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Found 4 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A2a' and Ligand = 'BDBM50214974'
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50214974((2R,3R,4S)-2-(2-chloro-6-(3-iodobenzylamino)-9H-pu...)
Affinity DataKi:  341nMAssay Description:Displacement of [3H]CGS21680 from human adenosine A2A receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50214974((2R,3R,4S)-2-(2-chloro-6-(3-iodobenzylamino)-9H-pu...)
Affinity DataKi:  341nMAssay Description:Displacement of [3H]CGS21680 from human A2A adenosine receptor expressed in HEK293 cell membranes after 60 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50214974((2R,3R,4S)-2-(2-chloro-6-(3-iodobenzylamino)-9H-pu...)
Affinity DataKi:  341nMAssay Description:Displacement of [3H]CGS 21680 from human adenosine A2A receptor expressed HEK293 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50214974((2R,3R,4S)-2-(2-chloro-6-(3-iodobenzylamino)-9H-pu...)
Affinity DataKi:  341nMAssay Description:Displacement of [3H]CGS21680 from human recombinant adenosine A2a receptor expressed in HEK293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed