Compile Data Set for Download or QSAR
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Found 11 of ic50 for monomerid = 50331682
TargetSialidase-3(Homo sapiens (Human))
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50331682((2R,3R,4S)-3-(2-azidoacetamido)-4-hydroxy-2-((1R,2...)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibition of N-terminal MBP-fused human NEU3 expressed in Escherichia coli using 4MU-NANA as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSialidase-4(Homo sapiens (Human))
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50331682((2R,3R,4S)-3-(2-azidoacetamido)-4-hydroxy-2-((1R,2...)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibition of human NEU4 using 4-MU-NANA as substrate preincubated for 15 mins before substrate addition measured after 30 mins by fluorescence plate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSialidase-3(Homo sapiens (Human))
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50331682((2R,3R,4S)-3-(2-azidoacetamido)-4-hydroxy-2-((1R,2...)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of human NEU3 using 4-MU-NANA as substrate preincubated for 15 mins before substrate addition measured after 30 mins by fluorescence plate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSialidase-4(Homo sapiens (Human))
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50331682((2R,3R,4S)-3-(2-azidoacetamido)-4-hydroxy-2-((1R,2...)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of MBP-fused human NEU4 expressed in Escherichia coli using 4MU-NANA as substrate preincubated for 15 mins followed by substrate addition ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSialidase-2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50331682((2R,3R,4S)-3-(2-azidoacetamido)-4-hydroxy-2-((1R,2...)
Affinity DataIC50:  8.30E+3nMAssay Description:Inhibition of NEU2 (unknown origin) using Neu5Acalpha2-3GalbetapNP as substrate incubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSialidase-2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50331682((2R,3R,4S)-3-(2-azidoacetamido)-4-hydroxy-2-((1R,2...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of NEU2 (unknown origin) using Neu5Acalpha2-6GalbetapNP as substrate incubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSialidase-3(Homo sapiens (Human))
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50331682((2R,3R,4S)-3-(2-azidoacetamido)-4-hydroxy-2-((1R,2...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of human neuraminidase 3 assessed as inhibition of 4-methylumbelliferyl-alpha-D-glucopyranoside hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSialidase-2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50331682((2R,3R,4S)-3-(2-azidoacetamido)-4-hydroxy-2-((1R,2...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of N-terminal MBP-fused human NEU2 expressed in Escherichia coli using 4MU-NANA as substrate preincubated for 15 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSialidase-1(Homo sapiens (Human))
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50331682((2R,3R,4S)-3-(2-azidoacetamido)-4-hydroxy-2-((1R,2...)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of human His6-tagged NEU1 expressed in HEK293 cells using 4MU-NANA as substrate preincubated for 15 mins followed by substrate addition an...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSialidase-1(Homo sapiens (Human))
University Of Alberta

Curated by ChEMBL
LigandPNGBDBM50331682((2R,3R,4S)-3-(2-azidoacetamido)-4-hydroxy-2-((1R,2...)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibition of human NEU1 using 4-MU-NANA as substrate preincubated for 15 mins before substrate addition measured after 30 mins by fluorescence plate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSialidase-2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50331682((2R,3R,4S)-3-(2-azidoacetamido)-4-hydroxy-2-((1R,2...)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of human NEU2 using 4-MU-NANA as substrate preincubated for 15 mins before substrate addition measured after 30 mins by fluorescence plate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed