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Found 103 Enz. Inhib. hit(s) with Target = 'L-selectin'
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50060512((R)-4-Methylcarbamoyl-4-[(R)-2-(2-tetradecyl-hexad...)
Affinity DataIC50:  700nMAssay Description:Inhibition of Selectin L bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50205383((5-{4-[(2',3',4'-trihydroxy-biphenyl-3-carbonyl)-a...)
Affinity DataIC50:  790nMAssay Description:Inhibition of human L-selectin after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50060511((R)-4-Methylcarbamoyl-4-[(S)-2-(2-tetradecyl-hexad...)
Affinity DataIC50:  800nMAssay Description:Inhibition of Selectin L bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50072620(1-[4-Methoxy-3-(3,4,5-trihydroxy-6-hydroxymethyl-t...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibitory activity of the compound against L-selectin IgG chimeras binding to sLex coating 96 wells using competitive cell-free ELISA assay was dete...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50205368((5-{3-[(2',3',4'-trihydroxy-biphenyl-3-carbonyl)-a...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of human L-selectin after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50205396(3-[2-(3,4,5-trihydroxy-phenyl)-acetylamino]-benzoi...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of human L-selectin after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50205377(CHEMBL220254 | {2'-[(3,4,5-trihydroxybenzoyl)oxy]-...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human L-selectin after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50060514((S)-4-Methylcarbamoyl-4-[(R)-2-(2-tetradecyl-hexad...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of Selectin L bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50205394((5-{2-[(2',3',4'-trihydroxy-biphenyl-4-carbonyl)-a...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human L-selectin after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50205403(5-{2-[(2'3',4'-hydroxy-biphenyl-3-carbonyl)-amino]...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human L-selectin after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50060515((S)-4-Methylcarbamoyl-4-[(S)-2-(2-tetradecyl-hexad...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of Selectin L bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50205375(CHEMBL220419 | {3-[3-(3,4,5-trihydroxy-phenyl)-pro...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of human L-selectin after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50091501(3-[(2S,5R)-3,6-Dioxo-7-(2-tetradecyl-hexadecyl)-5-...)
Affinity DataIC50:  2.34E+3nMAssay Description:In vitro inhibitory activity of compound was determined against Selectin L binding by ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50067552(2-[(R)-2-(2-Tetradecyl-hexadecanoylamino)-3-(3,4,5...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of Selectin L bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50072621(CHEMBL112485 | [4-Methoxy-3-(3,4,5-trihydroxy-6-me...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibitory activity of the compound against L-selectin IgG chimeras binding to sLex coating 96 wells using competitive cell-free ELISA assay was dete...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50205384((5-{2-[2-(3,4,5-trihydroxy-phenyl)-acetylamino]-ph...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of human L-selectin after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50205370(4-{[2-(3,4,5-trihydroxy-phenyl)-acetylamino]-methy...)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of human L-selectin after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50067553(CHEMBL133134 | N-Methyl-3-[(R)-2-(2-tetradecyl-hex...)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of Selectin L bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50091500((R)-4-Methylcarbamoyl-4-[(S)-2-(2-tetradecyl-hexad...)
Affinity DataIC50:  4.00E+3nMAssay Description:In vitro inhibitory activity of compound was determined against Selectin L binding by ELISA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50422276(CHEMBL2303755)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of Selectin L bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50422275(CHEMBL2303665)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of Selectin L bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50205371(4-methyl-3-[3-(3,4,5-trihydroxy-phenyl)-propionyla...)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of human L-selectin after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50205374((5-{2-[3-(2,3,4-trihydroxy-phenyl)-acryloylamino]-...)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of human L-selectin after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50422275(CHEMBL2303665)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibition of Selectin L bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50205401(4-{[3-(3,4,5-trihydroxy-phenyl)-propionylamino]-me...)
Affinity DataIC50:  5.70E+3nMAssay Description:Inhibition of human L-selectin after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Mus musculus)
Kanebo

Curated by ChEMBL
LigandPNGBDBM50060514((S)-4-Methylcarbamoyl-4-[(R)-2-(2-tetradecyl-hexad...)
Affinity DataIC50:  6.00E+3nMAssay Description:Blocking activity using seletin-IgG chimeras in a Selectin L competitive binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50205376((2'-{[(3,4,5-trihydroxyphenyl)acetyl]amino}-1,1'-b...)
Affinity DataIC50:  8.70E+3nMAssay Description:Inhibition of human L-selectin after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Mus musculus)
Kanebo

Curated by ChEMBL
LigandPNGBDBM50060511((R)-4-Methylcarbamoyl-4-[(S)-2-(2-tetradecyl-hexad...)
Affinity DataIC50:  9.40E+3nMAssay Description:Blocking activity using seletin-IgG chimeras in a Selectin L competitive binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50205392((5-{2-[2-(2',3',4'-trihydroxy-biphenyl-3-yl)-acety...)
Affinity DataIC50:  9.70E+3nMAssay Description:Inhibition of human L-selectin after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50205389((5-{2-[(2',3',4'-trihydroxy-biphenyl-3-carbonyl)-a...)
Affinity DataIC50:  9.80E+3nMAssay Description:Inhibition of human L-selectin after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50072618(1-[4-Methoxy-3-(3,4,5-trihydroxy-tetrahydro-pyran-...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibitory activity of the compound against L-selectin IgG chimeras binding to sLex coating 96 wells using competitive cell-free ELISA assay was dete...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50067554(4-Methylcarbamoyl-4-[(R)-3-(3,4,5-trihydroxy-6-met...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of Selectin L bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50205395((5-{2-[3-(3,4,5-trihydroxy-phenyl)-propionylamino]...)
Affinity DataIC50:  1.36E+4nMAssay Description:Inhibition of human L-selectin after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50205404((5-{2-[2-(2,3,4-trihydroxy-phenyl)-acetylamino]-ph...)
Affinity DataIC50:  1.46E+4nMAssay Description:Inhibition of human L-selectin after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50205386(2,3,4-trihydroxybenzoic acid | CHEMBL220779)
Affinity DataIC50:  1.52E+4nMAssay Description:Inhibition of human L-selectin after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Mus musculus)
Kanebo

Curated by ChEMBL
LigandPNGBDBM50060515((S)-4-Methylcarbamoyl-4-[(S)-2-(2-tetradecyl-hexad...)
Affinity DataIC50:  1.80E+4nMAssay Description:Blocking activity using seletin-IgG chimeras in a Selectin L competitive binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50205391((5-{2-[3-(3,4,5-trihydroxy-phenyl)-acryloylamino]-...)
Affinity DataIC50:  2.13E+4nMAssay Description:Inhibition of human L-selectin after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50205373(4-{[2-(3,4,5-trihydroxy-phenyl)-acetylamino]-methy...)
Affinity DataIC50:  2.62E+4nMAssay Description:Inhibition of human L-selectin after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50085536(3,4,5-Trihydroxybenzoate, X | 3,4,5-trihydroxybenz...)
Affinity DataIC50:  2.76E+4nMAssay Description:Inhibition of human L-selectin after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Mus musculus)
Kanebo

Curated by ChEMBL
LigandPNGBDBM50408284(CHEMBL2029056)
Affinity DataIC50:  3.00E+4nMAssay Description:Blocking activity using seletin-IgG chimeras in a Selectin L competitive binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50050500(CHEMBL3085443 | Sodium; 3,5-dihydroxy-2-[5-hydroxy...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibitory concentration against blocking of Selectin L during migration of inflammatory cells to inflammatory siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50408284(CHEMBL2029056)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of Selectin L bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50408284(CHEMBL2029056)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibitory activity against Selectin L expressed in endothelial cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50205393(4-{[3-(3,4,5-trihydroxy-phenyl)-propionylamino]-me...)
Affinity DataIC50:  3.08E+4nMAssay Description:Inhibition of human L-selectin after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50050461(5-(2-{2-[5-Acetylamino-2-hydroxymethyl-4-(2,3,4-tr...)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibitory activity against human chimeric L-selectin-IgMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50403679(CHEMBL2111731)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibitory activity of the compound against L-selectin IgG chimeras binding to sLex coating 96 wells using competitive cell-free ELISA assay was dete...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50205381((5-{2-[(3',4',5'-trihydroxy-biphenyl-3-carbonyl)-a...)
Affinity DataIC50:  3.76E+4nMAssay Description:Inhibition of human L-selectin after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50205372(5-methylbenzene-1,2,3-triol | CHEMBL374735)
Affinity DataIC50:  3.85E+4nMAssay Description:Inhibition of human L-selectin after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Mus musculus)
Kanebo

Curated by ChEMBL
LigandPNGBDBM50060512((R)-4-Methylcarbamoyl-4-[(R)-2-(2-tetradecyl-hexad...)
Affinity DataIC50:  3.90E+4nMAssay Description:Blocking activity using selectin-IgG chimeras in a Selectin L competitive binding assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-selectin(Homo sapiens (Human))
Kanebo

Curated by ChEMBL
LigandPNGBDBM50422136(CHEMBL2303852)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibitory concentration against blocking of Selectin L during migration of inflammatory cells to inflammatory siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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