Found 16 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a' and Ligand = 'BDBM50207816' 
3D Structure (crystal)Affinity DataKi: 1nMAssay Description:Displacement of [3H]HZ241385 from human A2AAR expressed in HeLa cell membrane incubated for 30 mins by microbeta trilux scintillation counter analysi...More data for this Ligand-Target Pair
Affinity DataKi: 5.80nMAssay Description:Antagonist activity at human adenosine A2A receptor assessed as cAMP level by cell based assayMore data for this Ligand-Target Pair
Affinity DataKi: 7.90nMAssay Description:Binding affinity for HA-tagged wild type human Adenosine A2A receptor (WT) using [3H]CGS-21680 as radioligand expressed in COS-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Binding affinity for HA-tagged mutant human Adenosine A2A receptor (H250N) using [3H]-CGS-21,680 as radioligand expressed in COS-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 18.4nMAssay Description:Antagonist activity against recombinant human adenosine A2A receptor expressed in HEK-293 cells in presence of [125I]-iodo-ZM241385 radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 25.1nMAssay Description:Displacement of [3H]ZM241385 from stabilized human adenosine receptor A2a expressed in HEK293 cells followed by receptor capturing on Biocore chips b...More data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Binding affinity for HA-tagged mutant human Adenosine A2A receptor (V84L), using [3H]CGS-21680 as radioligand expressed in COS-7 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Displacement of MRS5346 from C-terminal 10xHis and 1D4-tagged C-terminal-truncated human A2A adenosine receptor (1 to 316 residues) expressed in Pich...More data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Ability to displace the specific binding of [3H]-CGS- to adenosine A2A receptor form bovine brain striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Displacement of [3H]ZM-241385 binding in adenosine A2A receptor of rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Antagonist activity against adenosine A2A receptor in rat striatal membrane in presence of [3H]-CGS-21,680 radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Displacement of [3H]-CGS- 21680 from adenosine A2a receptors of rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Binding affinity towards rat Adenosine A2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Displacement of [3H] 4-2-7-amino-2-2-furyl1,2,4 triazolo2,3-a1,3,5triazin-5-ylaminoethyl phenol from human adenosine A2A receptor expressed in human ...More data for this Ligand-Target Pair
