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Found 22 Enz. Inhib. hit(s) with Target = 'Potassium voltage-gated channel subfamily A member 4'
TargetPotassium voltage-gated channel subfamily A member 4(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50279106(4-(4-phenoxybutoxy)-7H-furo[3,2-g]chromen-7-one | ...)
Affinity DataIC50:  170nMAssay Description:Inhibition of human Kv1.4 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 4(Rattus norvegicus)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456982(CHEMBL4208517)
Affinity DataIC50:  230nMAssay Description:Inhibition of rat Kv1.4 expressed in Xenopus laevis oocytes at -90 mV holding potential by two-electrode voltage clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 4(Rattus norvegicus)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456975(CHEMBL4213446)
Affinity DataIC50:  380nMAssay Description:Inhibition of rat Kv1.4 expressed in Xenopus laevis oocytes at -90 mV holding potential by two-electrode voltage clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 4(Rattus norvegicus)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456976(CHEMBL4207745)
Affinity DataIC50:  600nMAssay Description:Inhibition of rat Kv1.4 expressed in Xenopus laevis oocytes at -90 mV holding potential by two-electrode voltage clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 4(Rattus norvegicus)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456969(CHEMBL4202870)
Affinity DataIC50:  730nMAssay Description:Inhibition of rat Kv1.4 expressed in Xenopus laevis oocytes at -90 mV holding potential by two-electrode voltage clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 4(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456976(CHEMBL4207745)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human Kv1.4 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 4(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50220547(4,5-Dibromo-1H-pyrrole-2-carboxylic acid [3-(2-ami...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of human Kv1.4 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 4(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456974(CHEMBL3621636)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of human Kv1.4 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 4(Rattus norvegicus)
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50220547(4,5-Dibromo-1H-pyrrole-2-carboxylic acid [3-(2-ami...)
Affinity DataIC50:  5.70E+3nMAssay Description:Inhibition of rat Kv1.4 expressed in Xenopus laevis oocytes at -90 mV holding potential by two-electrode voltage clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 4(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456970(CHEMBL3261431)
Affinity DataIC50:  8.80E+3nMAssay Description:Inhibition of human Kv1.4 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 4(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456975(CHEMBL4213446)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of human Kv1.4 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 4(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456982(CHEMBL4208517)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of human Kv1.4 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 4(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456977(CHEMBL3261430)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of human Kv1.4 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 4(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456969(CHEMBL4202870)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of human Kv1.4 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 4(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456971(CHEMBL4210636)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of human Kv1.4 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 4(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50237157(CHEMBL4079366)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of Kv1.4 (unknown origin) expressed in HEK293 cells by whole cell patch clamp Qpatch methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 4(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456973(Clathrodin)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human Kv1.4 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 4(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50375409(CHEMBL408488)
Affinity DataEC50:  2.30E+3nMAssay Description:Inhibition of Kv1.4 channel inactivation expressed in xenopus oocytes by voltage clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 4(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50182585(5-acetyl-7-(4'-bromo)benzyloxy-6-hydroxy-4-methoxy...)
Affinity DataEC50:  4.30E+3nMAssay Description:Effect on blockade of Kv1.4 channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 4(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50182597(5-acetyl-4,7-benzyloxy-6-hydroxybenzofuran | CHEMB...)
Affinity DataEC50: >2.00E+4nMAssay Description:Effect on blockade of Kv1.4 channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 4(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50182587(5-acetyl-4-(4'-chloro)benzyloxy-6-hydroxy-7-methox...)
Affinity DataEC50:  4.80E+3nMAssay Description:Effect on blockade of Kv1.4 channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 4(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50375408(CHEMBL259345)
Affinity DataEC50:  1.30E+3nMAssay Description:Inhibition of Kv1.4 channel inactivation expressed in xenopus oocytes by voltage clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed