Found 23 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a' and Ligand = 'BDBM21221' 
Affinity DataKi: 56nMAssay Description:Binding affinity for adenosine A2a receptor as inhibition of 3[H]-CGS 21680 binding in rat striatumMore data for this Ligand-Target Pair
Affinity DataKi: 401nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 401nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cell membrane after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 401nMAssay Description:The membranes prepared from CHO cells transfected with human adenosine A2A receptors were used in binding assays. Nonspecific binding was determined ...More data for this Ligand-Target Pair
Affinity DataKi: 401nMAssay Description:Displacement of [3H]NECA from human A2A adenosine receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 470nMAssay Description:Binding affinity for adenosine A2A receptor as displacement of [3H]-CGS- 21680 from rat striatal membranes at 10e-4 MMore data for this Ligand-Target Pair
Affinity DataKi: 470nMAssay Description:Tested for the binding affinity of A2a receptor by displacing the [3H]-CGS- 21680 in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 470nMAssay Description:Displacement of radioligand from rat adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 470nMAssay Description:Displacement of [3H]CGS21680 from rat adenosine A2A receptor expressed in CHO cells after 60 mins by gamma counterMore data for this Ligand-Target Pair
Affinity DataKi: 5.36E+3nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cell membranes after 3 hrs by micro beta scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 5.36E+3nMAssay Description:Displacement of [3H]R-PIA form human adenosine A2A receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.36E+3nMAssay Description:Displacement of [3H]CGS-21680 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.36E+3nMAssay Description:Binding affinity towards recombinant human Adenosine A2a receptor was determined using [3H]CGS-21680 (10 nM) as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 5.36E+3nMAssay Description:Displacement of [3H]CGS21680 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.36E+3nMAssay Description:Displacement of [3H]CGS-21680 from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.36E+3nMAssay Description:Displacement of [3H]CGS21680 from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.36E+3nMAssay Description:Displacement of [3H]CGS21680 from human A2A adenosine receptor expressed in HEK293 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 5.37E+3nMAssay Description:Displacement of [3H]CGS21680 from human adenosine A2A receptor expressed in HEK293 cells after 60 mins by liquid scintillation analyzerMore data for this Ligand-Target Pair
Affinity DataKi: 5.40E+3nMAssay Description:Displacement of radioligand from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.40E+3nMAssay Description:Inhibition of [3H]-CGS- 21680 binding to human Adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.40E+3nMAssay Description:Displacement of [3 H]2-[p-(2-carboxyethyl)phenyl-ethylamino]-5'-N-ethylcarboxamidoadenosine from recombinant human adenosine receptor A2A expressed i...More data for this Ligand-Target Pair
Affinity DataKi: 5.40E+3nMAssay Description:Displacement of [3H]CGS21680 from human recombinant adenosine A2a receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Mus musculus)
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
Affinity DataKi: 1.00E+4nMAssay Description:Displacement of [3H]2-[p-(2-carboxyethyl)phenyl-ethylamino]-5'-N-ethylcarboxamidoadenosine from mouse recombinant adenosine A2A receptor expressed in...More data for this Ligand-Target Pair
