inhibition of [125I]-ET-3 (ETB assay) binding to human cloned Endothelin B receptor in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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