Query String: DOPAMINE
- dopamine d1
- dopamine d1b
- dopamine d2
- dopamine d3
- dopamine d4
- dopamine d4.4
- dopamine d5
- dopamine receptor
- dopamine transporter
- d1 dopamine receptor
- dopamine beta-hydroxylase
- dopamine d1 low
- dopamine d1 receptor
- dopamine d2 long
- dopamine d2 receptor
- dopamine d2 short
- dopamine d3 receptor
- dopamine d4 receptor
- dopamine d5 receptor
- dopamine receptor d2
- dopamine receptor d3
- dopamine receptor d4
- dopamine transporter (dat)
- d(1) dopamine receptor
- d(1a) dopamine receptor
- d(1b) dopamine receptor
- d(2) dopamine receptor
- d(2c) dopamine receptor
- d(3) dopamine receptor
- d(4) dopamine receptor
- d(5) dopamine receptor
- dopamine d2 receptor (d2r)
- dopamine d2 s receptor
- monoamine transporters; norepininephrine & dopamine
- sodium-dependent dopamine transporter
- soluble dopamine beta-hydroxylase
- sodium-dependent dopamine transporter (dat)
- d(1a)/d(2) dopamine receptor
- d(4) dopamine receptor [281-332]
- dopamine d2 receptor and serotonin 1a receptor
- dopamine receptor d2l/neurotensin receptor nts1
- d(2) dopamine receptor/metabotropic glutamate receptor 5
- dopamine d2 receptor/serotonin 2 (5-ht2) receptor
NPA+ (GTP+) Dopamine+ (GTP+) Dopamine+GTP BDBM81874
Oleoyl dopamine cid_5282106 N-oleoyl-dopamine BDBM50215899 CHEMBL250711
Dopamine+ (GTP-) BDBM81995
BDBM50049797 (3,4-dihydroxyphenethyl)ammonium DOPAMINE
Arachidonoyl dopamine N-arachidonoyl-dopamine (NADA) CHEMBL138921 (5Z,8Z,11Z,14Z)-N-[2-(3,4-dihydroxyphenyl)ethyl]icosa-5,8,11,14-tetraenamide BDBM20462
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- ChEMBL_62801 Inhibition of dopamine uptake at dopamine transporter.
- ChEMBL_405516 Inhibition of [3H]dopamine uptake at dopamine transporter
- ChEMBL_582830 Inhibition of [3H]dopamine reuptake at dopamine transporter
- ChEMBL_62170 Inhibition of [3H]dopamine uptake at the dopamine transporter.
- ChEMBL_62182 Inhibition of [3H]-dopamine uptake at dopamine transporter.
- ChEMBL_62183 Inhibition of [3H]dopamine uptake at dopamine transporter.
- ChEMBL_62798 Inhibition of [3H]dopamine uptake at the dopamine transporter.
- ChEMBL_62800 Inhibition of [3H]dopamine uptake at dopamine transporter.
- ChEBML_61651 Ability to inhibit the reuptake of dopamine at human dopamine transporter
- ChEMBL_351280 Inhibition of dopamine reuptake at human recombinant dopamine transporter
- ChEMBL_62972 Inhibition of dopamine uptake from dopamine uptake site
- ChEMBL_62636 Inhibition of [3H]dopamine uptake via rat dopamine receptor.
- ChEBML_62638 Inhibition of [3H]dopamine uptake at striatal nerve endings by dopamine transporter
- ChEMBL_216109 Inhibition of [3H]dopamine binding to dopamine receptor of rat corpus striatum
- ChEMBL_216110 Inhibition of [3H]dopamine binding to dopamine receptor of rat corpus striatum
- ChEMBL_59592 Inhibition of [3H]dopamine binding to Dopamine receptor in calf caudate nuclei.
- ChEMBL_61987 Inhibition of [3H]dopamine uptake at the dopamine transporter in rat striatal tissue
- ChEMBL_62476 Inhibition of [3H]dopamine binding to rat striatal synaptosome dopamine transporter
- ChEMBL_62638 Inhibition of [3H]dopamine uptake at striatal nerve endings by dopamine transporter
- ChEMBL_654116 Inhibition of dopamine reuptake at human dopamine transporter expressed in CHO cells
- ChEBML_60524 Dopamine agonist (Dopamine receptor D1) activity was measured as increase in cAMP formation relative to maximum increase in dopamine-sensitive adenylate cyclase
- ChEBML_58796 The binding affinity was measured on dopamine receptor D1 using [3H]- dopamine as radioligand.
- ChEBML_60499 In vitro binding affinity of compound against dopamine neuronal Dopamine receptor D1
- ChEBML_61514 Inhibition of [3H]dopamine uptake in HEK cells expressing human Dopamine transporter
- ChEBML_62496 Ability to inhibit reuptake of dopamine ([3H]DA) at dopamine transporter of rat striatum
- ChEBML_62899 The binding affinity was measured on dopamine receptor D3 using [3H]- dopamine as radioligand.
- ChEMBL_1615836 Inhibition of dopamine transporter (unknown origin) assessed as suppression of synaptosomal uptake of dopamine
- ChEMBL_306589 Inhibition of [3H]dopamine uptake in HEK293 cells expressing human dopamine transporter
- ChEMBL_339939 Inhibition of dopamine re-uptake at human dopamine transporter expressed in HEK293 cells
- ChEMBL_463819 Inhibition of [3H]dopamine uptake at human dopamine transporter expressed in HEK293 cells
- ChEMBL_58796 The binding affinity was measured on dopamine receptor D1 using [3H]- dopamine as radioligand.
- ChEMBL_608505 Inhibition of [3H]dopamine reuptake at rat brain frontal cortex dopamine transporter
- ChEMBL_61503 Inhibition of dopamine uptake in HEK cells expressing human dopamine transporter (hDAT)
- ChEMBL_61511 Inhibition of [3H]dopamine reuptake in HEK293 cells expressing human dopamine transporter
- ChEMBL_61512 Inhibition of dopamine (DA) reuptake using cloned human dopamine transporter was determined
- ChEMBL_61514 Inhibition of [3H]dopamine uptake in HEK cells expressing human Dopamine transporter
- ChEMBL_62302 Inhibition of dopamine uptake into rat striatal tissue, using [3H]- dopamine as the radioligand.
- ChEMBL_62496 Ability to inhibit reuptake of dopamine ([3H]DA) at dopamine transporter of rat striatum
- ChEMBL_62899 The binding affinity was measured on dopamine receptor D3 using [3H]- dopamine as radioligand.
- ChEMBL_839139 TP_TRANSPORTER: inhibition of Dopamine uptake (Dopamine: 200 uM) in Xenopus laevis oocytes
- ChEMBL_761552 Inhibition of dopamine transporter
- ChEBML_177229 Inhibition of dopamine uptake in synaptosomal preparation in rat corpus striatum, using [3H]dopamine
- ChEMBL_177229 Inhibition of dopamine uptake in synaptosomal preparation in rat corpus striatum, using [3H]dopamine
- ChEMBL_59582 Evaluated for the inhibition of binding of [3H]DA (dopamine) to dopamine receptor in calf striatal homogenate
- ChEMBL_60008 Evaluated for the inhibition of binding of [3H]DA (dopamine) to dopamine receptor in rat brain homogenate
- ChEMBL_61854 Compound was tested for Inhibition of [3H]dopamine uptake at the dopamine transporter in rat strial tissue
- ChEMBL_61986 Compound was tested for inhibition of [3H]dopamine uptake at the dopamine transporter in rat strial tissue
- ChEMBL_59586 In vitro inhibitory activity was evaluated against [3H]dopamine (DA) calf caudate dopamine receptor
- ChEMBL_59588 In vitro inhibitory activity was evaluated against,[3H]dopamine (DA),calf caudate dopamine receptor
- ChEBML_305233 Inhibition of dopamine D3 receptor
- ChEBML_305234 Inhibition of dopamine D4 receptor
- ChEBML_58646 Affinity for Dopamine receptor D1
- ChEBML_59102 Inhibition of Dopamine beta hydroxylase.
- ChEBML_62390 Affinity for Dopamine receptor D2
- ChEMBL_1554623 Inhibition of human dopamine transporter
- ChEMBL_447510 Inhibition of dopamine D2 receptor
- ChEMBL_447511 Inhibition of dopamine D3 receptor
- ChEMBL_458979 Inhibition of dopamine D2 receptor
- ChEMBL_458981 Binding affinity to dopamine transporter
- ChEMBL_476019 Inhibition of dopamine D1 receptor
- ChEMBL_476020 Inhibition of dopamine D2 receptor
- ChEMBL_514038 Inhibition of dopamine D2 receptor
- ChEMBL_520034 Binding affinity to dopamine transporter
- ChEMBL_532090 Inhibition of dopamine uptake at DAT
- ChEMBL_536127 Inhibition of dopamine D2 receptor
- ChEMBL_539365 Binding affinity to dopamine transporter
- ChEMBL_579693 Inhibition of human dopamine transporter
- ChEMBL_59102 Inhibition of Dopamine beta hydroxylase.
- ChEMBL_592332 Inhibition of dopamine D1 receptor
- ChEMBL_592333 Inhibition of dopamine D2 receptor
- ChEMBL_592334 Inhibition of dopamine D3 receptor
- ChEMBL_59302 Inhibition of dopamine beta hydroxylase
- ChEMBL_601708 Inhibition of dopamine D1 receptor
- ChEMBL_601709 Inhibition of dopamine D2 receptor
- ChEMBL_601710 Inhibition of dopamine D5 receptor
- ChEMBL_615841 Inhibition of dopamine D2 receptor
- ChEMBL_615842 Inhibition of dopamine D3 receptor
- ChEMBL_617090 Inhibition of dopamine D2 receptor
- ChEMBL_617091 Inhibition of dopamine D3 receptor
- ChEMBL_617092 Inhibition of dopamine D4 receptor
- ChEMBL_61988 Inhibition of dopamine DA reuptake
- ChEMBL_622531 Inhibition of human dopamine transporter
- ChEMBL_624451 Inhibition of dopamine D2 (receptor)
- ChEMBL_624452 Inhibition of dopamine D3 (receptor)
- ChEMBL_624453 Inhibition of dopamine D4 (receptor)
- ChEMBL_62478 Binding affinity for dopamine transporter
- ChEMBL_62951 Concentration inhibiting Dopamine transporter
- ChEMBL_630143 Inhibition of dopamine D1 receptor
- ChEMBL_630144 Inhibition of dopamine D2 receptor
- ChEMBL_630145 Inhibition of dopamine D3 receptor
- ChEMBL_649503 Inhibition of dopamine D2 receptor
- ChEMBL_649646 Binding affinity to dopamine D2
- ChEMBL_685495 Binding affinity to dopamine D1
- ChEMBL_685496 Binding affinity to dopamine D2
- ChEMBL_700864 Inhibition of dopamine D3 receptor
- ChEMBL_700868 Inhibition of dopamine D5 receptor
- ChEMBL_714780 Inhibition of human dopamine transporter
- ChEMBL_747461 Inhibition of dopamine D4 receptor
- ChEMBL_795936 Inhibition of dopamine D2 receptor
- ChEMBL_820281 Inhibition of D2 dopamine receptor
- ChEMBL_820282 Inhibition of D3 dopamine receptor
- ChEMBL_820284 Inhibition of D5 dopamine receptor
- ChEMBL_875717 Binding affinity to dopamine transporter
- ChEMBL_946917 Inhibition of human dopamine transporter
- ChEMBL_571436 Inhibition of [3H]dopamine uptake at human dopamine transporter expressed in mouse N2A cells by scintillation counting
- ChEMBL_58663 Dopamine receptor D1 antagonistic activity as ability to block dopamine-stimulated adenylate cyclase in rat caudate
- ChEMBL_59584 In vitro inhibitory activity against dopamine receptor from calf caudate using [3H]dopamine as radioligand
- ChEMBL_60523 Dopamine D1 agonist efficacy was measured with stimulation of dopamine-sensitive rat adenylate cyclase in caudate membranes
- ChEMBL_61686 Inhibitory activity against [3H]-Dopamine uptake from Dopamine transporter in rat caudate putamen tissue
- ChEMBL_61690 Inhibitory activity against [3H]dopamine uptake from Dopamine transporter in rat caudate putamen tissue
- ChEMBL_62144 Inhibition of high-affinity uptake of [3H]dopamine at dopamine transporter into rat striatal nerve endings (synaptosomes)
- ChEMBL_62174 Reuptake inhibition at the dopamine transporter labeled with radioligand [3H]dopamine on synaptosomes obtained from rat caudate.
- ChEBML_58154 Dopamine receptor D1 agonist efficacy was measured with stimulation of dopamine-sensitive rat adenylate cyclase in caudate membranes. Partial agonist, maximum effect 60% of dopamine maximum effect.
- ChEMBL_58154 Dopamine receptor D1 agonist efficacy was measured with stimulation of dopamine-sensitive rat adenylate cyclase in caudate membranes. Partial agonist, maximum effect 60% of dopamine maximum effect.
- ChEMBL_60526 Dopamine receptor D1 agonist efficacy was measured with stimulation of dopamine-sensitive rat adenylate cyclase in caudate membranes. Partial agonist, maximum effect 59% of dopamine maximum effect
- ChEBML_61990 Compound was tested for its ability to inhibit the neurotransmitter dopamine-DA reuptake system using [3H]dopamine as radioligand
- ChEMBL_507938 Inhibition of dopamine transporter-mediated [3H]dopamine uptake in Wistar rat striatal synaptosomes by liquid scintillation spectrometry
- ChEMBL_596936 Inhibition of dopamine reuptake at human dopamine transporter expressed in HEK293 cells after 5 mins by scintillation counting
- ChEMBL_61990 Compound was tested for its ability to inhibit the neurotransmitter dopamine-DA reuptake system using [3H]dopamine as radioligand
- ChEBML_1688592 Inhibition of human dopamine D1 receptor
- ChEBML_1688593 Inhibition of human dopamine D2 receptor
- ChEBML_1688594 Inhibition of human dopamine D3 receptor
- ChEBML_1688595 Inhibition of human dopamine D5 receptor
- ChEBML_302616 Binding affinity for dopamine D2 receptor
- ChEBML_302618 Binding affinity for dopamine D4 receptor
- ChEBML_305085 Inhibition of rat dopamine D3 receptor
- ChEBML_305086 Inhibition of rat dopamine D4 receptor
- ChEBML_58660 Binding affinity for dopamine receptor D1
- ChEBML_59436 Inhibitory activity against the dopamine decarboxylase
- ChEBML_62245 Binding affinity to dopamine receptor D2
- ChEBML_62472 Binding affinity for dopamine transporter (DAT)
- ChEBML_62576 Binding affinity for dopamine receptor D2
- ChEMBL_1339957 Inhibition of human dopamine D1 receptor
- ChEMBL_1339958 Inhibition of human dopamine D4 receptor
- ChEMBL_1439002 Inhibition of human dopamine D1 receptor
- ChEMBL_1439003 Inhibition of human dopamine D2 receptor
- ChEMBL_1439004 Inhibition of human dopamine D3 receptor
- ChEMBL_1439005 Inhibition of human dopamine D4 receptor
- ChEMBL_1439009 Inhibition of human dopamine D2L receptor
- ChEMBL_1688593 Inhibition of human dopamine D2 receptor
- ChEMBL_1688620 Inhibition of human dopamine D4 receptor
- ChEMBL_1817364 Inhibition of dopamine receptor (unknown origin)
- ChEMBL_1833862 Inhibition of dopamine transporter (unknown origin)
- ChEMBL_1859530 Inhibition of dopamine transporter (unknown origin)
- ChEMBL_2027265 Inhibition of dopamine transporter (unknown origin)
- ChEMBL_216102 The compound was tested for inhibition of dopamine reuptake
- ChEMBL_2162545 Inhibition of dopamine transporter (unknown origin)
- ChEMBL_302368 Binding affinity for Dopamine receptor D4
- ChEMBL_320747 Inhibition constant against dopamine transporter
- ChEMBL_320837 Inhibition of monoamine reuptake at dopamine transporter
- ChEMBL_321258 Inhibitory concentration against dopamine transporter
- ChEMBL_321339 Inhibitory concentration against dopamine transporter
- ChEMBL_325915 Inhibition of human dopamine receptor D1
- ChEMBL_325916 Inhibition of human dopamine receptor D2
- ChEMBL_325917 Inhibition of human dopamine receptor D3
- ChEMBL_325918 Inhibition of human dopamine receptor D4.4
- ChEMBL_328774 Binding affinity to dopamine D1 receptor
- ChEMBL_328775 Binding affinity to dopamine D2 receptor
- ChEMBL_329925 Binding affinity to dopamine D1 receptor
- ChEMBL_329926 Binding affinity to dopamine D2 receptor
- ChEMBL_329927 Binding affinity to dopamine D3 receptor
- ChEMBL_329928 Binding affinity to dopamine D4 receptor
- ChEMBL_329929 Binding affinity to dopamine D5 receptor
- ChEMBL_332082 Binding affinity to dopamine receptor D1
- ChEMBL_332083 Binding affinity to dopamine receptor D2
- ChEMBL_334933 Inhibitory activity against dopamine D1
- ChEMBL_334934 Inhibitory activity against dopamine D2
- ChEMBL_334935 Inhibitory activity against dopamine D3
- ChEMBL_391337 Binding affinity at dopamine D4 receptor
- ChEMBL_391338 Binding affinity at dopamine D2 receptor
- ChEMBL_391342 Binding affinity at dopamine D5 receptor
- ChEMBL_438895 Binding affinity for dopamine D2 receptor
- ChEMBL_449184 Activity against human dopamine transporter
- ChEMBL_458722 Binding affinity to dopamine D1 receptor
- ChEMBL_458723 Binding affinity to dopamine D5 receptor
- ChEMBL_460797 Binding affinity to dopamine D1 receptor
- ChEMBL_465424 Binding affinity to dopamine D2 receptor
- ChEMBL_474646 Binding affinity at dopamine D2 receptor
- ChEMBL_487760 Binding affinity to dopamine D2 receptor
- ChEMBL_491100 Binding affinity to dopamine D3 receptor
- ChEMBL_491101 Binding affinity to dopamine D2 receptor
- ChEMBL_492769 Antagonist activity at dopamine D2 receptor
- ChEMBL_510243 Antagonist activity at dopamine D2 receptor
- ChEMBL_514049 Agonist activity at dopamine D2 receptor
- ChEMBL_537457 Binding affinity at dopamine D2 receptor
- ChEMBL_538667 Antagonist activity at dopamine D2 receptor
- ChEMBL_538668 Antagonist activity at dopamine D3 receptor
- ChEMBL_555734 Binding affinity at dopamine D2 receptor
- ChEMBL_556740 Binding affinity to dopamine D3 receptor
- ChEMBL_556749 Binding affinity to dopamine D2 receptor
- ChEMBL_556750 Binding affinity to dopamine D1 receptor
- ChEMBL_556753 Binding affinity to dopamine D5 receptor
- ChEMBL_556760 Binding affinity to dopamine uptake transporter
- ChEMBL_58196 Inhibition of mouse Dopamine receptor D2
- ChEMBL_582222 Antagonist activity at dopamine D4 receptor
- ChEMBL_588078 Agonist activity at dopamine D1 receptor
- ChEMBL_58831 Affinity towards Dopamine receptor D1
- ChEMBL_59913 Inhibition of human dopamine receptor D2
- ChEMBL_60181 Binding affinity towards Dopamine receptor
- ChEMBL_60187 Affinity towards Dopamine receptor D1
- ChEMBL_60374 Affinity towards Dopamine receptor D2
- ChEMBL_60486 Inhibition of human dopamine receptor D1
- ChEMBL_608751 Antagonist activity at dopamine D4 receptor
- ChEMBL_608752 Agonist activity at dopamine D2 receptor
- ChEMBL_609554 Binding affinity to dopamine D1 receptor
- ChEMBL_609555 Binding affinity to dopamine D5 receptor
- ChEMBL_609556 Binding affinity to dopamine D2 receptor
- ChEMBL_609557 Binding affinity to dopamine D4 receptor
- ChEMBL_610407 Binding affinity to dopamine D2 receptor
- ChEMBL_61172 Inhibition of human dopamine receptor D4.4
- ChEMBL_61330 Inhibition of human dopamine receptor D5
- ChEMBL_61840 Binding affinity for rat Dopamine transporter.
- ChEMBL_61970 Inhibition of human dopamine receptor D3
- ChEMBL_62125 Binding affinity at dopamine receptor D3
- ChEMBL_62245 Binding affinity to dopamine receptor D2
- ChEMBL_62332 Ability to inhibition uptake of [2H]-Dopamine
- ChEMBL_62471 Binding affinity towards dopamine transporter
- ChEMBL_62819 The inhibition of reuptake against dopamine transporter
- ChEMBL_629543 Binding affinity to dopamine D3 receptor
- ChEMBL_629557 Binding affinity to dopamine D4 receptor
- ChEMBL_62968 Binding affinity against dopamine transporter
- ChEMBL_644064 Binding affinity to dopamine D1 receptor
- ChEMBL_644065 Binding affinity to dopamine D2 receptor
- ChEMBL_644069 Binding affinity to dopamine D4 receptor
- ChEMBL_652385 Binding affinity to dopamine D1 receptor
- ChEMBL_652386 Binding affinity to dopamine D2 receptor
- ChEMBL_652387 Binding affinity to dopamine D3 receptor
- ChEMBL_652388 Binding affinity to dopamine D4 receptor
- ChEMBL_652389 Binding affinity to dopamine D5 receptor
- ChEMBL_684873 Inhibition of human dopamine D2 receptor
- ChEMBL_685575 Antagonist activity at dopamine D2 receptor
- ChEMBL_697200 Binding affinity to dopamine receptor D1
- ChEMBL_697201 Binding affinity to dopamine receptor D2
- ChEMBL_697202 Binding affinity to dopamine receptor D3
- ChEMBL_697203 Binding affinity to dopamine receptor D4
- ChEMBL_697204 Binding affinity to dopamine receptor D5
- ChEMBL_699288 Binding affinity to dopamine D2 receptor
- ChEMBL_699575 Inhibition of human recombinant dopamine transporter
- ChEMBL_714776 Inhibition of human dopamine D1 receptor
- ChEMBL_714777 Inhibition of human dopamine D2 receptor
- ChEMBL_714778 Inhibition of human dopamine D3 receptor
- ChEMBL_718155 Binding affinity to dopamine D4 receptor
- ChEMBL_718156 Binding affinity to dopamine D5 receptor
- ChEMBL_718872 Binding affinity to dopamine D1 receptor
- ChEMBL_718873 Binding affinity to dopamine D2 receptor
- ChEMBL_718874 Binding affinity to dopamine D3 receptor
- ChEMBL_726928 Inhibition of human recombinant dopamine transporter
- ChEMBL_744202 Binding affinity to dopamine D3 receptor
- ChEMBL_759383 Binding affinity to dopamine 2 receptor
- ChEMBL_761642 Inhibition of recombinant human dopamine transporter
- ChEMBL_771226 Inhibition of human dopamine D2 receptor
- ChEMBL_788043 Antagonist activity at dopamine D2 receptor
- ChEMBL_794948 Binding affinity to dopamine D1 receptor
- ChEMBL_794949 Binding affinity to dopamine D2 receptor
- ChEMBL_804288 Antagonist activity at dopamine D1 receptor
- ChEMBL_804289 Antagonist activity at dopamine D2 receptor
- ChEMBL_818582 Binding affinity to dopamine D1 receptor
- ChEMBL_818583 Binding affinity to dopamine D2 receptor
- ChEMBL_849495 Binding affinity to dopamine D2 receptor
- ChEMBL_849496 Binding affinity to dopamine D3 receptor
- ChEMBL_875721 Binding affinity to dopamine D2 receptor
- ChEMBL_879204 Antagonist activity at dopamine D1 receptor
- ChEMBL_879321 Inhibition of human dopamine D5 receptor
- ChEMBL_879322 Inhibition of human dopamine D4 receptor
- ChEMBL_879323 Inhibition of human dopamine D2 receptor
- ChEMBL_879324 Inhibition of human dopamine D3 receptor
- ChEMBL_879325 Inhibition of human dopamine D1 receptor
- ChEMBL_884312 Binding affinity to D3 dopamine receptor
- ChEMBL_884318 Binding affinity to D1 dopamine receptor
- ChEMBL_884319 Binding affinity to D2 dopamine receptor
- ChEMBL_884320 Binding affinity to D4 dopamine receptor
- ChEMBL_884321 Binding affinity to D5 dopamine receptor
- ChEBML_61501 Ability to inhibit human dopamine uptake by the human dopamine transporter in EM4 cells stably infected with Flag HA-hDAT
- ChEBML_61991 Compound was tested for its ability to inhibit the uptake of [3H]dopamine in DAT (dopamine transporter system) expressing cell line
- ChEMBL_60062 Antagonism of dopamine-stimulated [35S]GTP-gamma-S binding against human Dopamine receptor D2 in CHO cells
- ChEMBL_60659 Antagonism of dopamine-stimulated [35S]GTP-gamma-S binding against human Dopamine receptor D4 in CHO cells
- ChEMBL_1356560 Inhibition of [3H]dopamine uptake at dopamine transporter expressed in rat striatal homogenate after 5 mins by scintillation counting analysis
- ChEMBL_52731 Reuptake inhibition was determined at the dopamine transporter labeled with radioligand [3H]dopamine in nonstandard conditions on brain membranes obtained from rat
- ChEMBL_62173 Reuptake inhibition was determined at the dopamine transporter labeled with radioligand [3H]dopamine in nonstandard conditions on brain membranes obtained from rat
- ChEMBL_1804344 Antagonist activity at human dopamine D1 receptor expressed in HEK293T cells assessed as inhibition of dopamine-induced cAMP accumulation preincubated for 15 mins followed by dopamine induction and measured after 30 mins by HTRF assay
- ChEBML_176345 Inhibition of dopamine uptake in rat synaptosomal fraction
- ChEBML_31418 In vitro inhibition of dopamine stimulated adenylate cyclase
- ChEBML_52581 Percent inhibition towards dopamine D2 receptor
- ChEBML_52597 Percent inhibition towards dopamine D3 receptor
- ChEBML_52724 Percent inhibition towards dopamine D4 receptor
- ChEBML_58202 Binding affinity towards Dopamine receptor D2
- ChEBML_58459 Binding affinity against dopamine D2 receptor
- ChEBML_58645 Binding affinity towards Dopamine receptor D1
- ChEBML_58971 Compound was evaluated for Dopamine receptor D1 binding
- ChEBML_59144 Binding affinity against dopamine receptor D1A
- ChEBML_59303 Inhibitory activity against the dopamine beta hydroxylase
- ChEBML_59636 Binding affinity towards Dopamine receptor D2
- ChEBML_60059 Affinity towards human dopamine receptor D2
- ChEBML_60490 Affinity towards human Dopamine receptor D1
- ChEBML_60810 Binding affinity for rat Dopamine receptor D2
- ChEBML_60811 Binding affinity for rat Dopamine receptor D2
- ChEBML_60843 Binding affinity against Dopamine receptor D4
- ChEBML_60988 Binding affinity to Dopamine receptor D4 was determined
- ChEBML_61114 Inhibitory concentration against Dopamine receptor D2
- ChEBML_61121 Binding affinity to Dopamine receptor D2 was determined
- ChEBML_61127 Compound was evaluated for Dopamine receptor D2 binding
- ChEBML_61144 Binding affinity towards dopamine receptor D2
- ChEBML_61273 Binding affinity of compound to Dopamine receptor D2
- ChEBML_61332 Affinity towards human dopamine receptor D5
- ChEBML_61647 Binding affinity against Dopamine receptor D2L
- ChEBML_62002 Effect on synaptosomal uptake inhibition of Dopamine transporter
- ChEBML_62114 Affinity towards human dopamine receptor D3
- ChEBML_62171 Inhibition of [3H]mazindol binding to the dopamine transporter.
- ChEBML_62452 Binding affinity against Dopamine receptor D3
- ChEBML_62473 Binding affinity towards dopamine transporter (DAT)
- ChEBML_62807 Displacement of [3H]mazindol from dopamine transporter
- ChEBML_62967 In vitro binding affinity for dopamine uptake site
- ChEBML_63109 Affinity towards human dopamine receptor D4
- ChEMBL_1445391 Inhibition of dopamine D2 receptor (unknown origin)
- ChEMBL_1469013 Inhibition of dopamine D1 receptor (unknown origin)
- ChEMBL_1502293 Binding affinity to human dopamine D2 receptor
- ChEMBL_1502686 Inhibition of dopamine beta-oxygenase (unknown origin)
- ChEMBL_1525544 Binding affinity to dopamine receptor (unknown origin)
- ChEMBL_1569998 Binding affinity to dopamine receptor (unknown origin)
- ChEMBL_1613487 Activity at dopamine D1 receptor (unknown origin)
- ChEMBL_1613488 Activity at dopamine D4 receptor (unknown origin)
- ChEMBL_1688623 Inhibition of human dopamine D2 (short) receptor
- ChEMBL_1722529 Inhibition of dopamine D1 receptor (unknown origin)
- ChEMBL_176345 Inhibition of dopamine uptake in rat synaptosomal fraction
- ChEMBL_1771297 Binding affinity to human dopamine D2 receptor
- ChEMBL_1771298 Binding affinity to human dopamine D3 receptor
- ChEMBL_2017999 Binding affinity to human dopamine D2 receptor
- ChEMBL_2018000 Binding affinity to human dopamine D1 receptor
- ChEMBL_2033536 Inhibition of D1 dopamine receptor (unknown origin)
- ChEMBL_2063344 Binding affinity to human dopamine D2 receptor
- ChEMBL_2109658 Inhibition of dopamine D5 receptor (unknown origin)
- ChEMBL_2109662 Inhibition of dopamine D3 receptor (unknown origin)
- ChEMBL_2109663 Inhibition of dopamine D1 receptor (unknown origin)
- ChEMBL_2134932 Binding affinity to human dopamine D3 receptor
- ChEMBL_2163944 Inhibition of dopamine D2 receptor (unknown origin)
- ChEMBL_302418 Inhibitory constant for Dopamine receptor D1-like
- ChEMBL_302443 Binding affinity for human dopamine D2 receptor
- ChEMBL_302444 Binding affinity for human dopamine receptor D3
- ChEMBL_302448 Binding affinity for rat Dopamine receptor D3
- ChEMBL_302474 Binding affinity for human Dopamine receptor D2
- ChEMBL_302580 Binding affinity for human dopamine D4 receptor
- ChEMBL_302694 Inhibitory constant against Dopamine receptor D2
- ChEMBL_302707 Binding affinity for human dopamine receptor D3
- ChEMBL_302736 Binding affinity for human dopamine D2 receptor
- ChEMBL_302737 Binding affinity for human dopamine D3 receptor
- ChEMBL_302843 Binding affinity for human dopamine D3 receptor
- ChEMBL_304000 Binding affinity for human dopamine receptor D2
- ChEMBL_304001 Binding affinity for human dopamine receptor D3
- ChEMBL_304002 Binding affinity for human dopamine receptor D4
- ChEMBL_320746 Inhibition constant against dopamine receptor D2
- ChEMBL_320765 Affinity towards cloned Dopamine receptor D1
- ChEMBL_320766 Affinity towards cloned Dopamine receptor D2
- ChEMBL_320767 Affinity towards cloned Dopamine receptor D3
- ChEMBL_320768 Affinity towards cloned Dopamine receptor D4
- ChEMBL_320769 Affinity towards cloned Dopamine receptor D5
- ChEMBL_320771 Ligand efficacy towards dopamine D3 receptor
- ChEMBL_320794 Binding inhibition towards human dopamine transporter
- ChEMBL_321093 Effective concentration against dopamine D3 receptor
- ChEMBL_321094 Effective concentration against dopamine D3 receptor
- ChEMBL_321165 Inhibitory concentration against dopamine receptor D4
- ChEMBL_321256 Inhibitory concentration against dopamine receptor D1
- ChEMBL_321257 Inhibitory concentration against dopamine receptor D3
- ChEMBL_326580 Inhibitory activity against dopamine D3 receptor
- ChEMBL_333001 Inhibitory activity against dopamine D1 receptor
- ChEMBL_333003 Inhibitory activity against dopamine D5 receptor
- ChEMBL_384221 Binding affinity to human dopamine D3 receptor
- ChEMBL_384500 Binding affinity to human dopamine D5 receptor
- ChEMBL_444279 Binding affinity to human dopamine D2 receptor
- ChEMBL_456086 Binding affinity to human dopamine D4 receptor
- ChEMBL_461996 Binding affinity to human dopamine D2 receptor
- ChEMBL_461997 Binding affinity to human dopamine D4 receptor
- ChEMBL_491873 Inhibition of dopamine uptake at human cloned DAT
- ChEMBL_512428 Displacement of radioligand from dopamine D1 receptor
- ChEMBL_512429 Displacement of radioligand from dopamine D2S receptor
- ChEMBL_512430 Displacement of radioligand from dopamine D3 receptor
- ChEMBL_552743 Binding affinity to human dopamine D2 receptor
- ChEMBL_58226 Binding affinity against dopamine D2 receptor
- ChEMBL_58312 Binding affinity against Dopamine D1 receptor
- ChEMBL_58313 Binding affinity against Dopamine D1 receptor
- ChEMBL_58468 Binding affinity towards dopamine D2 receptor
- ChEMBL_58622 Binding affinity towards dopamine D2 receptor
- ChEMBL_58625 Tested for binding affinity for Dopamine D2 receptor
- ChEMBL_58626 Tested for binding affinity for Dopamine D2 receptors
- ChEMBL_58630 Binding affinity against Dopamine D2 receptor
- ChEMBL_588133 Binding affinity to pig dopamine D1 receptor
- ChEMBL_58945 Binding affinity towards Dopamine D4 receptor
- ChEMBL_58984 Binding affinities towards Dopamine receptor D1
- ChEMBL_58985 Binding affinity against Dopamine receptor D1
- ChEMBL_58988 Binding affinity against Dopamine receptor D1
- ChEMBL_58989 Binding affinity towards Dopamine receptor D1
- ChEMBL_58998 Binding affinity against dopamine receptor D1
- ChEMBL_59428 Inhibition of dopamine beta-hydroxylase (DbetaH) enzyme
- ChEMBL_60071 Binding affinity at human dopamine receptor D2
- ChEMBL_60178 Effect on synaptosomal uptake inhibition of Dopamine receptor
- ChEMBL_60492 Binding affinity against dopamine receptor D1
- ChEMBL_60518 Binding affinity against dopamine receptor D1
- ChEMBL_60665 Binding affinity at human dopamine receptor D4
- ChEMBL_60843 Binding affinity against Dopamine receptor D4
- ChEMBL_60989 In vitro binding affinity for Dopamine receptor D4
- ChEMBL_60992 Binding affinity against Dopamine receptor D4
- ChEMBL_61119 Binding affinity towards Dopamine receptor D2
- ChEMBL_61132 In vitro binding affinity for Dopamine receptor D2
- ChEMBL_61142 Binding affinity for Dopamine receptor D2 was determined
- ChEMBL_61144 Binding affinity towards dopamine receptor D2
- ChEMBL_61147 In vitro binding affinity for Dopamine receptor D2
- ChEMBL_61284 Binding affinity against Dopamine receptor D2
- ChEMBL_61287 Binding affinity against Dopamine receptor D2
- ChEMBL_61290 Binding affinity towards Dopamine receptor D2
- ChEMBL_61315 Binding affinity against dopamine D2 receptor
- ChEMBL_61340 Binding affinity against Dopamine receptor D5
- ChEMBL_61341 Binding affinity towards Dopamine receptor D5
- ChEMBL_61350 Binding affinity against dopamine D4 receptor
- ChEMBL_61647 Binding affinity against Dopamine receptor D2L
- ChEMBL_61667 In vitro binding affinity on cloned Dopamine transporter
- ChEMBL_61763 Binding affinity against dopamine receptor D2
- ChEMBL_61803 Binding Affinity of Compound of Dopamine receptor D2S
- ChEMBL_61943 Effective concentration for Dopamine receptor D3 was determined
- ChEMBL_61945 Effective concentration for Dopamine receptor D3 was determined
- ChEMBL_62002 Effect on synaptosomal uptake inhibition of Dopamine transporter
- ChEMBL_62163 Inhibition of [3H]BTCP binding to the dopamine transporter.
- ChEMBL_62164 Inhibition of [3H]BTCP binding to the dopamine transporter.
- ChEMBL_62169 Inhibition of [3H]cocaine binding to the dopamine transporter.
- ChEMBL_62171 Inhibition of [3H]mazindol binding to the dopamine transporter.
- ChEMBL_62386 Binding affinity towards Dopamine receptor D2
- ChEMBL_62452 Binding affinity against Dopamine receptor D3
- ChEMBL_62621 Evaluated for the Competitive inhibition of uptake of dopamine transporter
- ChEMBL_62792 Inhibition of [3H]BTCP binding to the dopamine transporter.
- ChEMBL_62797 Inhibition of [3H]cocaine binding to the dopamine transporter.
- ChEMBL_62799 Inhibition of [3H]mazindol binding to the dopamine transporter.
- ChEMBL_62802 Inhibition constant of high-affinity dopamine uptake
- ChEMBL_62807 Displacement of [3H]mazindol from dopamine transporter
- ChEMBL_62814 Compound was tested for the inhibition of dopamine (DA) reuptake
- ChEMBL_62817 Inhibitory concentration against [3H]dopamine uptake
- ChEMBL_62926 Binding affinity for Dopamine receptor D3 was determined
- ChEMBL_62929 Binding affinity against Dopamine receptor D3
- ChEMBL_62930 Binding affinity against Dopamine receptor D3
- ChEMBL_62931 Binding affinity towards Dopamine receptor D3
- ChEMBL_62939 Binding affinity against dopamine D3 receptor
- ChEMBL_658549 Binding affinity to human recombinant dopamine transporter
- ChEMBL_664950 Binding affinity to rat dopamine D1 receptor
- ChEMBL_664951 Binding affinity to rat dopamine D2 receptor
- ChEMBL_664952 Binding affinity to rat dopamine D3 receptor
- ChEMBL_664953 Binding affinity to rat dopamine D4 receptor
- ChEMBL_664954 Binding affinity to human dopamine D5 receptor
- ChEMBL_767224 Inhibition of D1 dopamine receptor by NIMH PDSP
- ChEMBL_807237 Inhibition of rat DAT-mediated dopamine reuptake
- ChEMBL_816869 Binding affinity to human dopamine D3 receptor
- ChEMBL_816870 Binding affinity to human dopamine D2L receptor
- ChEMBL_816871 Binding affinity to human dopamine D2S receptor
- ChEMBL_816874 Binding affinity to rat dopamine D1 receptor
- ChEMBL_816875 Binding affinity to human dopamine D1 receptor
- ChEMBL_816877 Binding affinity to human dopamine D5 receptor
- ChEMBL_821614 Binding affinity to human dopamine D5 receptor
- ChEMBL_824329 Inhibition of rat DAT-mediated dopamine reuptake
- ChEMBL_942037 Inhibition of dopamine receptor D2 (unknown origin)
- ChEBML_58170 Affinity of the Compound for Dopamine D1 receptor in rat striatal membrane was determined in vitro using Dopamine Antagonist [3H]SCH-23390 as ligand.
- ChEMBL_1621627 Inhibition of human dopamine transporter expressed in HEK293 cells assessed as inhibition of dopamine uptake measured after 30 mins by fluorescence analysis
- ChEMBL_58170 Affinity of the Compound for Dopamine D1 receptor in rat striatal membrane was determined in vitro using Dopamine Antagonist [3H]SCH-23390 as ligand.
- ChEMBL_60023 Relative affinity for dopamine receptor by displacement of [3H]spiroperidol (2.2 nM) from (in vitro) dopamine binding sites in rat caudate nuclei
- ChEMBL_1878790 Inhibition of wild type human dopamine transporter expressed in HEK293 cells assessed as inhibition of [3H]dopamine reuptake preincubated for 5 mins followed by [3H]dopamine addition and measured after 1 min by liquid scintillation analysis
- ChEMBL_1561633 Antagonist activity at human dopamine D2L receptor expressed in CHO cells assessed as inhibition of dopamine-mediated Ca+2 stimulation pretreated for 10 mins followed by addition of dopamine by fluo-4 AM dye-based FLIPR assay
- ChEMBL_1613480 Antagonist activity at human dopamine D2L receptor expressed in CHO cells coexpressing Galpha16 assessed as inhibition of dopamine-induced Ca2+ stimulation pre-incubated for 10 mins followed by dopamine challenge by Fluo-4AM based fluorometric analysis
- ChEBML_131451 Tested in vitro for dopamine(DA) neuronal uptake inhibition
- ChEBML_1554004 Binding affinity to dopamine D1 receptor (unknown origin)
- ChEBML_1554005 Binding affinity to dopamine D4 receptor (unknown origin)
- ChEBML_178952 Inhibition of uptake of dopamine (DA) rat brain striatum
- ChEBML_184435 Inhibition of dopamine (DA) uptake into rat brain synaptosomes
- ChEBML_193333 Inhibition of the uptake of tritiated dopamine (DA) in rat synaptosomes
- ChEBML_58478 Compound was tested for its effect on dopamine saturation analysis
- ChEBML_58513 Ancillary Binding affinity to rat Dopamine receptor D1
- ChEBML_58603 Displacement of [3H]-spiperone from dopamine D2 receptor
- ChEBML_58991 Tested for binding affinity against dopamine receptor D1
- ChEBML_60493 Binding affinity towards Dopamine receptor D1 was determined
- ChEBML_60812 In vitro binding affinity to human Dopamine receptor D4
- ChEBML_60840 Binding affinity for human cloned Dopamine receptor D4
- ChEBML_60841 Binding affinity for human cloned Dopamine receptor D4
- ChEBML_61111 Compound was selective with respect to binding at the Dopamine receptor D2
- ChEBML_61306 Tested for binding affinity against dopamine receptor D2
- ChEBML_61645 Binding affinity for human cloned Dopamine receptor D2L
- ChEBML_61646 Binding affinity for human cloned Dopamine receptor D2L
- ChEBML_61997 In vivo inhibition of DA uptake at dopamine uptake site
- ChEBML_62229 Binding affinity against rat Dopamine receptor D2.
- ChEBML_62450 Binding affinity for human cloned Dopamine receptor D3
- ChEBML_62451 Binding affinity for human cloned Dopamine receptor D3
- ChEBML_62643 Reuptake inhibitory activity against dopamine DA transporter
- ChEBML_62872 Displacement of [3H]spiperone from dopamine receptor D2
- ChEBML_62950 Displacement of [3H]WIN-35428 from Dopamine transporter
- ChEMBL_1279266 Binding affinity to dopamine D2 receptor (unknown origin)
- ChEMBL_1282075 Binding affinity to dopamine D2 receptor (unknown origin)
- ChEMBL_1295491 Agonist activity at dopamine D2 receptor (unknown origin)
- ChEMBL_131451 Tested in vitro for dopamine(DA) neuronal uptake inhibition
- ChEMBL_1352906 Binding affinity to dopamine D3 receptor (unknown origin)
- ChEMBL_1353324 Agonist activity at dopamine D1 receptor (unknown origin)
- ChEMBL_1353325 Antagonist activity at dopamine D1 receptor (unknown origin)
- ChEMBL_1353326 Antagonist activity at dopamine D5 receptor (unknown origin)
- ChEMBL_1367803 Inhibition of DAT-mediated dopamine uptake in rat synaptosomes
- ChEMBL_1367804 Induction of DAT-mediated dopamine release in rat synaptosomes
- ChEMBL_1367904 Inhibition of DAT (unknown origin)-mediated dopamine reuptake
- ChEMBL_1437144 Binding affinity to dopamine D2 receptor (unknown origin)
- ChEMBL_1437145 Binding affinity to dopamine D3 receptor (unknown origin)
- ChEMBL_1440706 Binding affinity to dopamine D2 receptor (unknown origin)
- ChEMBL_1447545 Binding affinity to dopamine D2 receptor (unknown origin)
- ChEMBL_1473029 Binding affinity to dopamine D3 receptor (unknown origin)
- ChEMBL_1506471 Binding affinity to dopamine D3 receptor (unknown origin)
- ChEMBL_1506472 Binding affinity to dopamine D2 receptor (unknown origin)
- ChEMBL_1561663 Binding affinity to dopamine D4 receptor (unknown origin)
- ChEMBL_1586233 Binding affinity to dopamine D3 receptor (unknown origin)
- ChEMBL_1586234 Binding affinity to dopamine D4 receptor (unknown origin)
- ChEMBL_1615911 Binding affinity to dopamine D2 receptor (unknown origin)
- ChEMBL_1682172 Binding affinity to dopamine D4 receptor (unknown origin)
- ChEMBL_177781 Reuptake inhibition of [3H]-labeled dopamine (DA) in rat.
- ChEMBL_177956 Inhibition of [3H]dopamine uptake in rat caudate putamen.
- ChEMBL_1789232 Agonist activity at dopamine D2 receptor (unknown origin)
- ChEMBL_1789233 Agonist activity at dopamine D5 receptor (unknown origin)
- ChEMBL_1803920 Inhibition of [3H]dopamine uptake at DAT (unknown origin)
- ChEMBL_184435 Inhibition of dopamine (DA) uptake into rat brain synaptosomes
- ChEMBL_1912575 Agonist activity at dopamine D4 receptor (unknown origin)
- ChEMBL_1926106 Binding affinity to dopamine D3 receptor (unknown origin)
- ChEMBL_1926107 Binding affinity to dopamine D2 receptor (unknown origin)
- ChEMBL_193333 Inhibition of the uptake of tritiated dopamine (DA) in rat synaptosomes
- ChEMBL_193486 [3H]-Dopamine uptake inhibition in rat caudate putamen
- ChEMBL_1979076 Binding affinity to dopamine D1 receptor (unknown origin)
- ChEMBL_1979077 Binding affinity to dopamine D2 receptor (unknown origin)
- ChEMBL_1979078 Binding affinity to dopamine D3 receptor (unknown origin)
- ChEMBL_1979079 Binding affinity to dopamine D4 receptor (unknown origin)
- ChEMBL_1979080 Binding affinity to dopamine D5 receptor (unknown origin)
- ChEMBL_1988754 Binding affinity to dopamine D5 receptor (unknown origin)
- ChEMBL_1991500 Antagonist activity at dopamine D1 receptor (unknown origin)
- ChEMBL_1991501 Antagonist activity at dopamine D5 receptor (unknown origin)
- ChEMBL_1991502 Agonist activity at dopamine D1 receptor (unknown origin)
- ChEMBL_1991503 Agonist activity at dopamine D5 receptor (unknown origin)
- ChEMBL_2068264 Antagonist activity at dopamine D2 receptor (unknown origin)
- ChEMBL_2112202 Binding affinity to dopamine D2 receptor (unknown origin)
- ChEMBL_2112203 Binding affinity to dopamine D3 receptor (unknown origin)
- ChEMBL_302285 Binding affinity against human Dopamine receptor D2
- ChEMBL_302583 Binding affinity for human recombinant dopamine D2 receptor
- ChEMBL_302584 Binding affinity for human recombinant dopamine receptor D1
- ChEMBL_302585 Binding affinity for human recombinant dopamine receptor D3
- ChEMBL_302586 Binding affinity for human recombinant dopamine receptor D5
- ChEMBL_302602 Binding affinity for human recombinant dopamine receptor D2L
- ChEMBL_302619 Binding affinity for human recombinant dopamine receptor D4.2
- ChEMBL_302620 Binding affinity for human recombinant dopamine receptor D4.4
- ChEMBL_302793 Binding affinity for human dopamine receptor D2 long
- ChEMBL_303308 Inhibition of [3H]spiperone binding to Dopamine receptor D2
- ChEMBL_303309 Inhibition of [3H]spiperone binding to Dopamine receptor D4
- ChEMBL_303376 Inhibition of [125I]-iodosulpiride binding to Dopamine receptor D3
- ChEMBL_307366 Ability of compound to inhibit dopamine uptake of receptor was determined
- ChEMBL_311949 Partial agonist intrinsic activity at dopamine D3 receptor
- ChEMBL_326581 Inhibitory activity against dopamine D2(long) receptor
- ChEMBL_331690 Binding affinity to human cloned dopamine D3 receptor
- ChEMBL_331691 Binding affinity to human cloned dopamine D2 receptor
- ChEMBL_332996 Binding affinity to human cloned dopamine D3 receptor
- ChEMBL_332997 Binding affinity to human cloned dopamine D2 receptor
- ChEMBL_337502 Displacement of [3H]spiperone from D2L dopamine receptor
- ChEMBL_346082 Binding affinity to cloned human dopamine D3 receptor
- ChEMBL_346083 Binding affinity to cloned human dopamine D2 receptor
- ChEMBL_357782 Binding affinity to dopamine receptor by radioligand binding assay
- ChEMBL_357807 Binding affinity to dopamine transporter by radioligand binding assay
- ChEMBL_410547 Binding affinity to human cloned dopamine D1 receptor
- ChEMBL_410548 Binding affinity to human cloned dopamine D2 receptor
- ChEMBL_410549 Binding affinity to human cloned dopamine D3 receptor
- ChEMBL_410550 Binding affinity to human cloned dopamine D4 receptor
- ChEMBL_410554 Binding affinity to human cloned dopamine D5 receptor
- ChEMBL_450225 Binding affinity to human cloned dopamine D2 receptor
- ChEMBL_454685 Displacement of [3H]spiperone from dopamine D2 receptor
- ChEMBL_460878 Blockade of N-arachidonoyl-dopamine-induced activation of TRPV1
- ChEMBL_466543 Displacement of [3H]spiperone from dopamine D2 receptor
- ChEMBL_466544 Displacement of [3H]spiperone from dopamine D3 receptor
- ChEMBL_466546 Displacement of [3H]SCH23390 from dopamine D5 receptor
- ChEMBL_468370 Binding affinity to human dopamine D2 long receptor
- ChEMBL_472677 Inhibition of [3H]dopamine uptake in DAT in rat striatum
- ChEMBL_485923 Displacement of [3H]SCH23390 from dopamine D1 receptor
- ChEMBL_485924 Displacement of [3H]sulpiride from dopamine D2 receptor
- ChEMBL_490804 Binding affinity to human cloned dopamine D1 receptor
- ChEMBL_490806 Binding affinity to human cloned dopamine D2 receptor
- ChEMBL_490807 Binding affinity to human cloned dopamine D3 receptor
- ChEMBL_490808 Binding affinity to human cloned dopamine D4 receptor
- ChEMBL_537766 Displacement of [3H]spiperone from dopamine D2 receptor
- ChEMBL_538665 Displacement of [3H]SCH23390 from dopamine D1 receptor
- ChEMBL_556593 Displacement of [3H]WIN-35428 from dopamine transporter
- ChEMBL_58478 Compound was tested for its effect on dopamine saturation analysis
- ChEMBL_58672 In vitro binding affinity towards Dopamine receptor D1
- ChEMBL_58981 Inhibition of SCH 23390 binding to Dopamine receptor D1
- ChEMBL_59479 Compound was evaluated for the binding affinity at Dopamine receptor D2
- ChEMBL_59905 Inhibition of [3H]thymidine uptake by Dopamine receptor D2
- ChEMBL_59916 Binding affinity towards human Dopamine receptor D2
- ChEMBL_60038 Compound was tested for its effect on dopamine saturation analysis
- ChEMBL_60063 Binding ability of compound to human Dopamine receptor D2
- ChEMBL_60177 Effect of compound on synaptosomal uptake inhibition of Dopamine (DA)
- ChEMBL_60206 Binding affinity towards human Dopamine receptor D2
- ChEMBL_60207 Binding affinity towards human Dopamine receptor D2
- ChEMBL_60217 Binding affinity towards human D2 dopamine receptor.
- ChEMBL_60222 Displacement of [3H]quinpirole from Dopamine receptor D2
- ChEMBL_60223 Inhibition of [3H]raclopride binding to Dopamine receptor D2
- ChEMBL_60224 Inhibition of [3H]raclopride binding to Dopamine receptor D2
- ChEMBL_60494 Binding affinity towards human Dopamine receptor D1
- ChEMBL_60673 Binding affinity of compound was tested for Dopamine receptor D4
- ChEMBL_60679 Binding affinity to recombinant human dopamine receptor D4
- ChEMBL_60684 Binding affinity towards human dopamine receptor D4
- ChEMBL_60994 Binding affinity towards human Dopamine receptor D4
- ChEMBL_61111 Compound was selective with respect to binding at the Dopamine receptor D2
- ChEMBL_61316 The compound's binding affinity against Dopamine receptor D2
- ChEMBL_61484 Binding affinity of compound was tested for Dopamine receptor D2L
- ChEMBL_61606 Inhibition of spiropiperidone binding at dopamine receptor D2 of rat.
- ChEMBL_61655 Inhibition of [125I]RTI-55 binding to dopamine transporter
- ChEMBL_61759 Displacement of [3H]spiroperidol from D2 dopamine receptor
- ChEMBL_61848 Inhibition of [3H]WIN-35428 binding to Dopamine transporter
- ChEMBL_61851 Inhibition of [3H]WIN-35428l binding to Dopamine transporter
- ChEMBL_61946 Effective concentration for Dopamine receptor D3 was determined in monkeys
- ChEMBL_61972 Binding affinity towards human Dopamine receptor D3
- ChEMBL_62009 In vitro potency for inhibiting [3H]- dopamine uptake was determined
- ChEMBL_62018 Inhibition of [3H]dopamine uptake in rat striatal synaptosomes
- ChEMBL_62165 Inhibition of [3H]GBR-12935 binding to the dopamine transporter.
- ChEMBL_62167 Inhibition of [3H]WIN-35428 binding to the dopamine transporter.
- ChEMBL_62262 Binding affinity towards human Dopamine receptor D3
- ChEMBL_62268 Binding affinity towards human dopamine receptor D3
- ChEMBL_62275 Displacement of [3H]raclopride from Dopamine receptor D3
- ChEMBL_62317 The potency of the [125I]RTI-55 for Dopamine transporter site
- ChEMBL_62402 Binding constant against dopamine receptor D2 (in vitro)
- ChEMBL_62403 Binding constant against dopamine receptor D2 (in vivo)
- ChEMBL_62487 Inhibition of reuptake of [3H]DA at Dopamine transporter (DAT)
- ChEMBL_62567 Binding affinity against rat Dopamine receptor D2.
- ChEMBL_62643 Reuptake inhibitory activity against dopamine DA transporter
- ChEMBL_62647 Binding affinity for dopamine transporters in rat brain tissue.
- ChEMBL_62748 Tested for binding affinity against dopamine receptor D3
- ChEMBL_62753 Binding affinity of compound was tested for Dopamine receptor D3
- ChEMBL_62793 Inhibition of [3H]GBR-12935 binding to the dopamine transporter.
- ChEMBL_62795 Inhibition of [3H]WIN-35428 binding to the dopamine transporter.
- ChEMBL_62796 Inhibition of [3H]WIN-35428 binding to the dopamine transporter
- ChEMBL_62805 Ability to displace [3H]-Mazindol from dopamine receptor
- ChEMBL_62806 Ability to displace [3H]mazindol from dopamine transporter
- ChEMBL_62879 In vitro binding affinity towards Dopamine receptor D2
- ChEMBL_62932 Binding affinity towards human Dopamine receptor D3
- ChEMBL_62950 Displacement of [3H]WIN-35428 from Dopamine transporter
- ChEMBL_62952 Inhibition of [3H]DA uptake evaluated at the dopamine transporter
- ChEMBL_63063 Displacement of [3H]spiperone from dopamine receptor D2
- ChEMBL_63078 Effective concentration against human Dopamine receptor D4
- ChEMBL_658545 Binding affinity to human recombinant dopamine D1 receptor
- ChEMBL_658546 Binding affinity to human recombinant dopamine D2 receptor
- ChEMBL_658547 Binding affinity to human recombinant dopamine D3 receptor
- ChEMBL_766799 Inhibition of dopamine D2 receptor by competition binding assay
- ChEMBL_766800 Inhibition of dopamine D3 receptor by competition binding assay
- ChEMBL_766801 inhibition of dopamine D4 receptor by competition binding assay
- ChEMBL_818823 Binding affinity to human recombinant Dopamine D1 receptor
- ChEMBL_818824 Binding affinity to human recombinant Dopamine D2 receptor
- ChEMBL_818825 Binding affinity to human recombinant Dopamine D3 receptor
- ChEMBL_818826 Binding affinity to human recombinant Dopamine D4 receptor
- ChEMBL_818827 Binding affinity to human recombinant Dopamine D5 receptor
- ChEMBL_827294 Displacement of [3H]SCH23390 from dopamine D1 receptor
- ChEMBL_875982 Inhibition of radioligand binding to human dopamine D1 receptor
- ChEMBL_932187 Binding affinity to dopamine D2 receptor (unknown origin)
- ChEMBL_932188 Binding affinity to dopamine D3 receptor (unknown origin)
- ChEMBL_932189 Binding affinity to dopamine D1 receptor (unknown origin)
- ChEMBL_934615 Inhibition of DAT (unknown origin) assessed as dopamine reuptake
- ChEMBL_963021 Binding affinity to dopamine D2 receptor (unknown origin)
- ChEMBL_977143 Binding affinity to dopamine 2 receptor (unknown origin)
- ChEMBL_1437794 Antagonist activity at human dopamine D3 receptor expressed in CHO-K1 cells assessed as reduction in dopamine-induced response by [35S]GTPgammaS binding assay
- ChEMBL_1450571 Antagonist activity against human D3R expressed in CHO cells assessed as inhibition of dopamine-induced [35S]GTPgammaS binding by dopamine potency shift assay
- ChEMBL_1450572 Antagonist activity against human D2LR expressed in CHO cells assessed as inhibition of dopamine-induced [35S]GTPgammaS binding by dopamine potency shift assay
- ChEMBL_63075 Agonist activation of human dopamine receptor stimulating mitogenesis in Dopamine receptor D4-transfected CHO pro-5 cells using [3H]thymidine as radioligand
- ChEMBL_2024048 Positive allosteric modulator activity at human dopamine D1 receptor expressed in HEK293 cells assessed as potentiation of dopamine-induced cAMP accumulation by measuring dopamine EC50 at 50 uM measured after 30 mins by HitHunter assay (Rvb = 214 nM)
- ChEMBL_2024044 Positive allosteric modulator activity at human dopamine D5 receptor expressed in CHO-K1 cells assessed as potentiation of dopamine-induced beta-arrestin2 recruitment by measuring dopamine EC50 at 50 uM incubated for 90 mins by PathHunter assay (Rvb = 81.7 nM)
- ChEMBL_2024046 Positive allosteric modulator activity at human dopamine D1 receptor expressed in CHO-K1 cells assessed as potentiation of dopamine-induced beta-arrestin2 recruitment by measuring dopamine EC50 at 50 uM incubated for 90 mins by PathHunter assay (Rvb = 1.4 uM)
- ChEMBL_1290765 Antagonist activity at dopamine D2 receptor (unknown origin) expressed in HEK cells co-expressing Gqi5 assessed as inhibition of dopamine-induced effect by FLIPR assay
- ChEMBL_1698014 Antagonist activity at human SP/Myc epitope-tagged dopamine D4 receptor expressed in HEK293T cells assessed as inhibition of dopamine-induced RLuc8-fused Galphai1 activation preincubated for 15 mins followed by dopamine induction measured after 2 mins by BRET assay
- ChEBML_58311 Compound was tested for inhibitory activity against Dopamine D1 receptor
- ChEBML_58516 Binding affinity against Dopamine receptor D1 in rat radioligand
- ChEBML_59142 Compound was evaluated for the ability to bind to dopamine beta-hydroxylase of bovine
- ChEBML_60189 Formation of cAMP on Dopamine receptor D1 in vitro in carp retina
- ChEBML_60201 Binding affinity towards cloned human Dopamine receptor D2
- ChEBML_61120 Binding affinity for Dopamine receptor D2 by displacement of [3H]-spiperone
- ChEBML_61513 Inhibitory activity against human dopamine transporter at 10 uM
- ChEBML_62005 In vitro inhibition of [3H]dopamine uptake in rat brain synaptosomes
- ChEBML_62094 Ancillary Binding affinity towards rat Dopamine receptor D2
- ChEBML_62149 Inhibitory activity against dopamine transporter in rat striatal membranes
- ChEBML_62342 Displacement of [3H]WIN-35428 from dopamine transporter (DAT)
- ChEBML_62479 Binding affinity to dopamine transporter (DAT) in rat forebrain tissue
- ChEBML_62632 Inhibition of [3H]DA uptake at Dopamine transporter in rat cortex.
- ChEMBL_1274783 Binding affinity to human dopamine D2 receptor by PDSP assay
- ChEMBL_1498085 Inhibition of dopamine transporter (unknown origin) by cell-based assay
- ChEMBL_166352 Inhibition of high affinity dopamine uptake at concentration of 1 uM
- ChEMBL_1724719 Displacement of [3H]-spiperone from rat caudate dopamine receptor
- ChEMBL_1724720 Displacement of [3H]apomorphine from rat caudate dopamine receptor
- ChEMBL_201668 Ratio of IC50 value against Serotonin transporter to that of dopamine transporter
- ChEMBL_202133 Ratio of Ki value towards Serotonin transporter to that of dopamine transporter
- ChEMBL_216232 Functional cocaine antagonism was evaluated by inhibition of [3H]dopamine reuptake
- ChEMBL_302722 Inhibition of [3H]WIN-35428 binding to rat dopamine transporter
- ChEMBL_302723 Inhibition of [3H]WIN-35428 binding to rat dopamine transporter
- ChEMBL_303035 Inhibition of [3H]spiperone binding to rat dopamine D2 receptor
- ChEMBL_303119 Inhibition of rat brain dopamine transporter as accumulation of [3H]DA
- ChEMBL_303146 Inhibition of [3H]-spiperone binding to human Dopamine receptor D2
- ChEMBL_303165 Inhibition of [18F]PET binding to dopamine transporter of human brain
- ChEMBL_303244 Inhibition of [125I]iodosulpiride binding to human Dopamine receptor D3
- ChEMBL_303257 Inhibition of [3H]raclopride binding to Dopamine receptor D2A in rat
- ChEMBL_303446 Binding affinity for dopamine transporter expressed in LCK PK1 cells
- ChEMBL_307370 Binding affinity towards human dopamine receptor D4 was determined
- ChEMBL_31571 Inhibitory concentration against Dopamine sensitive adenylate cyclase in rats
- ChEMBL_31583 Inhibitory activity against Dopamine sensitive adenylate cyclase in rats
- ChEMBL_337501 Displacement of [3H]SCH 23390 from D1 dopamine receptor
- ChEMBL_337503 Binding affinity to D3 dopamine receptor by radioligand binding assay
- ChEMBL_337504 Binding affinity to D5 dopamine receptor by radioligand binding assay
- ChEMBL_337505 Binding affinity to D4 dopamine receptor by radioligand binding assay
- ChEMBL_346852 Binding affinity to D2 dopamine receptor by radioligand binding assay
- ChEMBL_346853 Binding affinity to D5 dopamine receptor by radioligand binding assay
- ChEMBL_447582 Displacement of [3H]nemonapride from rat dopamine D2 receptor
- ChEMBL_456713 Displacement of [3H]spiperone human cloned dopamine D2 receptor
- ChEMBL_461138 Displacement of [3H]raclopride from rat dopamine D2 receptor
- ChEMBL_465004 Antagonist activity at dopamine D2 receptor by GTPgammaS binding assay
- ChEMBL_468366 Binding affinity to pig cortical membrane dopamine D1 receptor
- ChEMBL_469572 Inhibition of dopamine uptake at VMAT in bovine chromaffin granule ghosts
- ChEMBL_486190 Displacement of [3H]WIN-from cocaine site of dopamine transporter
- ChEMBL_491607 Inhibition of dopamine uptake at human DAT in human HEK293 cells
- ChEMBL_491870 Inhibition of dopamine uptake at cloned DAT in rat brain synaptosome
- ChEMBL_510093 Inhibition of dopamine uptake at human DAT expressed in HEK293 cells
- ChEMBL_523087 Inhibition of dopamine uptake at human DAT expressed in HEK293 cells
- ChEMBL_538666 Displacement of [125I]IABN from human dopamine D4 receptor
- ChEMBL_539628 Displacement of [3H]N-methylspiperone from dopamine D4 receptor
- ChEMBL_556326 Displacement of radioligand from human cloned dopamine D2 receptor
- ChEMBL_558435 Inhibition of dopamine uptake at human DAT transfected in HEK cells
- ChEMBL_563770 Displacement of [3H]spiperone from human dopamine D3 receptor
- ChEMBL_578982 Displacement of [3H]SCH23390 from bovine dopamine D1 receptor
- ChEMBL_58169 Affinity for displacement of [3H]clonidine labeled Dopamine receptor D1
- ChEMBL_58195 Inhibitory activity against Dopamine receptor D2 from mice
- ChEMBL_58682 Binding affinity towards Dopamine receptor D2 in rat was evaluated
- ChEMBL_58770 Binding affinity to the dopamine receptor D2L in rat brain membranes
- ChEMBL_589389 Inhibition of dopamine uptake at human DAT expressed in HEK293 cells
- ChEMBL_58967 Binding affinity against Dopamine receptor D1 in rat radioligand
- ChEMBL_59268 Compound was evaluated for the inhibition of Dopamine beta hydroxylase at pH 4.5
- ChEMBL_59269 Compound was evaluated for the inhibition of Dopamine beta hydroxylase at pH 6.6
- ChEMBL_59771 Binding affinity of [3H]-NPA to striatal Dopamine receptor D2
- ChEMBL_59780 Binding affinity of [3H]NPA to striatal Dopamine receptor D2
- ChEMBL_60018 Inhibitory activity against dopamine receptor in rat striatal membranes
- ChEMBL_60060 Affinity was evaluated as inhibition constant for dopamine D-2 receptor
- ChEMBL_60189 Formation of cAMP on Dopamine receptor D1 in vitro in carp retina
- ChEMBL_60191 Binding affinity towards dopamine receptor D1 in calf striatum
- ChEMBL_60398 Displacement of [3H]spiperone from human Dopamine receptor D2
- ChEMBL_604286 Displacement of [3H]SCH233930 from human dopamine D1 receptor
- ChEMBL_604290 Displacement of [3H]SCH233930 from human dopamine D5 receptor
- ChEMBL_60500 Binding affinity towards dopamine receptor D1 (human clone)
- ChEMBL_60677 Binding affinity towards cloned human Dopamine receptor D4
- ChEMBL_60846 Displacement of [3H]spiperone from human Dopamine receptor D4
- ChEMBL_61001 Effective dose was measured by the stimulation of mitogenesis at Dopamine receptor D4.2
- ChEMBL_61110 In vitro receptor binding affinity against Dopamine receptor D2
- ChEMBL_61337 Binding affinity towards Dopamine receptor D5 (rat clone)
- ChEMBL_61348 Affinity was evaluated as inhibition constant for dopamine D-4 receptor
- ChEMBL_61353 Displacement of [3H]WIN-35428 from monkey dopamine transporter
- ChEMBL_61453 Displacement of [3H]raclopride from human Dopamine receptor D2A
- ChEMBL_61673 Inhibition of reuptake of [3H]DA (20 nM) by dopamine transporter
- ChEMBL_61838 Inhibition of [3H]cocaine binding to rat forebrain dopamine receptor
- ChEMBL_61849 Inhibition of [3H]dopamine uptake in rat caudate putamen tissue.
- ChEMBL_62005 In vitro inhibition of [3H]dopamine uptake in rat brain synaptosomes
- ChEMBL_62013 Inhibition of [3H]WIN-35428 binding at dopamine transporter was determined
- ChEMBL_62014 Inhibition of [3H]WIN-35428 binding at dopamine transporter was determined
- ChEMBL_62149 Inhibitory activity against dopamine transporter in rat striatal membranes
- ChEMBL_62162 Inhibition of [125I]RTI-55 cocaine binding to the dopamine transporter.
- ChEMBL_62166 Inhibition of [3H]WIN-35065-2 binding to the dopamine transporter.
- ChEMBL_62168 Potency for the inhibition of [3H]WIN-35428 binding to the dopamine transporter
- ChEMBL_62250 Binding affinity towards Dopamine receptor D2 in rat was evaluated
- ChEMBL_62327 Ability to inhibit [3H]dopamine uptake into rat striatal synaptosomes
- ChEMBL_62468 Binding affinity for dopamine transporter was determined in rat striatal membrane
- ChEMBL_62469 Binding affinity for dopamine transporter was determined in rat striatal membrane.
- ChEMBL_62632 Inhibition of [3H]DA uptake at Dopamine transporter in rat cortex.
- ChEMBL_62637 Inhibition of [3H]DA uptake by rat striatal dopamine transporter
- ChEMBL_62791 Inhibition of [125I]RTI-55 cocaine binding to the dopamine transporter.
- ChEMBL_62794 Inhibition of [3H]WIN-35065-2 binding to the dopamine transporter.
- ChEMBL_62960 In vitro inhibition of [3H]dopamine uptake in rat brain synaptosomes
- ChEMBL_63038 Affinity against the dopamine receptor D2 using [3H]spiperinone.
- ChEMBL_652494 Antagonist activity at dopamine D3 receptor by GTPgammaS binding assay
- ChEMBL_652495 Antagonist activity at dopamine D2 receptor by GTPgammaS binding assay
- ChEMBL_659509 Binding affinity to human dopamine transporter by radioligand displacement assay
- ChEMBL_746271 Inhibition of DAT in rat striatum assessed as [3H]dopamine accumulation
- ChEMBL_761940 Displacement of [3H]SCH23390 from human dopamine D1 receptor
- ChEMBL_836778 TP_TRANSPORTER: inhibition of Dopamine uptake in OCT2-expressing HEK293 cells
- ChEMBL_932175 Binding affinity to Homo sapiens (human) dopamine D4.4 receptor
- ChEMBL_932176 Binding affinity to Homo sapiens (human) dopamine D3 receptor
- ChEMBL_932177 Binding affinity to Homo sapiens (human) dopamine D2S receptor
- ChEMBL_985425 Inhibition of dopamine D2 receptor (unknown origin) by PDSP assay