Found 11 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 2C' and Ligand = 'BDBM85098'
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]mesulergine from human 5-HT2C receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]mesulergine from human recombinant 5-HT2C receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Displacement of [3H]mesulergine from human cloned 5-hydroxytryptamine 2C receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Roche Bioscience
Curated by PDSP Ki Database
Roche Bioscience
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Target5-hydroxytryptamine receptor 2C(Mus musculus (Mouse))
National Institutes Of Health
Curated by PDSP Ki Database
National Institutes Of Health
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Displacement of [3H]mesuleregine from human recombinant 5-HT2C receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Jagiellonian University Collegium Medicum
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Displacement of [3H]mesulergine from human recombinant 5HT2C receptor expressed in HEK293 cells measured after 120 mins by scintillation counting met...More data for this Ligand-Target Pair