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Found 1 Enz. Inhib. hit(s) with Target = 'Protein-glutamine gamma-glutamyltransferase 2/Tyrosine-protein kinase JAK3'
TargetProtein-glutamine gamma-glutamyltransferase 2/Tyrosine-protein kinase JAK3(Homo sapiens (Human))
Duke University Medical Center

LigandPNGBDBM81345(Z4626 (ZM 39923))
Affinity DataIC50:  10nMT: 2°CAssay Description:In order to eliminated fluorescence interference, chemicals were subjected to a secondary screening using colorimetric BP incorporation assay. TGase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed