Compile Data Set for Download or QSAR
maximum 50k data
Found 60 Enz. Inhib. hit(s) with Target = 'Protein-tyrosine-phosphatase'
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM26193(2-Hydroxybenzoate, I | 2-hydroxybenzoic acid | CHE...)
Affinity DataKi:  1.00E+6nMAssay Description:Inhibition of Yersinia pseudotuberculosis YopHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50326496(4, 4'-[[2-[[(4-(4-Trifluoromethylthio)phenoxy phen...)
Affinity DataIC50:  30nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50326497(4, 4'-[[2-[[(4-(4-Trifluoromethylthio)phenoxypheny...)
Affinity DataIC50:  50nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50326498(4, 4'-[[2-[[(4-(4-Ethyl)phenoxyphenyl)amino]carbon...)
Affinity DataIC50:  70nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50326499(4, 4'-[[2-[[(4-(4-n-Hexyl)phenoxyphenyl)amino]carb...)
Affinity DataIC50:  90nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50326500(2,2'-(4,4'-(2-(3-(benzyloxy)phenylcarbamoyl)-1,4-p...)
Affinity DataIC50:  100nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Homo sapiens (Human))
Sejong University

Curated by ChEMBL
LigandPNGBDBM50391713(CHEMBL2146956)
Affinity DataIC50:  100nMAssay Description:Inhibition of His-tagged PTPsigma catalytic domain amino acid 1369 to 1948 using DiFMUP as substrate after 20 mins by spectrofluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50326502(2,2'-(4,4'-(2-(4-(4-fluorophenoxy)phenylcarbamoyl)...)
Affinity DataIC50:  110nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50326501(2,2'-(4,4'-(2-(4-(4-(methylthio)phenoxy)phenylcarb...)
Affinity DataIC50:  110nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50342237((E)-5-((((3'-(Difluoro(phosphono)methyl)-[1,1'-bip...)
Affinity DataIC50:  190nMAssay Description:Inhibition of Yersinia pestis outer protein H expressed in Escherichia coli after 15 to 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50326503(2,2'-(4,4'-(2-(4-(p-tolyloxy)phenylcarbamoyl)-1,4-...)
Affinity DataIC50:  190nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50326504(2,2'-(4,4'-(2-(4-(4-butylphenoxy)phenylcarbamoyl)-...)
Affinity DataIC50:  200nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Homo sapiens (Human))
Sejong University

Curated by ChEMBL
LigandPNGBDBM50237957(4-(2-((2,5-dioxoimidazolidin-4-ylidene)methyl)-1H-...)
Affinity DataIC50:  200nMAssay Description:Inhibition of His-tagged PTPsigma catalytic domain amino acid 1369 to 1948 using DiFMUP as substrate after 20 mins by spectrofluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50326505(2,2'-(4,4'-(2-(4-(3,4-dichlorophenoxy)phenylcarbam...)
Affinity DataIC50:  210nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50326506(2,2'-(4,4'-(2-(4-(3-chlorophenoxy)phenylcarbamoyl)...)
Affinity DataIC50:  220nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50326507(2,2'-(4,4'-(2-(4-(o-tolyloxy)phenylcarbamoyl)-1,4-...)
Affinity DataIC50:  230nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50326508(2,2'-(4,4'-(2-(4-phenoxyphenylcarbamoyl)-1,4-pheny...)
Affinity DataIC50:  240nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Homo sapiens (Human))
Sejong University

Curated by ChEMBL
LigandPNGBDBM50391714(CHEMBL2146957)
Affinity DataIC50:  600nMAssay Description:Inhibition of His-tagged PTPsigma catalytic domain amino acid 1369 to 1948 using DiFMUP as substrate after 20 mins by spectrofluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Homo sapiens (Human))
Sejong University

Curated by ChEMBL
LigandPNGBDBM50391715(CHEMBL2146960)
Affinity DataIC50:  700nMAssay Description:Inhibition of His-tagged PTPsigma catalytic domain amino acid 1369 to 1948 using DiFMUP as substrate after 20 mins by spectrofluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50342236(CHEMBL1766711 | difluoro(4'-(((5-(hydroxymethyl)fu...)
Affinity DataIC50:  730nMAssay Description:Inhibition of Yersinia pestis outer protein H expressed in Escherichia coli after 15 to 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50326509(2,2'-(4,4'-(2-(4-(4-isopropylphenoxy)phenylcarbamo...)
Affinity DataIC50:  800nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Homo sapiens (Human))
Sejong University

Curated by ChEMBL
LigandPNGBDBM50391711(CHEMBL2146958)
Affinity DataIC50:  900nMAssay Description:Inhibition of His-tagged PTPsigma catalytic domain amino acid 1369 to 1948 using DiFMUP as substrate after 20 mins by spectrofluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50326510(2,2'-(4,4'-(2-(4-(2,4-difluorophenoxy)phenylcarbam...)
Affinity DataIC50:  910nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50342235(CHEMBL1766710 | difluoro(4'-(((5-methylfuran-2-yl)...)
Affinity DataIC50:  910nMAssay Description:Inhibition of Yersinia pestis outer protein H expressed in Escherichia coli after 15 to 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50326511(2,2'-(4,4'-(2-(4-(4-methoxyphenoxy)phenylcarbamoyl...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50342234(CHEMBL1766709 | difluoro(4'-((furan-2-ylmethylenea...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of Yersinia pestis outer protein H expressed in Escherichia coli after 15 to 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Homo sapiens (Human))
Sejong University

Curated by ChEMBL
LigandPNGBDBM50387974(CHEMBL2057830)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of His-tagged PTPsigma catalytic domain amino acid 1369 to 1948 using DiFMUP as substrate after 20 mins by spectrofluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50326512(2,2'-(4,4'-(2-(4-(4-cyanophenoxy)phenylcarbamoyl)-...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of Yersinia pestis YOpHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Homo sapiens (Human))
Sejong University

Curated by ChEMBL
LigandPNGBDBM50391712(CHEMBL2146959)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of His-tagged PTPsigma catalytic domain amino acid 1369 to 1948 using DiFMUP as substrate after 20 mins by spectrofluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50170983((S)-4-[(S)-4-(R)-Carbamoyl-1-(4-carboxymethoxy-ben...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibitory concentration against Yersinia pestis YopH expressed in Escherichia coli BL21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50170984((S)-4-{(S)-4-(R)-Carbamoyl-1-[4-(carboxy-difluoro-...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibitory concentration against Yersinia pestis YopH expressed in Escherichia coli BL21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50170988((4-{(S)-2-[(S)-3-Benzyloxycarbonylamino-2-(9H-fluo...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibitory concentration against Yersinia pestis YopH expressed in Escherichia coli BL21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50170995((S)-4-[(S)-4-(R)-Carbamoyl-1-(4-carboxymethyl-benz...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibitory concentration against Yersinia pestis YopH expressed in Escherichia coli BL21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50317073(16-(4-(benzyloxy)phenyl)-3,14-dioxa-2,15-diazahexa...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of Yersinia pestis YopH after 15 mins by pNPP hydrolysis assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50170990((S)-4-{(S)-4-(R)-Carbamoyl-1-[4-(carboxy-difluoro-...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibitory concentration against Yersinia pestis YopH expressed in Escherichia coli BL21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50131099((S)-4-[(S)-1-((S)-1-Carbamoyl-3-methyl-butylcarbam...)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of Tyrosine phosphatase from Yersinia pestis expressed in E. coli BL21 (DE3) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50131100(2-{4-[(S)-2-[(S)-4-Benzyloxycarbonyl-2-(9H-fluoren...)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of Tyrosine phosphatase from Yersinia pestis expressed in E. coli BL21 (DE3) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50131102(2-{4-[(S)-2-[(S)-4-Benzyloxycarbonyl-2-(9H-fluoren...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of Tyrosine phosphatase from Yersinia pestis expressed in E. coli BL21 (DE3) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50342233(CHEMBL1766708 | difluoro(4'-((furan-3-ylmethylenea...)
Affinity DataIC50:  3.69E+3nMAssay Description:Inhibition of Yersinia pestis outer protein H expressed in Escherichia coli after 15 to 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50170993(CHEMBL364349 | {4-[(S)-2-[3-Benzyloxycarbonylamino...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibitory concentration against Yersinia pestis YopH expressed in Escherichia coli BL21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50131104((S)-4-{(S)-1-((S)-1-Carbamoyl-3-methyl-butylcarbam...)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of Tyrosine phosphatase from Yersinia pestis expressed in E. coli BL21 (DE3) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50170986((S)-4-[(S)-4-(R)-Carbamoyl-1-(4-carboxymethoxy-ben...)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibitory concentration against Yersinia pestis YopH expressed in Escherichia coli BL21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50131091((S)-4-[(S)-1-((S)-1-Carbamoyl-3-methyl-butylcarbam...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of Tyrosine phosphatase from Yersinia pestis expressed in E. coli BL21 (DE3) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50131095(5-[(S)-2-[(S)-4-Benzyloxycarbonyl-2-(9H-fluoren-9-...)
Affinity DataIC50:  1.05E+4nMAssay Description:Inhibition of Tyrosine phosphatase from Yersinia pestis expressed in E. coli BL21 (DE3) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50170982((S)-4-(3-Anthracen-9-yl-propionylamino)-4-[(S)-4-(...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibitory concentration against Yersinia pestis YopH expressed in Escherichia coli BL21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50170989((S)-4-[(S)-4-(R)-Carbamoyl-1-(4-carboxymethoxy-ben...)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibitory concentration against Yersinia pestis YopH expressed in Escherichia coli BL21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50379184(CHEMBL2010868)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of Yersinia pseudotuberculosis YopHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50131093((S)-4-[(S)-2-(3,4-Bis-carboxymethoxy-phenyl)-1-((S...)
Affinity DataIC50:  1.94E+4nMAssay Description:Inhibition of Tyrosine phosphatase from Yersinia pestis expressed in E. coli BL21 (DE3) cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50170994((S)-4-[(S)-4-(R)-Carbamoyl-1-(4-carboxymethoxy-ben...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibitory concentration against Yersinia pestis YopH expressed in Escherichia coli BL21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein-tyrosine-phosphatase(Yersinia pestis)
Indiana University

Curated by ChEMBL
LigandPNGBDBM50170992((S)-4-[(S)-4-(R)-Carbamoyl-1-(4-carboxymethoxy-ben...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibitory concentration against Yersinia pestis YopH expressed in Escherichia coli BL21 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 60 total ) | Next | Last >>
Jump to: