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Found 5 Enz. Inhib. hit(s) with Target = 'Acetylcholinesterase' and Ligand = 'BDBM50399977'
TargetAcetylcholinesterase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50399977(CHEMBL2181432)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human AChEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50399977(CHEMBL2181432)
Affinity DataIC50:  8.90E+5nMAssay Description:Inhibition of human acetylcholinesterase by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50399977(CHEMBL2181432)
Affinity DataKd:  2.20E+4nMAssay Description:Reactivation of VX-inhibited human acetylcholinesterase assessed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50399977(CHEMBL2181432)
Affinity DataKd:  8.80E+4nMAssay Description:Reactivation of sarin-inhibited human acetylcholinesterase assessed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50399977(CHEMBL2181432)
Affinity DataKd:  1.80E+4nMAssay Description:Reactivation of tabun-inhibited human acetylcholinesterase assessed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed