TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
TargetSerotonin 2 (5-HT2) receptor(RAT)
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
R. W. Johnson Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:Binding affinity determined in radioreceptor binding assay by using [3H]ketanserin radioligand against 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of North Carolina
Curated by PDSP Ki Database
University Of North Carolina
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of North Carolina
Curated by PDSP Ki Database
University Of North Carolina
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of North Carolina
Curated by PDSP Ki Database
University Of North Carolina
Curated by PDSP Ki Database
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]-N-methylspiperone from human dopamine D2long receptor expressed in HEK293 cells after 30 mins by scintillation countingMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of North Carolina
Curated by PDSP Ki Database
University Of North Carolina
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of North Carolina
Curated by PDSP Ki Database
University Of North Carolina
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of North Carolina
Curated by PDSP Ki Database
University Of North Carolina
Curated by PDSP Ki Database
Affinity DataKi: 1.20nMAssay Description:Compound was tested for inhibitory activity against the binding of [3H]-spiperone to Dopamine receptor D2 in rat striatal membranesMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of North Carolina
Curated by PDSP Ki Database
University Of North Carolina
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of North Carolina
Curated by PDSP Ki Database
University Of North Carolina
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of North Carolina
Curated by PDSP Ki Database
University Of North Carolina
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of North Carolina
Curated by PDSP Ki Database
University Of North Carolina
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of North Carolina
Curated by PDSP Ki Database
University Of North Carolina
Curated by PDSP Ki Database
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Solvay Pharma
Curated by ChEMBL
Solvay Pharma
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha1 receptor in rat cerebral cortexMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of North Carolina
Curated by PDSP Ki Database
University Of North Carolina
Curated by PDSP Ki Database
Affinity DataKi: 1.80nMAssay Description:Compound was evaluated for binding affinity towards Dopamine receptor D2 in striatal membranes, using [3H]- spiperone as radioligand in the absence o...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Toronto
Curated by PDSP Ki Database
University Of Toronto
Curated by PDSP Ki Database
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]-raclopride from recombinant human D2 receptor expressed in HEK293 cells measured after 1 hr by microbeta scintillation counting ...More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]-raclopride from human D2 receptor expressed in HEK cells incubated for 1 hr by Cheng-Prusoff analysis based microbeta scintillat...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of North Carolina
Curated by PDSP Ki Database
University Of North Carolina
Curated by PDSP Ki Database
Affinity DataKi: 2nMAssay Description:In vitro binding affinity against Dopamine D2 receptor in rat striatal tissue.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of North Carolina
Curated by PDSP Ki Database
University Of North Carolina
Curated by PDSP Ki Database
Affinity DataKi: 2nMAssay Description:Binding affinity against dopamine D2 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of North Carolina
Curated by PDSP Ki Database
University Of North Carolina
Curated by PDSP Ki Database
Affinity DataKi: 2.20nMAssay Description:Compound was evaluated for binding affinity towards dopamine receptor D2 in striatal membranes, using [3H]- spiperone as radioligand in the presence ...More data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Displacement of [3H]-methylspiperone from human D2 receptor transfected in CHO-K1 cells measured after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of North Carolina
Curated by PDSP Ki Database
University Of North Carolina
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of North Carolina
Curated by PDSP Ki Database
University Of North Carolina
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of North Carolina
Curated by PDSP Ki Database
University Of North Carolina
Curated by PDSP Ki Database