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Found 132 Enz. Inhib. hit(s) with Target = 'UDP-N-acetylmuramoylalanine--D-glutamate ligase'
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046818(CHEMBL3310464)
Affinity DataKi:  2.10E+4nMAssay Description:Competitive inhibition of Escherichia coli MurD using D-Glu substrate by steady-state enzyme kinetics assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046818(CHEMBL3310464)
Affinity DataKi:  2.90E+4nMAssay Description:Partial non-competitive inhibition of Escherichia coli MurD using UMA substrate by steady-state enzyme kinetics assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046818(CHEMBL3310464)
Affinity DataKi:  3.90E+4nMAssay Description:Partial un-competitive inhibition of Escherichia coli MurD using ATP substrate by steady-state enzyme kinetics assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50021359(CHEMBL3288597)
Affinity DataKi:  1.15E+5nMAssay Description:Competitive inhibition of Escherichia coli MurD ligase activity using UDP-N-acetylmuramyl-L-alanine as a substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM119097(MurD inhibitor (compound 36))
Affinity DataIC50: <1nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM119123(MurD/E/F inhibitor (compound 69))
Affinity DataIC50:  2.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM119104(MurD inhibitor (compound 46))
Affinity DataIC50:  3.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus (Firmicutes))
University Of Ljubljana

LigandPNGBDBM119107(MurD/E inhibitor (compound 49))
Affinity DataIC50:  6.40E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM119107(MurD/E inhibitor (compound 49))
Affinity DataIC50:  8.20E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM119100(MurD inhibitor (compound 42))
Affinity DataIC50:  8.40E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM119105(MurD inhibitor (compound 47))
Affinity DataIC50:  1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus (Firmicutes))
University Of Ljubljana

LigandPNGBDBM50475587(CHEMBL426651)
Affinity DataIC50:  1.04E+4nMAssay Description:Inhibitory activity against MurD in Staphylococcus aureusMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus (Firmicutes))
University Of Ljubljana

LigandPNGBDBM50475591(CHEMBL382328)
Affinity DataIC50:  1.25E+4nMAssay Description:Inhibitory activity against MurD in Staphylococcus aureusMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50475586(CHEMBL198030)
Affinity DataIC50:  1.25E+4nMAssay Description:Inhibitory activity against MurD in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus (Firmicutes))
University Of Ljubljana

LigandPNGBDBM119122(MurA/B/C/D/E inhibitor (compound 67))
Affinity DataIC50:  1.30E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50475590(CHEMBL370421)
Affinity DataIC50:  1.35E+4nMAssay Description:Inhibitory activity against MurD in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50475579(CHEMBL382202)
Affinity DataIC50:  1.46E+4nMAssay Description:Inhibitory activity against MurD in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM85276(HEA derivative, 7c | MurC/D/E/F inhibitor (compoun...)
Affinity DataIC50:  1.80E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50475601(CHEMBL199812)
Affinity DataIC50:  1.95E+4nMAssay Description:Inhibitory activity against MurD in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus (Firmicutes))
University Of Ljubljana

LigandPNGBDBM50475599(CHEMBL200097)
Affinity DataIC50:  2.05E+4nMAssay Description:Inhibitory activity against MurD in Staphylococcus aureusMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus (Firmicutes))
University Of Ljubljana

LigandPNGBDBM50475603(CHEMBL199320)
Affinity DataIC50:  2.62E+4nMAssay Description:Inhibitory activity against MurD in Staphylococcus aureusMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM119086(MurC/D inhibitor (compound 25) | MurD inhibitor (c...)
Affinity DataIC50:  3.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM119086(MurC/D inhibitor (compound 25) | MurD inhibitor (c...)
Affinity DataIC50:  3.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus (Firmicutes))
University Of Ljubljana

LigandPNGBDBM50221037(CHEMBL87262)
Affinity DataIC50:  3.02E+4nMAssay Description:In vitro inhibitory activity against Staphylococcus aureus UDP-N-acetylmuramoyl-L-alanyl-D-glutamate synthetaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus (Firmicutes))
University Of Ljubljana

LigandPNGBDBM50221022(CHEMBL86525)
Affinity DataIC50:  3.28E+4nMAssay Description:In vitro inhibitory activity against Staphylococcus aureus UDP-N-acetylmuramoyl-L-alanyl-D-glutamate synthetaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus (Firmicutes))
University Of Ljubljana

LigandPNGBDBM50475582(CHEMBL199511)
Affinity DataIC50:  3.35E+4nMAssay Description:Inhibitory activity against MurD in Staphylococcus aureusMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus (Firmicutes))
University Of Ljubljana

LigandPNGBDBM50221032(CHEMBL86526)
Affinity DataIC50:  3.45E+4nMAssay Description:In vitro inhibitory activity against Staphylococcus aureus UDP-N-acetylmuramoyl-L-alanyl-D-glutamate synthetaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50475607(CHEMBL199629)
Affinity DataIC50:  3.47E+4nMAssay Description:Inhibitory activity against MurD in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus (Firmicutes))
University Of Ljubljana

LigandPNGBDBM50221030(CHEMBL313078)
Affinity DataIC50:  3.60E+4nMAssay Description:In vitro inhibitory activity against Staphylococcus aureus UDP-N-acetylmuramoyl-L-alanyl-D-glutamate synthetaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus (Firmicutes))
University Of Ljubljana

LigandPNGBDBM50221020(CHEMBL87126)
Affinity DataIC50:  4.19E+4nMAssay Description:In vitro inhibitory activity against Staphylococcus aureus UDP-N-acetylmuramoyl-L-alanyl-D-glutamate synthetaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM119122(MurA/B/C/D/E inhibitor (compound 67))
Affinity DataIC50:  4.40E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM119106(MurD inhibitor (compound 48))
Affinity DataIC50:  4.50E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM119103(MurD inhibitor (compound 45))
Affinity DataIC50:  4.50E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus (Firmicutes))
University Of Ljubljana

LigandPNGBDBM50221027(CHEMBL327438)
Affinity DataIC50:  4.52E+4nMAssay Description:In vitro inhibitory activity against Staphylococcus aureus UDP-N-acetylmuramoyl-L-alanyl-D-glutamate synthetaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus (Firmicutes))
University Of Ljubljana

LigandPNGBDBM50221018(CHEMBL85772)
Affinity DataIC50:  4.74E+4nMAssay Description:In vitro inhibitory activity against Staphylococcus aureus UDP-N-acetylmuramoyl-L-alanyl-D-glutamate synthetaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus (Firmicutes))
University Of Ljubljana

LigandPNGBDBM50221038(CHEMBL87521)
Affinity DataIC50:  4.87E+4nMAssay Description:In vitro inhibitory activity against Staphylococcus aureus UDP-N-acetylmuramoyl-L-alanyl-D-glutamate synthetaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus (Firmicutes))
University Of Ljubljana

LigandPNGBDBM50475596(CHEMBL200015)
Affinity DataIC50:  4.88E+4nMAssay Description:Inhibitory activity against MurD in Staphylococcus aureusMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus (Firmicutes))
University Of Ljubljana

LigandPNGBDBM50221023(CHEMBL84684)
Affinity DataIC50:  4.93E+4nMAssay Description:In vitro inhibitory activity against Staphylococcus aureus UDP-N-acetylmuramoyl-L-alanyl-D-glutamate synthetaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus (Firmicutes))
University Of Ljubljana

LigandPNGBDBM50221033(CHEMBL420601)
Affinity DataIC50:  4.97E+4nMAssay Description:In vitro inhibitory activity against Staphylococcus aureus UDP-N-acetylmuramoyl-L-alanyl-D-glutamate synthetaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus (Firmicutes))
University Of Ljubljana

LigandPNGBDBM50475597(CHEMBL380752)
Affinity DataIC50: >5.32E+4nMAssay Description:Inhibitory activity against MurD in Staphylococcus aureusMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50475600(CHEMBL381006)
Affinity DataIC50: >5.32E+4nMAssay Description:Inhibitory activity against MurD in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50475593(CHEMBL199553)
Affinity DataIC50: >5.86E+4nMAssay Description:Inhibitory activity against MurD in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50046818(CHEMBL3310464)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibition of Escherichia coli MurD after 15 mins in presence of 0.005% Triton X-114 by Malachite green assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50475595(CHEMBL199757)
Affinity DataIC50: >6.12E+4nMAssay Description:Inhibitory activity against MurD in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Staphylococcus aureus (Firmicutes))
University Of Ljubljana

LigandPNGBDBM50221019(CHEMBL87584)
Affinity DataIC50:  6.37E+4nMAssay Description:In vitro inhibitory activity against Staphylococcus aureus UDP-N-acetylmuramoyl-L-alanyl-D-glutamate synthetaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50475584(CHEMBL197817)
Affinity DataIC50: >6.40E+4nMAssay Description:Inhibitory activity against MurD in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50475602(CHEMBL199929)
Affinity DataIC50: >6.40E+4nMAssay Description:Inhibitory activity against MurD in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50475606(CHEMBL199580)
Affinity DataIC50: >6.53E+4nMAssay Description:Inhibitory activity against MurD in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50475583(CHEMBL372594)
Affinity DataIC50: >6.53E+4nMAssay Description:Inhibitory activity against MurD in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-N-acetylmuramoylalanine--D-glutamate ligase(Escherichia coli (strain K12))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50475598(CHEMBL381658)
Affinity DataIC50: >6.53E+4nMAssay Description:Inhibitory activity against MurD in Escherichia coliMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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