TargetcAMP-dependent protein kinase catalytic subunit alpha(Homo sapiens (Human))
Nagoya University School of Medicine
Nagoya University School of Medicine
Affinity DataKi: 48nM ΔG°: -42.5kJ/moleT: 2°CAssay Description:Protein kinase C, cAMP dependent protein kinase, cGMP dependent protein kinase and myosin light chain kinase activity were measure under conditions d...More data for this Ligand-Target Pair
TargetcAMP-dependent protein kinase catalytic subunit beta(RAT)
Temple University
Curated by PDSP Ki Database
Temple University
Curated by PDSP Ki Database
TargetRho-associated protein kinase 2(Rattus norvegicus (Rat))
Temple University
Curated by PDSP Ki Database
Temple University
Curated by PDSP Ki Database
Affinity DataKi: 480nM ΔG°: -36.7kJ/moleT: 2°CAssay Description:Protein kinase C, cAMP dependent protein kinase, cGMP dependent protein kinase and myosin light chain kinase activity were measure under conditions d...More data for this Ligand-Target Pair
TargetMyosin light chain kinase, smooth muscle(Gallus gallus (chicken))
Institute for Biochemistry
Curated by ChEMBL
Institute for Biochemistry
Curated by ChEMBL
Affinity DataKi: 2.83E+4nMAssay Description:Inhibitory constant against MLCKMore data for this Ligand-Target Pair
Affinity DataKi: 2.83E+4nM ΔG°: -26.4kJ/moleT: 2°CAssay Description:Protein kinase C, cAMP dependent protein kinase, cGMP dependent protein kinase and myosin light chain kinase activity were measure under conditions d...More data for this Ligand-Target Pair
TargetMyosin light chain kinase, smooth muscle(Homo sapiens (Human))
University of Oxford
Curated by ChEMBL
University of Oxford
Curated by ChEMBL
Affinity DataKi: 2.83E+4nMAssay Description:Binding affinity at MLCKChecked by AuthorMore data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase type II subunit beta(Homo sapiens (Human))
Nagoya University School of Medicine
Nagoya University School of Medicine
Affinity DataKi: 2.97E+4nM ΔG°: -26.3kJ/moleT: 2°CAssay Description:Protein kinase C, cAMP dependent protein kinase, cGMP dependent protein kinase and myosin light chain kinase activity were measure under conditions d...More data for this Ligand-Target Pair
TargetCalcium/calmodulin-dependent protein kinase kinase 2(Homo sapiens (Human))
University of Oxford
Curated by ChEMBL
University of Oxford
Curated by ChEMBL
Affinity DataKi: 2.97E+4nMAssay Description:Inhibition of CaM-KKbetaChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 3.17E+4nM ΔG°: -26.1kJ/moleT: 2°CAssay Description:Protein kinase C, cAMP dependent protein kinase, cGMP dependent protein kinase and myosin light chain kinase activity were measure under conditions d...More data for this Ligand-Target Pair
Affinity DataKi: 3.83E+4nMAssay Description:Inhibition of casein kinase 1Checked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 3.83E+4nM ΔG°: -25.6kJ/moleT: 2°CAssay Description:Protein kinase C, cAMP dependent protein kinase, cGMP dependent protein kinase and myosin light chain kinase activity were measure under conditions d...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha (Homo sapiens (Human))
Institute for Biochemistry
Curated by ChEMBL
Institute for Biochemistry
Curated by ChEMBL
Affinity DataKi: 1.37E+5nMAssay Description:Inhibitory constant against bovine CK2More data for this Ligand-Target Pair
Affinity DataKi: 1.37E+5nM ΔG°: -22.4kJ/moleT: 2°CAssay Description:Protein kinase C, cAMP dependent protein kinase, cGMP dependent protein kinase and myosin light chain kinase activity were measure under conditions d...More data for this Ligand-Target Pair
