Affinity DataKi: 48nMAssay Description:Antagonist activity at human recombinant adenosine A1 receptor by cAMP assayMore data for this Ligand-Target Pair
Affinity DataKi: 48.2nMAssay Description:Antagonistic activity at adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 48.2nMAssay Description:Antagonist activity at human Adenosine receptor A1 assessed as inhibition of cAMP productionMore data for this Ligand-Target Pair
Affinity DataEC50: 48nMAssay Description:Binding affinity to human recombinant adenosine A1 receptor expressed in CHO cells using [3H]CCPA by functional activity assayMore data for this Ligand-Target Pair