RS-43285-003 BDBM50173335 Ranexa CHEBI:87690 CVT-303 Ranolazine
- Koltun, DO; Parkhill, EQ; Elzein, E; Kobayashi, T; Jiang, RH; Li, X; Perry, TD; Avila, B; Wang, WQ; Hirakawa, R; Smith-Maxwell, C; Wu, L; Dhalla, AK; Rajamani, S; Mollova, N; Stafford, B; Tang, J; Belardinelli, L; Zablocki, JA Discovery of triazolopyridinone GS-462808, a late sodium current inhibitor (Late INai) of the cardiac Nav1.5 channel with improved efficacy and potency relative to ranolazine. Bioorg Med Chem Lett 26: 3207-11 (2016)
- Koltun, DO; Parkhill, EQ; Elzein, E; Kobayashi, T; Notte, GT; Kalla, R; Jiang, RH; Li, X; Perry, TD; Avila, B; Wang, WQ; Smith-Maxwell, C; Dhalla, AK; Rajamani, S; Stafford, B; Tang, J; Mollova, N; Belardinelli, L; Zablocki, JA Discovery of triazolopyridine GS-458967, a late sodium current inhibitor (Late INai) of the cardiac NaV 1.5 channel with improved efficacy and potency relative to ranolazine. Bioorg Med Chem Lett 26: 3202-6 (2016)