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Found 1 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM21239'
TargetAdenosine receptor A1(Homo sapiens (Human))
Universita Di Napoli

LigandPNGBDBM21239(2-mercaptopyrimidine analogue, 5r | N-{6-[(4-chlor...)
Affinity DataKi:  4.48E+3nM ΔG°:  -30.5kJ/molepH: 7.4 T: 2°CAssay Description:The membranes prepared from CHO cells transfected with human adenosine A1 receptors were used in binding assays. Nonspecific binding was determined i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed