Found 5 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 2A' and Ligand = 'BDBM50017452'
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Vernalis Research
Curated by PDSP Ki Database
Vernalis Research
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Stanford University
Curated by PDSP Ki Database
Stanford University
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Vernalis Research
Curated by PDSP Ki Database
Vernalis Research
Curated by PDSP Ki Database
Affinity DataKi: 2.10E+4nMAssay Description:Displacement of [3H]ketanserin from human 5HT2A receptor expressed in tsA201 cell membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Vernalis Research
Curated by PDSP Ki Database
Vernalis Research
Curated by PDSP Ki Database
Affinity DataEC50: 1.20E+3nMAssay Description:Agonist activity at human 5HT2A receptor expressed in HEK293 cells assessed as accumulation of IP1 incubated for 1 hr at 37 degC followed by 15 mins ...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Vernalis Research
Curated by PDSP Ki Database
Vernalis Research
Curated by PDSP Ki Database
Affinity DataEC50: 420nMAssay Description:Agonist activity at human 5HT2A receptor expressed in HEK293 cells assessed as induction of intracellular calcium release measured for 90 secs by flu...More data for this Ligand-Target Pair