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Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM50097423'
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50097423(4-Methoxy-N-(3-phenyl-[1,2,4]thiadiazol-5-yl)-benz...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]-DPCPX from Adenosine A1 receptor of rat cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50097423(4-Methoxy-N-(3-phenyl-[1,2,4]thiadiazol-5-yl)-benz...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in rat brain cortical membrane in presence of 100 uM GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50097423(4-Methoxy-N-(3-phenyl-[1,2,4]thiadiazol-5-yl)-benz...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed