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Found 35 Enz. Inhib. hit(s) with Target = 'DNA nucleotidylexotransferase'
TargetDNA nucleotidylexotransferase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50442248(CHEMBL2441983)
Affinity DataKi:  400nMAssay Description:Non-competitive inhibition of human TdT using 3'-OH as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50442215(CHEMBL2441974)
Affinity DataKi:  450nMAssay Description:Competitive inhibition of human TdT using TTP as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50442215(CHEMBL2441974)
Affinity DataKi:  500nMAssay Description:Non-competitive inhibition of human TdT using 3'-OH as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50442248(CHEMBL2441983)
Affinity DataKi:  500nMAssay Description:Competitive inhibition of human TdT using TTP as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50442209(CHEMBL2441980)
Affinity DataKi:  1.50E+3nMAssay Description:Competitive inhibition of human TdT using TTP as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50442209(CHEMBL2441980)
Affinity DataKi:  1.70E+3nMAssay Description:Non-competitive inhibition of human TdT using 3'-OH as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50143524((3aR,4R,7R,7aS)-3,5-Dihexadecyl-3a,4,7,7a-tetrahyd...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibitory activity of the compound against human terminal deoxynucleotidyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184755((3aS,4S,7R,7aR)-1,6-dihexadecyl-2,7-bis(methoxycar...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of human TdTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Bos taurus)
Kyoto Prefectural University

Curated by ChEMBL
LigandPNGBDBM50356642(CHEMBL1917196)
Affinity DataIC50:  8.40E+3nMAssay Description:Inhibition of calf thymus TdT using oligo(dT)18 (3'-OH) and dTTP as the DNA template-primer and nucleotide substrate after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184758((3aS,4S,7R,7aR)-1,6-didodecyl-2,7-bis(methoxycarbo...)
Affinity DataIC50:  8.60E+3nMAssay Description:Inhibition of human TdTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Bos taurus)
Kyoto Prefectural University

Curated by ChEMBL
LigandPNGBDBM50356643(CHEMBL1917198)
Affinity DataIC50:  1.19E+4nMAssay Description:Inhibition of calf thymus TdT using oligo(dT)18 (3'-OH) and dTTP as the DNA template-primer and nucleotide substrate after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184753((1R,1bR,2R,5S,5aS)-1a,3-dihexadecyl-6-oxo-1a,1b,2,...)
Affinity DataIC50: >1.25E+4nMAssay Description:Inhibition of human TdTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184761((3aR,4R,7S,7aS)-dimethyl 3,5-dihexadecyl-1-oxo-7-(...)
Affinity DataIC50: >1.25E+4nMAssay Description:Inhibition of human TdTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50143526(CHEMBL366792 | Untenone A)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibitory activity of the compound against human terminal deoxynucleotidyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50143528((1S,2S)-2-Hexadecyl-2-methoxymethoxy-5-oxo-cyclope...)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibitory activity of the compound against human terminal deoxynucleotidyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184752((3aS,4S,7R,7aR)-1,6-dihexadecyl-2,7-bis(isopropoxy...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of human TdTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184748((2S,3S,4R)-methyl 2-ethyl-4-hydroxy-5-(2-oxononade...)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of human TdTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184757((3aR,4R,7S,7aS)-7-ethyl 2,4-dimethyl 3,5-dihexadec...)
Affinity DataIC50:  3.97E+4nMAssay Description:Inhibition of human TdTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184756((3aR,4S,7S,7aS)-7-ethyl 2,4-dimethyl 3,5-dihexadec...)
Affinity DataIC50:  4.84E+4nMAssay Description:Inhibition of human TdTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184759((2R,3S,4R)-methyl 1-(2-(1H-indol-3-yl)ethyl)-4-hyd...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human TdTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184760((2S,3S,4S)-methyl 1-benzyl-2-ethyl-4-hydroxy-5-(2-...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human TdTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184750((2R,3S,4R)-4-hydroxy-5-[2-oxo-nonadec-ylidene]-1-p...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human TdTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184751((2S,3S,4R)-methyl 2-ethyl-4-hydroxy-5-(2-oxotetrad...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human TdTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184749((2S,3S,4R)-methyl 1-benzyl-2-ethyl-4-hydroxy-5-(2-...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human TdTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50184763((3aS,4S,7R,7aR)-1,6-diethyl-2,7-bis(methoxycarbony...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human TdTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50143527((1R,2S)-2-Hexadecyl-5-oxo-cyclopent-3-enecarboxyli...)
Affinity DataIC50:  8.40E+4nMAssay Description:Inhibitory activity of the compound against human terminal deoxynucleotidyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50143523(2-Hexadecyl-5-oxo-cyclopent-1-enecarboxylic acid m...)
Affinity DataIC50:  1.29E+5nMAssay Description:Inhibitory activity of the compound against human terminal deoxynucleotidyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Bos taurus)
Kyoto Prefectural University

Curated by ChEMBL
LigandPNGBDBM50448691(CHEMBL3127729)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of calf thymus TdT assessed as inhibition of incorporation of dTTP into oligo(dT)18(3'OH) after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Bos taurus)
Kyoto Prefectural University

Curated by ChEMBL
LigandPNGBDBM50448688(Pecilocin | Variotin)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of calf thymus TdT assessed as inhibition of incorporation of dTTP into oligo(dT)18(3'OH) after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Bos taurus)
Kyoto Prefectural University

Curated by ChEMBL
LigandPNGBDBM50379294(CHEMBL2011647)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of calf TdT assessed as inhibition of incorporation of dTTP into oligo(dT)18(3'OH) after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Bos taurus)
Kyoto Prefectural University

Curated by ChEMBL
LigandPNGBDBM50379293(CHEMBL2011648)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of calf TdT assessed as inhibition of incorporation of dTTP into oligo(dT)18(3'OH) after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Bos taurus)
Kyoto Prefectural University

Curated by ChEMBL
LigandPNGBDBM50379292(CHEMBL2011646)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of calf TdT assessed as inhibition of incorporation of dTTP into oligo(dT)18(3'OH) after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Bos taurus)
Kyoto Prefectural University

Curated by ChEMBL
LigandPNGBDBM50448690(CHEMBL3127728)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of calf thymus TdT assessed as inhibition of incorporation of dTTP into oligo(dT)18(3'OH) after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Bos taurus)
Kyoto Prefectural University

Curated by ChEMBL
LigandPNGBDBM50448689(CHEMBL3127730)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of calf thymus TdT assessed as inhibition of incorporation of dTTP into oligo(dT)18(3'OH) after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA nucleotidylexotransferase(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50143525((R)-4-Hexadecyl-4-hydroxy-cyclopent-2-enone | CHEM...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibitory activity of the compound against human terminal deoxynucleotidyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed