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Found 32 Enz. Inhib. hit(s) with Target = 'Signal peptidase I'
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50501358(CHEMBL3947604)
Affinity DataIC50:  6nMAssay Description:Inhibition of full length Escherichia coli His6-tagged LepB expressed in Escherichia coli C43(DE3) using dabcyl-VEVGGTATAGAFSRPGLE-(EDANS) as substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50469157(CHEMBL4284736)
Affinity DataIC50:  6nMAssay Description:Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50501352(CHEMBL3922978)
Affinity DataIC50:  12nMAssay Description:Inhibition of full length Escherichia coli His6-tagged LepB expressed in Escherichia coli C43(DE3) using dabcyl-VEVGGTATAGAFSRPGLE-(EDANS) as substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50469159(CHEMBL4283840)
Affinity DataIC50:  17nMAssay Description:Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50501354(CHEMBL3934222)
Affinity DataIC50:  18nMAssay Description:Inhibition of full length Escherichia coli His6-tagged LepB expressed in Escherichia coli C43(DE3) using dabcyl-VEVGGTATAGAFSRPGLE-(EDANS) as substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50469154(CHEMBL4283678)
Affinity DataIC50:  29nMAssay Description:Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50469162(CHEMBL4282733)
Affinity DataIC50:  41nMAssay Description:Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50469165(CHEMBL4291540)
Affinity DataIC50:  41nMAssay Description:Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50469170(CHEMBL4291025)
Affinity DataIC50:  42nMAssay Description:Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50501357(CHEMBL3957297)
Affinity DataIC50:  48nMAssay Description:Inhibition of full length Escherichia coli His6-tagged LepB expressed in Escherichia coli C43(DE3) using dabcyl-VEVGGTATAGAFSRPGLE-(EDANS) as substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50469166(CHEMBL4294422)
Affinity DataIC50:  52nMAssay Description:Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50469169(CHEMBL4292925)
Affinity DataIC50:  72nMAssay Description:Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50469164(CHEMBL4287199)
Affinity DataIC50:  98nMAssay Description:Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50469160(CHEMBL4280386)
Affinity DataIC50:  104nMAssay Description:Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50469167(CHEMBL4279276)
Affinity DataIC50:  105nMAssay Description:Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50469161(CHEMBL4290610)
Affinity DataIC50:  107nMAssay Description:Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50501351(CHEMBL3924425)
Affinity DataIC50:  110nMAssay Description:Inhibition of full length Escherichia coli His6-tagged LepB expressed in Escherichia coli C43(DE3) using dabcyl-VEVGGTATAGAFSRPGLE-(EDANS) as substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50469163(CHEMBL4282334)
Affinity DataIC50:  175nMAssay Description:Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50480585(CHEMBL555725)
Affinity DataIC50:  180nMAssay Description:Inhibition of Escherichia coli signal peptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50469168(CHEMBL4281328)
Affinity DataIC50:  225nMAssay Description:Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50469156(CHEMBL4291944)
Affinity DataIC50:  227nMAssay Description:Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50501353(CHEMBL3895001)
Affinity DataIC50:  230nMAssay Description:Inhibition of full length Escherichia coli His6-tagged LepB expressed in Escherichia coli C43(DE3) using dabcyl-VEVGGTATAGAFSRPGLE-(EDANS) as substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50469158(CHEMBL4280228)
Affinity DataIC50:  495nMAssay Description:Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50501356(CHEMBL2306366)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of full length Escherichia coli His6-tagged LepB expressed in Escherichia coli C43(DE3) using dabcyl-VEVGGTATAGAFSRPGLE-(EDANS) as substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50469155(CHEMBL4288133)
Affinity DataIC50:  1.66E+3nMAssay Description:Inhibition of Escherichia coli type 1 signal peptidase lepB preincubated for 10 mins followed by Dabcyl-VGGTATAYGAFSRPGLE-(EDANS)-OH substrate additi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal peptidase IB(Staphylococcus aureus)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50441139(ARYLOMYCIN C16)
Affinity DataIC50:  1.80E+3nMAssay Description:Binding affinity to Staphylococcus aureus type-1 signal peptidase using decanoyl-LSSPAYNO2A-ADKabzPD and decanyol-LTPTAYNO2A-ASKKabzDD as substrate b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50501356(CHEMBL2306366)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibition of full length Escherichia coli His6-tagged LepB expressed in Escherichia coli C43(DE3) using dabcyl-VEVGGTATAGAFSRPGLE-(EDANS) as substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50480486(CHEMBL539137)
Affinity DataIC50:  1.34E+4nMAssay Description:Inhibition of Escherichia coli type I signal peptidase lepBMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50480486(CHEMBL539137)
Affinity DataIC50:  1.34E+4nMAssay Description:Inhibition of Escherichia coli type I signal peptidase lepBMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50501355(CHEMBL3952118)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of full length Escherichia coli His6-tagged LepB expressed in Escherichia coli C43(DE3) using dabcyl-VEVGGTATAGAFSRPGLE-(EDANS) as substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50441139(ARYLOMYCIN C16)
Affinity DataKd:  39nMAssay Description:Binding affinity to full length His-tagged Escherichia coli PAS0232 SPase 1 P84S mutant expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSignal peptidase I(Escherichia coli (strain K12))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50441139(ARYLOMYCIN C16)
Affinity DataKd:  979nMAssay Description:Binding affinity to full length His-tagged Escherichia coli MG1665 SPase 1 expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed