Found 27 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 1A' and Ligand = 'BDBM50005127' Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of Alberta
Curated by PDSP Ki Database
University Of Alberta
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of Alberta
Curated by PDSP Ki Database
University Of Alberta
Curated by PDSP Ki Database
Affinity DataKi: 0.240nMAssay Description:Displacement of [3H]8-OH-DAPT from human recombinant 5-HT1A receptor expressed in COS7 cells measured after 60 to 90 mins by radioligand completion a...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of Alberta
Curated by PDSP Ki Database
University Of Alberta
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Cracow University Of Technology
Curated by ChEMBL
Cracow University Of Technology
Curated by ChEMBL
Affinity DataKi: 3.40nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in rat brain hippocampus by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Cracow University Of Technology
Curated by ChEMBL
Cracow University Of Technology
Curated by ChEMBL
Affinity DataKi: 3.40nMAssay Description:Inhibitory affinity constant against 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Cracow University Of Technology
Curated by ChEMBL
Cracow University Of Technology
Curated by ChEMBL
Affinity DataKi: 3.40nMAssay Description:In vitro ability to displace [3H]-8-hydroxy-2-(di-n-propylamino) tetralin binding from 5-hydroxytryptamine 1A receptor site in rat brain hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of Alberta
Curated by PDSP Ki Database
University Of Alberta
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of Alberta
Curated by PDSP Ki Database
University Of Alberta
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Cracow University Of Technology
Curated by ChEMBL
Cracow University Of Technology
Curated by ChEMBL
Affinity DataKi: 5.5nMAssay Description:Displacement of [3H]8-OH-DPAT from 5HT1A receptor in CRL:CD(SD)BR-COBS rat hippocampusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Cracow University Of Technology
Curated by ChEMBL
Cracow University Of Technology
Curated by ChEMBL
Affinity DataKi: 5.5nMAssay Description:Inhibition of [3H]8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor of rat frontal cortex membranesMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Cracow University Of Technology
Curated by ChEMBL
Cracow University Of Technology
Curated by ChEMBL
Affinity DataKi: 5.5nMAssay Description:Displacement of radioligand [3H]-2-(di-N-propylamino)-8-hydroxytetralin from 5-hydroxytryptamine 1A receptor in rat frontal cortex homogenateMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of Alberta
Curated by PDSP Ki Database
University Of Alberta
Curated by PDSP Ki Database
Affinity DataKi: 6nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5HT1A receptor in HEK293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of Alberta
Curated by PDSP Ki Database
University Of Alberta
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of Alberta
Curated by PDSP Ki Database
University Of Alberta
Curated by PDSP Ki Database
Affinity DataKi: 7.90nMAssay Description:Displacement of [3H]-5-OH-DPAT from human 5-HT1AR expressed in human HEK293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Cracow University Of Technology
Curated by ChEMBL
Cracow University Of Technology
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:In vitro inhibition of [3H]spiperone binding to 5-hydroxytryptamine 1A receptor from rat hippocampal tissue.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of Alberta
Curated by PDSP Ki Database
University Of Alberta
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Cracow University Of Technology
Curated by ChEMBL
Cracow University Of Technology
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:In vitro ability to inhibit [3H]8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor of rat hippocampusMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Compound was tested for binding affinity to 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT as a radioligandMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of Alberta
Curated by PDSP Ki Database
University Of Alberta
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of Alberta
Curated by PDSP Ki Database
University Of Alberta
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of Alberta
Curated by PDSP Ki Database
University Of Alberta
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of Alberta
Curated by PDSP Ki Database
University Of Alberta
Curated by PDSP Ki Database
Affinity DataKi: 50nMAssay Description:Displacement of [3H]5-CT from human recombinant 5-HT1A receptor expressed in CHO cells measured after 60 to 90 mins by radioligand completion assay r...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of Alberta
Curated by PDSP Ki Database
University Of Alberta
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Cracow University Of Technology
Curated by ChEMBL
Cracow University Of Technology
Curated by ChEMBL
Affinity DataIC50: 8.20nMAssay Description:Inhibition of 8-OH DPAT bindign to rat hydroxytryptamine 1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Cracow University Of Technology
Curated by ChEMBL
Cracow University Of Technology
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A (5-HT1A) receptor in rat hippocampus membranesMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Cracow University Of Technology
Curated by ChEMBL
Cracow University Of Technology
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Binding affinity to 5-hydroxytryptamine 1A receptor in rat hippocampus membranes,3H-8-OH-DPAT and buspirone for nonspecific binding (NSB)More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
University Of Alberta
Curated by PDSP Ki Database
University Of Alberta
Curated by PDSP Ki Database
Affinity DataEC50: 68nMAssay Description:Compound was tested for its potency against human 5-hydroxytryptamine 1A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
