Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with Target = 'Ras-related protein Rap-1A'
TargetRas-related protein Rap-1A(Homo sapiens (Human))
Universite£

Curated by ChEMBL
LigandPNGBDBM50101929(3-oxo-18-oxa-2,5,9,11-tetraazahexacyclo[17.6.2.22,...)
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of Rap1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRas-related protein Rap-1A(Homo sapiens (Human))
Universite£

Curated by ChEMBL
LigandPNGBDBM50139187(4-(2-cyclohexylethyl)-23-oxo-8-oxa-1,15,17,21-tetr...)
Affinity DataEC50:  140nMAssay Description:Inhibition of Rap1aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRas-related protein Rap-1A(Homo sapiens (Human))
Universite£

Curated by ChEMBL
LigandPNGBDBM50310364(CHEMBL1077126 | YESSOTOXIN)
Affinity DataKd:  4.00E+3nMAssay Description:Binding affinity to RAP1A in human RBC membrane by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRas-related protein Rap-1A(Homo sapiens (Human))
Universite£

Curated by ChEMBL
LigandPNGBDBM50310364(CHEMBL1077126 | YESSOTOXIN)
Affinity DataKd:  4.00E+3nMAssay Description:Binding affinity to RAP1A in human RBC membrane by western blot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRas-related protein Rap-1A(Homo sapiens (Human))
Universite£

Curated by ChEMBL
LigandPNGBDBM50330178(CHEMBL1269578 | desulfo-Yessotoxin)
Affinity DataKd:  500nMAssay Description:Binding affinity to RAP1A in human RBC membrane by surface plasmon resonance analysis with inverted configurationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed