Query String: PITAVASTATIN
- ChEMBL_2016319 Inhibition of human ABCC1 expressed in MDCK2-LE cells in presence of pitavastatin
- ChEMBL_1487740 Inhibition of OATP1B1 (unknown origin) expressed in HEK293 cells using pitavastatin substrate
- ChEMBL_1707614 Inhibition of BCRP (unknown origin) transfected in MDCK cells assessed as decrease in pitavastatin transport
- ChEMBL_1487744 Inhibition of OATP1B1 (unknown origin) expressed in HEK293 cells assessed as protein-mediated pitavastatin uptake
- ChEMBL_2151352 Inhibition of OATP1B1 (unknown origin) expressed in HEK293 cells assessed as reduction in OATP 1B1-mediated [3H]-pitavastatin uptake preincubated for 30 mins followed by [3H]-pitavastatin addition and measured after 2 mins by liquid scintillation analysis