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Found 6 Enz. Inhib. hit(s) with Target = 'Acetylcholinesterase' and Ligand = 'BDBM50240416'
TargetAcetylcholinesterase(Homo sapiens (Human))
University Of Missouri St. Louis

Curated by ChEMBL
LigandPNGBDBM50240416(CHEMBL23838 | O,O-diethyl O-p-nitrophenyl phosphat...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human AChE using p-nitrophenyl acetate as substrate measured for 30 secs by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Mus musculus (mouse))
University Of California

Curated by ChEMBL
LigandPNGBDBM50240416(CHEMBL23838 | O,O-diethyl O-p-nitrophenyl phosphat...)
Affinity DataIC50:  13nMAssay Description:Displacement of acetylcholine from AChE in Swiss Webster mouse brain after 5 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Missouri St. Louis

Curated by ChEMBL
LigandPNGBDBM50240416(CHEMBL23838 | O,O-diethyl O-p-nitrophenyl phosphat...)
Affinity DataKd:  1.70E+5nMAssay Description:Binding affinity to Electric eel AChE using acetylthiocholine as substrate measured for 30 secs by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Missouri St. Louis

Curated by ChEMBL
LigandPNGBDBM50240416(CHEMBL23838 | O,O-diethyl O-p-nitrophenyl phosphat...)
Affinity DataKoff:  333s-1Assay Description:Inhibition of electric eel AChE by concentration-dependent inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50240416(CHEMBL23838 | O,O-diethyl O-p-nitrophenyl phosphat...)
Affinity DataKoff:  567s-1Assay Description:Inhibition of rat brain AChE by time-dependent inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
The University Of Montana

Curated by ChEMBL
LigandPNGBDBM50240416(CHEMBL23838 | O,O-diethyl O-p-nitrophenyl phosphat...)
Affinity DataKoff:  267s-1Assay Description:Inhibition of rat brain AChE by concentration-dependent inhibition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed