Affinity DataIC50: 10nMAssay Description:Inhibition of human AChE using p-nitrophenyl acetate as substrate measured for 30 secs by spectrophotometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Displacement of acetylcholine from AChE in Swiss Webster mouse brain after 5 minsMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Missouri St. Louis
Curated by ChEMBL
University Of Missouri St. Louis
Curated by ChEMBL
Affinity DataKd: 1.70E+5nMAssay Description:Binding affinity to Electric eel AChE using acetylthiocholine as substrate measured for 30 secs by Ellman's methodMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Missouri St. Louis
Curated by ChEMBL
University Of Missouri St. Louis
Curated by ChEMBL
Affinity DataKoff: 333s-1Assay Description:Inhibition of electric eel AChE by concentration-dependent inhibition assayMore data for this Ligand-Target Pair
Affinity DataKoff: 567s-1Assay Description:Inhibition of rat brain AChE by time-dependent inhibition assayMore data for this Ligand-Target Pair
Affinity DataKoff: 267s-1Assay Description:Inhibition of rat brain AChE by concentration-dependent inhibition assayMore data for this Ligand-Target Pair