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Found 168 Enz. Inhib. hit(s) with Target = 'Protein Tat'
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50097337(CHEMBL349996 | Neamine derivative)
Affinity DataIC50:  28nMAssay Description:Inhibition of Tat peptide binding to HIV-1 TAR RNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50097335(2-Amino-5-guanidino-pentanoic acid [(4R,5S,6S)-5-a...)
Affinity DataIC50:  600nMAssay Description:Inhibition of Tat peptide binding to HIV-1 TAR RNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate HXB2 ...)
Niddk

Curated by ChEMBL
LigandPNGBDBM50481913(CHEMBL1075826)
Affinity DataIC50:  900nMAssay Description:Inhibition of HIV1 TAT transfected to human HeLa cells assessed as decrease in luminescence after 48 hrs by duel luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50097336(CHEMBL152397 | Pyrene-1-carboxylic acid [(4R,5S,6S...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibitory concentration against human telomeraseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50045403(Acetic acid 2-carbamoyl-3-hydroxy-10,13-dimethyl-1...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of HIV-1 nuclear regulatory protein TatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50407474(CHEMBL3137917)
Affinity DataIC50:  2.60E+3nMAssay Description:The compound was tested for inhibition of HIV-1 replication in SW480 cells using HIV tat assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50407473(CHEMBL3137919)
Affinity DataIC50:  2.60E+3nMAssay Description:The compound was tested for inhibition of HIV-1 replication in SW480 cells using HIV tat assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50045400(Acetic acid 2-methanesulfonyl-10,13-dimethyl-3-oxo...)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of HIV-1 nuclear regulatory protein TatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50407488(CHEMBL3137916)
Affinity DataIC50:  2.70E+3nMAssay Description:The compound was tested for inhibition of HIV-1 replication in SW480 cells using HIV tat assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50407477(CHEMBL109492)
Affinity DataIC50:  2.80E+3nMAssay Description:The compound was tested for inhibition of HIV-1 replication in SW480 cells using HIV tat assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50407490(CHEMBL3137910)
Affinity DataIC50:  3.60E+3nMAssay Description:The compound was tested for inhibition of HIV-1 replication in SW480 cells using HIV tat assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50032828(7-Chloro-5-(1H-pyrrol-2-yl)-1,3-dihydro-benzo[e][1...)
Affinity DataIC50:  4.00E+3nMAssay Description:The compound was tested for inhibition of HIV-1 replication in SW480 cells using HIV tat assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50032828(7-Chloro-5-(1H-pyrrol-2-yl)-1,3-dihydro-benzo[e][1...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of HIV-1 nuclear regulatory protein TatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50407479(CHEMBL323490)
Affinity DataIC50:  4.50E+3nMAssay Description:The compound was tested for inhibition of HIV-1 replication in SW480 cells using HIV tat assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate HXB2 ...)
Niddk

Curated by ChEMBL
LigandPNGBDBM50481920(CHEMBL1075815)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of HIV1 TAT transfected to human HeLa cells assessed as decrease in luminescence after 48 hrs by duel luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50407471(CHEMBL320506)
Affinity DataIC50:  7.00E+3nMAssay Description:The compound was tested for inhibition of HIV-1 replication in SW480 cells using HIV tat assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate HXB2 ...)
Niddk

Curated by ChEMBL
LigandPNGBDBM50481917(CHEMBL1075830)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of HIV1 TAT transfected to human HeLa cells assessed as decrease in luminescence after 48 hrs by duel luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50407480(CHEMBL3137920)
Affinity DataIC50:  8.40E+3nMAssay Description:The compound was tested for inhibition of HIV-1 replication in SW480 cells using HIV tat assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50045401(17-Hydroxy-2-methanesulfonyl-10,13-dimethyl-tetrad...)
Affinity DataIC50:  8.40E+3nMAssay Description:Inhibition of HIV-1 nuclear regulatory protein TatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50407487(CHEMBL2373330)
Affinity DataIC50:  8.40E+3nMAssay Description:The compound was tested for inhibition of HIV-1 replication in SW480 cells using HIV tat assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50407483(CHEMBL108427)
Affinity DataIC50:  9.90E+3nMAssay Description:The compound was tested for inhibition of HIV-1 replication in SW480 cells using HIV tat assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate HXB2 ...)
Niddk

Curated by ChEMBL
LigandPNGBDBM50481915(CHEMBL1075824)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of HIV1 TAT transfected to human HeLa cells assessed as decrease in luminescence after 48 hrs by duel luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50407472(CHEMBL3137913)
Affinity DataIC50:  1.03E+4nMAssay Description:The compound was tested for inhibition of HIV-1 replication in SW480 cells using HIV tat assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate HXB2 ...)
Niddk

Curated by ChEMBL
LigandPNGBDBM50481919(CHEMBL1075821)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of HIV1 TAT transfected to human HeLa cells assessed as decrease in luminescence after 48 hrs by duel luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50407475(CHEMBL3137911)
Affinity DataIC50:  1.43E+4nMAssay Description:The compound was tested for inhibition of HIV-1 replication in SW480 cells using HIV tat assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50045402(3,17-Dihydroxy-10,13-dimethyl-1,4,6,7,8,9,10,11,12...)
Affinity DataIC50:  1.43E+4nMAssay Description:Inhibition of HIV-1 nuclear regulatory protein TatMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50407485(CHEMBL3137914)
Affinity DataIC50:  1.54E+4nMAssay Description:The compound was tested for inhibition of HIV-1 replication in SW480 cells using HIV tat assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate HXB2 ...)
Niddk

Curated by ChEMBL
LigandPNGBDBM50481914(CHEMBL1075825)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of HIV1 TAT transfected to human HeLa cells assessed as decrease in luminescence after 48 hrs by duel luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50407482(CHEMBL107878)
Affinity DataIC50:  1.65E+4nMAssay Description:The compound was tested for inhibition of HIV-1 replication in SW480 cells using HIV tat assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate HXB2 ...)
Niddk

Curated by ChEMBL
LigandPNGBDBM50481918(CHEMBL1081563)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of HIV1 TAT transfected to human HeLa cells assessed as decrease in luminescence after 48 hrs by duel luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50407486(CHEMBL108485)
Affinity DataIC50:  2.14E+4nMAssay Description:The compound was tested for inhibition of HIV-1 replication in SW480 cells using HIV tat assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50407478(CHEMBL3138234)
Affinity DataIC50:  2.45E+4nMAssay Description:The compound was tested for inhibition of HIV-1 replication in SW480 cells using HIV tat assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50407481(CHEMBL111446)
Affinity DataIC50:  2.57E+4nMAssay Description:The compound was tested for inhibition of HIV-1 replication in SW480 cells using HIV tat assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM8580((2R,3S,4R,5R,6R)-5-amino-2-(aminomethyl)-6-{[(1R,2...)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of Tat peptide binding to HIV-1 TAR RNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate HXB2 ...)
Niddk

Curated by ChEMBL
LigandPNGBDBM50481921(CHEMBL1075829)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of HIV1 TAT transfected to human HeLa cells assessed as decrease in luminescence after 48 hrs by duel luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50407489(CHEMBL111424)
Affinity DataIC50:  3.17E+4nMAssay Description:The compound was tested for inhibition of HIV-1 replication in SW480 cells using HIV tat assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50407469(CHEMBL323217)
Affinity DataIC50:  3.21E+4nMAssay Description:The compound was tested for inhibition of HIV-1 replication in SW480 cells using HIV tat assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50407476(CHEMBL325765)
Affinity DataIC50:  3.35E+4nMAssay Description:The compound was tested for inhibition of HIV-1 replication in SW480 cells using HIV tat assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50407468(CHEMBL110573)
Affinity DataIC50:  3.40E+4nMAssay Description:The compound was tested for inhibition of HIV-1 replication in SW480 cells using HIV tat assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate HXB2 ...)
Niddk

Curated by ChEMBL
LigandPNGBDBM50481916(CHEMBL1075823)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of HIV1 TAT transfected to human HeLa cells assessed as decrease in luminescence after 48 hrs by duel luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50407484(CHEMBL320265)
Affinity DataIC50:  7.20E+4nMAssay Description:The compound was tested for inhibition of HIV-1 replication in SW480 cells using HIV tat assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50407470(CHEMBL326009)
Affinity DataIC50:  2.78E+5nMAssay Description:The compound was tested for inhibition of HIV-1 replication in SW480 cells using HIV tat assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50097337(CHEMBL349996 | Neamine derivative)
Affinity DataKd:  30nMAssay Description:Compound was evaluated for its inhibitory activity against Klenow enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50097336(CHEMBL152397 | Pyrene-1-carboxylic acid [(4R,5S,6S...)
Affinity DataKd:  290nMAssay Description:Dissociation constant for TAR RNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate PCV12...)
Graduate School Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50097338(CHEMBL408877 | Neamine derivative)
Affinity DataKd:  25nMAssay Description:Dissociation constant for TAR RNAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate HXB2 ...)
Niddk

Curated by ChEMBL
LigandPNGBDBM50410416(CHEMBL196072)
Affinity DataKd:  1.80E+3nMT: 2°CAssay Description:In vitro binding affinity towards Tat/TAR to determine interaction between TAR RNA and Tat peptide at room temperature using fluorescence spectrophot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate HXB2 ...)
Niddk

Curated by ChEMBL
LigandPNGBDBM50410417(CHEMBL371627)
Affinity DataKd:  7.70E+3nMT: 2°CAssay Description:In vitro binding affinity towards Tat/TAR to determine interaction between TAR RNA and Tat peptide at room temperature using fluorescence spectrophot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate HXB2 ...)
Niddk

Curated by ChEMBL
LigandPNGBDBM50410418(CHEMBL194688)
Affinity DataKd:  7.41E+5nMT: 2°CAssay Description:In vitro binding affinity towards Tat/TAR to determine interaction between TAR RNA and Tat peptide at room temperature using fluorescence spectrophot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate HXB2 ...)
Niddk

Curated by ChEMBL
LigandPNGBDBM50410419(CHEMBL364677)
Affinity DataKd:  9.52E+5nMT: 2°CAssay Description:In vitro binding affinity towards Tat/TAR to determine interaction between TAR RNA and Tat peptide at room temperature using fluorescence spectrophot...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Tat(Human immunodeficiency virus type 1 (isolate HXB2 ...)
Niddk

Curated by ChEMBL
LigandPNGBDBM50398244(CHEMBL609728)
Affinity DataEC50:  1.00E+4nMAssay Description:Inhibition of Tat-mediated transcription of viral promoter in 293 T cells transfected with HIV1 tat by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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