Found 19 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 1B' and Ligand = 'BDBM21393'
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Veterans Affairs Medical Center
Curated by PDSP Ki Database
Veterans Affairs Medical Center
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Veterans Affairs Medical Center
Curated by PDSP Ki Database
Veterans Affairs Medical Center
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Veterans Affairs Medical Center
Curated by PDSP Ki Database
Veterans Affairs Medical Center
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Veterans Affairs Medical Center
Curated by PDSP Ki Database
Veterans Affairs Medical Center
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Veterans Affairs Medical Center
Curated by PDSP Ki Database
Veterans Affairs Medical Center
Curated by PDSP Ki Database
Affinity DataKi: 559nMAssay Description:The intrinsic activity of the compound was evaluated for its ability to inhibit forskolin-stimulated c-AMP formation mediated by cloned 5-hydroxytryp...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Veterans Affairs Medical Center
Curated by PDSP Ki Database
Veterans Affairs Medical Center
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Veterans Affairs Medical Center
Curated by PDSP Ki Database
Veterans Affairs Medical Center
Curated by PDSP Ki Database
Affinity DataKi: 638nMAssay Description:Binding affinity against 5-hydroxytryptamine 1D receptor beta expressed in CHO-K1 cells, using [3H]-5-HT as the radioligand.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Veterans Affairs Medical Center
Curated by PDSP Ki Database
Veterans Affairs Medical Center
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Veterans Affairs Medical Center
Curated by PDSP Ki Database
Veterans Affairs Medical Center
Curated by PDSP Ki Database
Affinity DataKi: 2.57E+3nMAssay Description:Inhibition of [3H]5-HT binding to 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Veterans Affairs Medical Center
Curated by PDSP Ki Database
Veterans Affairs Medical Center
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Veterans Affairs Medical Center
Curated by PDSP Ki Database
Veterans Affairs Medical Center
Curated by PDSP Ki Database
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in rat striatal membranes using [3H]-5-HT as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Evaluated for binding affinity towards 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.30E+4nMAssay Description:Binding affinity (Ki) to rat cortical membranes at 5-HT1B binding site by using [125 I] ICYP as a radioligand.More data for this Ligand-Target Pair
Affinity DataIC50: 3.80E+3nMAssay Description:Binding affinity against 5-HT1B receptor in rat frontal cortex using [3H]-5-HT in presence of 0.1 uM [3H]-8-OH-DPAT as a radioligandMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Veterans Affairs Medical Center
Curated by PDSP Ki Database
Veterans Affairs Medical Center
Curated by PDSP Ki Database
Affinity DataEC50: 260nMAssay Description:The intrinsic activity of the compound was evaluated for its ability to inhibit forskolin-stimulated c-AMP formation mediated by cloned 5-hydroxytryp...More data for this Ligand-Target Pair