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Found 1643 Enz. Inhib. hit(s) with Target = 'Phospholipase A2'
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
National Chung-Hsing University

Curated by ChEMBL
LigandPNGBDBM50139531(CHEMBL165545 | Octyl-carbamic acid 3-octylcarbamoy...)
Affinity DataKi:  4.00E+3nMAssay Description:Binding affinity of the compound against phospholipase A2 of Naja mocambique mocambiqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
National Chung-Hsing University

Curated by ChEMBL
LigandPNGBDBM50139529(CHEMBL166217 | Octyl-carbamic acid 2-octylcarbamoy...)
Affinity DataKi:  1.10E+4nMAssay Description:Binding affinity of the compound against phospholipase A2 of Naja mocambique mocambiqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
National Chung-Hsing University

Curated by ChEMBL
LigandPNGBDBM50139530(CHEMBL434865 | Octyl-carbamic acid 4-octylcarbamoy...)
Affinity DataKi:  1.50E+4nMAssay Description:Binding affinity of the compound against phospholipase A2 of Naja mocambique mocambiqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50053109(CHEMBL331755 | [1-Aminooxalyl-3-(2-benzyl-benzyl)-...)
Affinity DataIC50:  1.30nMAssay Description:Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50053136((1-Aminooxalyl-3-biphenyl-2-ylmethyl-2-methyl-indo...)
Affinity DataIC50:  1.40nMAssay Description:Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50601469(CHEMBL5172164)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of human group IIA phospholipase A2 preincubated with compound for 10 mins followed by enzyme addition and measured after 30 mins by PC/DO...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50053137((1-Aminooxalyl-3-biphenyl-2-ylmethyl-2-ethyl-indol...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human group IIA phospholipase A2 preincubated with compound for 10 mins followed by enzyme addition and measured after 30 mins by PC/DO...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPhospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50053102(CHEMBL121245 | [1-Aminooxalyl-3-(3-chloro-benzyl)-...)
Affinity DataIC50:  3nMAssay Description:Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50161301(2-[4-(2-Benzenesulfonylamino-2-oxo-ethoxy)-1-benzy...)
Affinity DataIC50:  3nMAssay Description:Inhibitory concentration against human nonpancreatic secretory phospholipase A2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50053108((1-Aminooxalyl-3-benzyl-2-methyl-indolizin-8-yloxy...)
Affinity DataIC50:  3nMAssay Description:Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50053137((1-Aminooxalyl-3-biphenyl-2-ylmethyl-2-ethyl-indol...)
Affinity DataIC50:  3nMAssay Description:Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
National Chung-Hsing University

Curated by ChEMBL
LigandPNGBDBM50055367(CHEMBL345986 | [3-Aminooxalyl-1-(3-chloro-benzyl)-...)
Affinity DataIC50:  3nMAssay Description:Compound wastested for inhibition of porcine secreted pancreatic PLA2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50055371((3-aminooxalyl-1-biphenyl-2-ylmethyl-2-methyl-1H-i...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human nonpancreatic secretory Phospholipase A2 through DOC/PC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50053106(CHEMBL120112 | [1-Aminooxalyl-2-ethyl-3-(3-trifluo...)
Affinity DataIC50:  3nMAssay Description:Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50161305((3-Aminooxalyl-1-cyclohexylmethyl-2-methyl-2,3-dih...)
Affinity DataIC50:  4nMAssay Description:Inhibitory concentration against human nonpancreatic secretory phospholipase A2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50055374(CHEMBL436456 | [3-Aminooxalyl-1-(2-benzyl-benzyl)-...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human nonpancreatic secretory Phospholipase A2 through DOC/PC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50055374(CHEMBL436456 | [3-Aminooxalyl-1-(2-benzyl-benzyl)-...)
Affinity DataIC50:  4nMAssay Description:Inhibition of human nonpancreatic secretory Phospholipase A2 through chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50053114((1-Aminooxalyl-3-biphenyl-3-ylmethyl-2-ethyl-indol...)
Affinity DataIC50:  4.20nMAssay Description:Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50601472(CHEMBL5208632)
Affinity DataIC50:  5nMAssay Description:Inhibition of human group IIA phospholipase A2 preincubated with compound for 10 mins followed by enzyme addition and measured after 30 mins by PC/DO...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50053123((1-Aminooxalyl-2-ethyl-3-naphthalen-1-ylmethyl-ind...)
Affinity DataIC50:  5nMAssay Description:Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50053096(CHEMBL123774 | [1-Aminooxalyl-3-(4-butyl-benzyl)-2...)
Affinity DataIC50:  5nMAssay Description:Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50053133((1-Aminooxalyl-3-benzyl-2-ethyl-indolizin-8-yloxy)...)
Affinity DataIC50:  5nMAssay Description:Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50055371((3-aminooxalyl-1-biphenyl-2-ylmethyl-2-methyl-1H-i...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human group IIA phospholipase A2 incubated for 1 hrs by scintillation counter analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50053137((1-Aminooxalyl-3-biphenyl-2-ylmethyl-2-ethyl-indol...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human group IIA phospholipase A2 incubated for 30 mins by automatic plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPhospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50053147((1-Aminooxalyl-3-biphenyl-2-ylmethyl-2-cyclopropyl...)
Affinity DataIC50:  6nMAssay Description:Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50161293((3-Aminooxalyl-1-benzyl-2-methyl-1,6,7,8-tetrahydr...)
Affinity DataIC50:  6nMAssay Description:Inhibitory concentration against human nonpancreatic secretory phospholipase A2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50053109(CHEMBL331755 | [1-Aminooxalyl-3-(2-benzyl-benzyl)-...)
Affinity DataIC50:  6nMAssay Description:Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50055401((3-Aminooxalyl-1-biphenyl-2-ylmethyl-2-ethyl-1H-in...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human nonpancreatic secretory Phospholipase A2 through chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50055387((R)-2-(3-Aminooxalyl-1-benzyl-2-methyl-1H-indol-4-...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human nonpancreatic secretory Phospholipase A2 through DOC/PC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50055378(CHEMBL345488 | [3-Aminooxalyl-1-(2,6-dichloro-benz...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human nonpancreatic secretory Phospholipase A2 through chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50053137((1-Aminooxalyl-3-biphenyl-2-ylmethyl-2-ethyl-indol...)
Affinity DataIC50:  6nMAssay Description:Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50055371((3-aminooxalyl-1-biphenyl-2-ylmethyl-2-methyl-1H-i...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human nonpancreatic secretory Phospholipase A2 through chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50055379((3-Aminooxalyl-1-biphenyl-2-ylmethyl-2-cyclopropyl...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human nonpancreatic secretory Phospholipase A2 through chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50055401((3-Aminooxalyl-1-biphenyl-2-ylmethyl-2-ethyl-1H-in...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human nonpancreatic secretory Phospholipase A2 through DOC/PC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50053102(CHEMBL121245 | [1-Aminooxalyl-3-(3-chloro-benzyl)-...)
Affinity DataIC50:  6nMAssay Description:Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
National Chung-Hsing University

Curated by ChEMBL
LigandPNGBDBM50055384((3-Aminooxalyl-1-biphenyl-3-ylmethyl-2-methyl-1H-i...)
Affinity DataIC50:  7nMAssay Description:Inhibition of pig group IB phospholipase A2 incubated for 1 hrs by scintillation counter analysisMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50601470(CHEMBL5177527)
Affinity DataIC50:  7nMAssay Description:Inhibition of human group IIA phospholipase A2 incubated for 30 mins by automatic plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50601470(CHEMBL5177527)
Affinity DataIC50:  7nMAssay Description:Inhibition of human group IIA phospholipase A2 preincubated with compound for 10 mins followed by enzyme addition and measured after 30 mins by PC/DO...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  7nMAssay Description:Inhibitory concentration against human nonpancreatic secretory phospholipase A2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50161299((3-Aminooxalyl-1-benzyl-2-ethyl-1,6,7,8-tetrahydro...)
Affinity DataIC50:  7nMAssay Description:Inhibitory concentration against human nonpancreatic secretory phospholipase A2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50161301(2-[4-(2-Benzenesulfonylamino-2-oxo-ethoxy)-1-benzy...)
Affinity DataIC50:  7nMAssay Description:Inhibitory concentration against human nonpancreatic secretory phospholipase A2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
National Chung-Hsing University

Curated by ChEMBL
LigandPNGBDBM50055384((3-Aminooxalyl-1-biphenyl-3-ylmethyl-2-methyl-1H-i...)
Affinity DataIC50:  7nMAssay Description:Compound was tested for inhibition of porcine secretory pancreatic Phospholipase A2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50055366((3-Aminooxalyl-1-benzyl-2-ethyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  7nMAssay Description:Inhibition of human nonpancreatic secretory Phospholipase A2 through DOC/PC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50055367(CHEMBL345986 | [3-Aminooxalyl-1-(3-chloro-benzyl)-...)
Affinity DataIC50:  7nMAssay Description:Inhibition of human nonpancreatic secretory Phospholipase A2 through chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50053095((1-Aminooxalyl-2-ethyl-3-naphthalen-2-ylmethyl-ind...)
Affinity DataIC50:  7.30nMAssay Description:Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50601469(CHEMBL5172164)
Affinity DataIC50:  8nMAssay Description:Inhibition of human group IIA phospholipase A2 incubated for 30 mins by automatic plate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50053136((1-Aminooxalyl-3-biphenyl-2-ylmethyl-2-methyl-indo...)
Affinity DataIC50:  8nMAssay Description:Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50053133((1-Aminooxalyl-3-benzyl-2-ethyl-indolizin-8-yloxy)...)
Affinity DataIC50:  8nMAssay Description:Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50055370((3-Aminooxalyl-2-methyl-1-octyl-1H-indol-4-yloxy)-...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human nonpancreatic secretory Phospholipase A2 through chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50055380((3-Aminooxalyl-1-benzyl-2-ethyl-6-methyl-1H-indol-...)
Affinity DataIC50:  8nMAssay Description:Inhibition of human nonpancreatic secretory Phospholipase A2 through chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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