Affinity DataKi: 270nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]-CHA or [3H]PIA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 270nMAssay Description:Binding affinity towards adenosine A1 receptor in rat cortical membranes using N6-[3H]cyclohexyladenosine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 270nMAssay Description:Tested for the displacement [3H]-PIA from Adenosine A1 receptor in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 6.90E+3nMAssay Description:Binding affinity against adenosine A1 receptor in guinea pig forebrain membranes using N6-[3H]cyclohexyladenosine as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 270nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair