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Found 1 of ec50 for monomerid = 14971
TargetSerine/threonine-protein kinase B-raf [V600E](Homo sapiens (Human))
Amgen

LigandPNGBDBM14971(4-Methyl-3-(3-(pyrimidin-4-yl)pyridin-2-ylamino)-N...)
Affinity DataIC50:  0.460nM EC50:  15nMpH: 7.0 T: 2°CAssay Description:The in vitro kinase activities of wild type or mutants were determined by measuring phosphorylation of biotinylated-MEK protein using Perkin-Elmer s ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed