Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM50078430'
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50078430(CHEMBL3414944)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]-CCPA from human recombinant adenosine A1 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Camerino

Curated by ChEMBL
LigandPNGBDBM50078430(CHEMBL3414944)
Affinity DataEC50:  8.70nMAssay Description:Agonist activity at human recombinant adenosine A1 receptor transfected in CHO cells assessed as inhibition of forskolin-induced adenylyl cyclase act...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed