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Compile Data Set for Download or QSAR

Found 1 hit of ic50 for monomerid = 50101681   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Histone chaperone ASF1A


(Homo sapiens (Human))
BDBM50101681
PNG
(CHEMBL3394917)
Show SMILES O=C(N\N=C\c1ccncc1)c1ccc(NC(=O)c2ccccc2)cc1
Show InChI InChI=1S/C20H16N4O2/c25-19(16-4-2-1-3-5-16)23-18-8-6-17(7-9-18)20(26)24-22-14-15-10-12-21-13-11-15/h1-14H,(H,23,25)(H,24,26)/b22-14+
PDB

UniProtKB/SwissProt

GoogleScholar
PC cid
PC sid
UniChem

Patents


Similars

Article
PubMed
n/an/a>1.00E+5n/an/an/an/an/an/a



Colorado State University

Curated by ChEMBL


Assay Description
Inhibition of His-tagged human Asf1a binding with H3/H4 assessed as fluorescence intensity after 30 mins by ALPHA assay


Bioorg Med Chem Lett 25: 963-8 (2015)


Article DOI: 10.1016/j.bmcl.2014.11.067
BindingDB Entry DOI: 10.7270/Q2VM4F0G
More data for this
Ligand-Target Pair