Compile Data Set for Download or QSAR
maximum 50k data
Found 9 Enz. Inhib. hit(s) with Target = 'Insulin receptor substrate 1 [1-264]'
TargetInsulin receptor substrate 1 [1-264](Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM223477(US9320734, 316)
Affinity DataKd:  1.99E+3nMAssay Description:KT1 PH domain small molecule inhibitors were identified using the crystal structure of the AKT1 PH domain bound by PtdIns(1,3,4,5)P4 as descried in T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInsulin receptor substrate 1 [1-264](Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM223486(US9320734, 331)
Affinity DataKd:  2.40E+3nMAssay Description:KT1 PH domain small molecule inhibitors were identified using the crystal structure of the AKT1 PH domain bound by PtdIns(1,3,4,5)P4 as descried in T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInsulin receptor substrate 1 [1-264](Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM223488(US9320734, 332)
Affinity DataKd:  1.07E+4nMAssay Description:KT1 PH domain small molecule inhibitors were identified using the crystal structure of the AKT1 PH domain bound by PtdIns(1,3,4,5)P4 as descried in T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInsulin receptor substrate 1 [1-264](Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM223487(US9320734, 333)
Affinity DataKd:  1.80E+3nMAssay Description:KT1 PH domain small molecule inhibitors were identified using the crystal structure of the AKT1 PH domain bound by PtdIns(1,3,4,5)P4 as descried in T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInsulin receptor substrate 1 [1-264](Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM223489(US9320734, 360)
Affinity DataKd:  1.74E+3nMAssay Description:KT1 PH domain small molecule inhibitors were identified using the crystal structure of the AKT1 PH domain bound by PtdIns(1,3,4,5)P4 as descried in T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInsulin receptor substrate 1 [1-264](Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM223490(US9320734, 335)
Affinity DataKd:  520nMAssay Description:KT1 PH domain small molecule inhibitors were identified using the crystal structure of the AKT1 PH domain bound by PtdIns(1,3,4,5)P4 as descried in T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInsulin receptor substrate 1 [1-264](Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM223477(US9320734, 316)
Affinity DataKd:  390nMAssay Description:KT1 PH domain small molecule inhibitors were identified using the crystal structure of the AKT1 PH domain bound by PtdIns(1,3,4,5)P4 as descried in T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInsulin receptor substrate 1 [1-264](Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM223487(US9320734, 333)
Affinity DataKd:  140nMAssay Description:KT1 PH domain small molecule inhibitors were identified using the crystal structure of the AKT1 PH domain bound by PtdIns(1,3,4,5)P4 as descried in T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetInsulin receptor substrate 1 [1-264](Homo sapiens (Human))
The University Of Texas System

US Patent
LigandPNGBDBM223489(US9320734, 360)
Affinity DataKd:  1.07E+4nMAssay Description:KT1 PH domain small molecule inhibitors were identified using the crystal structure of the AKT1 PH domain bound by PtdIns(1,3,4,5)P4 as descried in T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent