TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Reading
Curated by PDSP Ki Database
University Of Reading
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Reading
Curated by PDSP Ki Database
University Of Reading
Curated by PDSP Ki Database
Affinity DataKi: 1.10nMAssay Description:Inhibition constant against dopamine receptor D2 in ratMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Reading
Curated by PDSP Ki Database
University Of Reading
Curated by PDSP Ki Database
Affinity DataKi: 1.10nMAssay Description:Competitive binding assay against Dopamine receptor D2 in rat striatal membranes and [125I]-IBF radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]spiperone from human D2 receptor transfected in HEK cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Reading
Curated by PDSP Ki Database
University Of Reading
Curated by PDSP Ki Database
Affinity DataKi: 1.30nMAssay Description:Inhibition of [3H]raclopride binding to rat striatal dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Reading
Curated by PDSP Ki Database
University Of Reading
Curated by PDSP Ki Database
Affinity DataKi: 1.30nMAssay Description:Inhibition of [3H]spiperone binding to rat striatal membrane Dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Reading
Curated by PDSP Ki Database
University Of Reading
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Reading
Curated by PDSP Ki Database
University Of Reading
Curated by PDSP Ki Database
Affinity DataKi: 1.80nMAssay Description:In vitro binding affinity against dopamine receptor D2 in rat striata; value ranges from 1.8-3.0 nMMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Reading
Curated by PDSP Ki Database
University Of Reading
Curated by PDSP Ki Database
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Reading
Curated by PDSP Ki Database
University Of Reading
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Reading
Curated by PDSP Ki Database
University Of Reading
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Reading
Curated by PDSP Ki Database
University Of Reading
Curated by PDSP Ki Database
Affinity DataKi: 2.60nMAssay Description:Displacement of [3H]raclopride from dopamine D2 receptor in Sprague-Dawley rat striatal membranes after 30 minsMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Reading
Curated by PDSP Ki Database
University Of Reading
Curated by PDSP Ki Database
Affinity DataKi: 3.70nMAssay Description:Compound was measured for its ability to compete with [3H]spiperone binding to the human Dopamine receptor D3 transfected in CHO cellsMore data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 5.10nMAssay Description:In vitro inhibition of [3H]-Spiperone binding to Dopamine receptor D2 in Macaca nemestrina striatal membranes (using L-tartrate salt of authentic rac...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Reading
Curated by PDSP Ki Database
University Of Reading
Curated by PDSP Ki Database
Affinity DataKi: 8.30nMAssay Description:Displacement of [3H]- spiperone from dopamine receptor D2 of striatal membranes without sodium chlorideMore data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Homo sapiens (Human))
Washington University
Curated by ChEMBL
Washington University
Curated by ChEMBL
Affinity DataKi: 8.70nMAssay Description:In vitro inhibition of [3H]spiperone binding to Dopamine receptor D2 in Macaca nemestrina striatal membranesMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Reading
Curated by PDSP Ki Database
University Of Reading
Curated by PDSP Ki Database
Affinity DataKi: 9.30nMAssay Description:Tested for binding affinity against dopamine receptor D3 expressed in Sf9 cells.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Reading
Curated by PDSP Ki Database
University Of Reading
Curated by PDSP Ki Database
Affinity DataKi: 9.5nMAssay Description:Compound was evaluated for binding affinity towards DA D-2 receptor using radioligand [3H]SPIMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity to dopamine D2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity to dopamine D3 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor expressed in HEK293 cells after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D3 receptor expressed in HEK293 cells after 1 hr by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Displacement of [3H]spiperone from dopamine D3 receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Displacement of [3H]spiperone from dopamine D2long receptor in CHO cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Reading
Curated by PDSP Ki Database
University Of Reading
Curated by PDSP Ki Database
Affinity DataKi: 31nMAssay Description:Displacement of [3H]spiperone from dopamine D2short receptor in CHO cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Reading
Curated by PDSP Ki Database
University Of Reading
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Reading
Curated by PDSP Ki Database
University Of Reading
Curated by PDSP Ki Database
Affinity DataKi: 33nMAssay Description:Displacement of [3H]- spiperone from dopamine receptor D2 of striatal membranes without sodium chlorideMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Reading
Curated by PDSP Ki Database
University Of Reading
Curated by PDSP Ki Database
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Reading
Curated by PDSP Ki Database
University Of Reading
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University Of Toronto
Curated by PDSP Ki Database
University Of Toronto
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Case Western Reserve University
Curated by PDSP Ki Database
Case Western Reserve University
Curated by PDSP Ki Database